DK138327B - Analogifremgangsmåde til fremstilling af pyrido(1,2a)pyrimidinderivater. - Google Patents

Analogifremgangsmåde til fremstilling af pyrido(1,2a)pyrimidinderivater.

Info

Publication number
DK138327B
DK138327B DK174074AA DK174074A DK138327B DK 138327 B DK138327 B DK 138327B DK 174074A A DK174074A A DK 174074AA DK 174074 A DK174074 A DK 174074A DK 138327 B DK138327 B DK 138327B
Authority
DK
Denmark
Prior art keywords
pyrido
preparation
pyrimidine derivatives
analogous process
analogous
Prior art date
Application number
DK174074AA
Other languages
Danish (da)
English (en)
Other versions
DK138327C (pl
Inventor
Zoltan Meszaros
Jozsef Knoll
Istvan Hermecz
Lelle Vasvari
Agnes Horvath
Original Assignee
Chinoin Gyogyszer Es Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer Es Vegyeszet filed Critical Chinoin Gyogyszer Es Vegyeszet
Publication of DK138327B publication Critical patent/DK138327B/da
Application granted granted Critical
Publication of DK138327C publication Critical patent/DK138327C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK174074AA 1973-03-30 1974-03-29 Analogifremgangsmåde til fremstilling af pyrido(1,2a)pyrimidinderivater. DK138327B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HUCI1361A HU168014B (pl) 1973-03-30 1973-03-30

Publications (2)

Publication Number Publication Date
DK138327B true DK138327B (da) 1978-08-14
DK138327C DK138327C (pl) 1979-01-22

Family

ID=10994473

Family Applications (1)

Application Number Title Priority Date Filing Date
DK174074AA DK138327B (da) 1973-03-30 1974-03-29 Analogifremgangsmåde til fremstilling af pyrido(1,2a)pyrimidinderivater.

Country Status (20)

Country Link
JP (1) JPS505396A (pl)
AT (1) AT336624B (pl)
BE (1) BE813021A (pl)
CA (1) CA1032938A (pl)
CH (1) CH605940A5 (pl)
CS (1) CS189872B1 (pl)
DD (1) DD110661A1 (pl)
DE (1) DE2414751A1 (pl)
DK (1) DK138327B (pl)
ES (1) ES424758A1 (pl)
FI (1) FI57949C (pl)
FR (1) FR2223036B1 (pl)
GB (1) GB1454312A (pl)
HU (1) HU168014B (pl)
IL (1) IL44417A (pl)
NL (1) NL7403901A (pl)
NO (1) NO140821C (pl)
PL (1) PL93755B1 (pl)
SE (1) SE418087B (pl)
SU (1) SU566524A3 (pl)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK153150B (da) * 1975-11-27 1988-06-20 Chinoin Gyogyszer Es Vegyeszet Analogifremgangsmaade til fremstilling af 4-oxo-1,6,7,8-tetrahydro-4h-pyridooe1,2aaapyrimidinderivater

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU174693B (hu) * 1976-02-12 1980-03-28 Chinoin Gyogyszer Es Vegyeszet Sposob poluchenija kondensirovannykh proizvodnykh pirimidina
HU174901B (hu) * 1976-06-25 1980-04-28 Chinoin Gyogyszer Es Vegyeszet Sposob poluchenija novykh proizvodnykh pirido/1,2-a/pirimidina
HU178910B (en) * 1977-08-19 1982-07-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 2,3-disubstituted-4-oxo-4h-pyrido/1,2-a/-pyrimidines
HU178496B (en) * 1977-12-29 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 6,7,8,9-tetrahydro-4h-pyrido/1,2-a/pyrimidine derivatives with antiallergic activity
HU179143B (en) * 1977-12-29 1982-08-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 9-hydroxy-groops-containing 6,7-dihydro-pyrido-square bracket-1,2-a-square bracket closed-pyrimidin derivatives and esters thereof
HU185925B (en) * 1977-12-29 1985-04-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing compounds with nitrogen bridge head
HU180701B (en) * 1977-12-29 1983-04-29 Chinoin Gyogyszer Es Vegyeszet Process for preparing pyrido-/1,2-a/pyrimidines containing a carboxylic or ester group on the pirimidimering
AT376675B (de) * 1979-05-08 1984-12-27 Erba Farmitalia Verfahren zum herstellen von neuen substituierten pyrido(1,2-a)pyrimidinen
US4661592A (en) * 1984-06-27 1987-04-28 G. D. Searle & Co. 4H-pyrimido[2,1-a]isoquinolin-4-one derivatives
HU201551B (en) * 1988-02-03 1990-11-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 4-oxo-4h-pyrido(1,2-a)pyrimidine-3-carboxylic acid amide derivatives and pharmaceutical compositions comprising same
JP5419894B2 (ja) * 2008-01-11 2014-02-19 グレンマーク ファーマシューティカルズ, エセ.アー. Trpv3モジュレーターとしての縮合ピリミジン誘導体

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT299212B (de) * 1966-11-02 1972-06-12 Chinoin Gyogyszer Es Vegyeszet Verfahren zur Herstellung von neuen Homopyrimidazol-Derivaten sowie von deren Salzen

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK153150B (da) * 1975-11-27 1988-06-20 Chinoin Gyogyszer Es Vegyeszet Analogifremgangsmaade til fremstilling af 4-oxo-1,6,7,8-tetrahydro-4h-pyridooe1,2aaapyrimidinderivater

Also Published As

Publication number Publication date
CH605940A5 (pl) 1978-10-13
HU168014B (pl) 1976-02-28
FR2223036A1 (pl) 1974-10-25
CS189872B1 (en) 1979-05-31
AT336624B (de) 1977-05-10
SE418087B (sv) 1981-05-04
ES424758A1 (es) 1976-06-16
IL44417A0 (en) 1974-06-30
CA1032938A (en) 1978-06-13
IL44417A (en) 1978-01-31
ATA252674A (de) 1976-09-15
FI57949C (fi) 1980-11-10
DD110661A1 (pl) 1975-01-05
NO741125A (no) 1974-10-01
PL93755B1 (en) 1977-06-30
DK138327C (pl) 1979-01-22
AU6670474A (en) 1975-09-18
NL7403901A (pl) 1974-10-02
GB1454312A (en) 1976-11-03
DE2414751A1 (de) 1974-10-10
BE813021A (fr) 1974-07-15
NO140821B (no) 1979-08-13
NO140821C (no) 1979-11-21
FR2223036B1 (pl) 1977-05-06
JPS505396A (pl) 1975-01-21
FI57949B (fi) 1980-07-31
SU566524A3 (ru) 1977-07-25

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