NO140821C - Analogifremgangsmaate ved fremstilling av terapeutisk aktive pyrido-pyrimidin-derivater - Google Patents

Analogifremgangsmaate ved fremstilling av terapeutisk aktive pyrido-pyrimidin-derivater

Info

Publication number
NO140821C
NO140821C NO741125A NO741125A NO140821C NO 140821 C NO140821 C NO 140821C NO 741125 A NO741125 A NO 741125A NO 741125 A NO741125 A NO 741125A NO 140821 C NO140821 C NO 140821C
Authority
NO
Norway
Prior art keywords
preparation
therapeutically active
pyrimidine derivatives
analogical procedure
active pyrido
Prior art date
Application number
NO741125A
Other languages
English (en)
Norwegian (no)
Other versions
NO741125A (no
NO140821B (no
Inventor
Zoltan Meszaros
Jozsef Knoll
Istvan Hermecz
Lelle Vasvari
Agnes Horvath
Original Assignee
Chinoin Gyogyszer Es Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer Es Vegyeszet filed Critical Chinoin Gyogyszer Es Vegyeszet
Publication of NO741125A publication Critical patent/NO741125A/no
Publication of NO140821B publication Critical patent/NO140821B/no
Publication of NO140821C publication Critical patent/NO140821C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO741125A 1973-03-30 1974-03-29 Analogifremgangsmaate ved fremstilling av terapeutisk aktive pyrido-pyrimidin-derivater NO140821C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HUCI1361A HU168014B (pl) 1973-03-30 1973-03-30

Publications (3)

Publication Number Publication Date
NO741125A NO741125A (no) 1974-10-01
NO140821B NO140821B (no) 1979-08-13
NO140821C true NO140821C (no) 1979-11-21

Family

ID=10994473

Family Applications (1)

Application Number Title Priority Date Filing Date
NO741125A NO140821C (no) 1973-03-30 1974-03-29 Analogifremgangsmaate ved fremstilling av terapeutisk aktive pyrido-pyrimidin-derivater

Country Status (20)

Country Link
JP (1) JPS505396A (pl)
AT (1) AT336624B (pl)
BE (1) BE813021A (pl)
CA (1) CA1032938A (pl)
CH (1) CH605940A5 (pl)
CS (1) CS189872B1 (pl)
DD (1) DD110661A1 (pl)
DE (1) DE2414751A1 (pl)
DK (1) DK138327B (pl)
ES (1) ES424758A1 (pl)
FI (1) FI57949C (pl)
FR (1) FR2223036B1 (pl)
GB (1) GB1454312A (pl)
HU (1) HU168014B (pl)
IL (1) IL44417A (pl)
NL (1) NL7403901A (pl)
NO (1) NO140821C (pl)
PL (1) PL93755B1 (pl)
SE (1) SE418087B (pl)
SU (1) SU566524A3 (pl)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU173438B (hu) * 1975-11-27 1979-05-28 Chinoin Gyogyszer Es Vegyeszet Sposob poluchenija novykh proizvodnykh 4-okso-1,6,7,8-/tetragidro-4h-pirido/1,2/pirimidina s zaderzhivajuhhejj vozgoranie aktivnot'ju i protivosvertivajuhhem effektom
HU174693B (hu) * 1976-02-12 1980-03-28 Chinoin Gyogyszer Es Vegyeszet Sposob poluchenija kondensirovannykh proizvodnykh pirimidina
HU174901B (hu) * 1976-06-25 1980-04-28 Chinoin Gyogyszer Es Vegyeszet Sposob poluchenija novykh proizvodnykh pirido/1,2-a/pirimidina
HU178910B (en) * 1977-08-19 1982-07-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 2,3-disubstituted-4-oxo-4h-pyrido/1,2-a/-pyrimidines
HU178496B (en) * 1977-12-29 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing 6,7,8,9-tetrahydro-4h-pyrido/1,2-a/pyrimidine derivatives with antiallergic activity
HU179143B (en) * 1977-12-29 1982-08-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 9-hydroxy-groops-containing 6,7-dihydro-pyrido-square bracket-1,2-a-square bracket closed-pyrimidin derivatives and esters thereof
HU185925B (en) * 1977-12-29 1985-04-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing compounds with nitrogen bridge head
HU180701B (en) * 1977-12-29 1983-04-29 Chinoin Gyogyszer Es Vegyeszet Process for preparing pyrido-/1,2-a/pyrimidines containing a carboxylic or ester group on the pirimidimering
AT376675B (de) * 1979-05-08 1984-12-27 Erba Farmitalia Verfahren zum herstellen von neuen substituierten pyrido(1,2-a)pyrimidinen
US4661592A (en) * 1984-06-27 1987-04-28 G. D. Searle & Co. 4H-pyrimido[2,1-a]isoquinolin-4-one derivatives
HU201551B (en) * 1988-02-03 1990-11-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 4-oxo-4h-pyrido(1,2-a)pyrimidine-3-carboxylic acid amide derivatives and pharmaceutical compositions comprising same
JP5419894B2 (ja) * 2008-01-11 2014-02-19 グレンマーク ファーマシューティカルズ, エセ.アー. Trpv3モジュレーターとしての縮合ピリミジン誘導体

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT299212B (de) * 1966-11-02 1972-06-12 Chinoin Gyogyszer Es Vegyeszet Verfahren zur Herstellung von neuen Homopyrimidazol-Derivaten sowie von deren Salzen

Also Published As

Publication number Publication date
CH605940A5 (pl) 1978-10-13
HU168014B (pl) 1976-02-28
FR2223036A1 (pl) 1974-10-25
CS189872B1 (en) 1979-05-31
AT336624B (de) 1977-05-10
SE418087B (sv) 1981-05-04
ES424758A1 (es) 1976-06-16
IL44417A0 (en) 1974-06-30
CA1032938A (en) 1978-06-13
IL44417A (en) 1978-01-31
ATA252674A (de) 1976-09-15
FI57949C (fi) 1980-11-10
DD110661A1 (pl) 1975-01-05
NO741125A (no) 1974-10-01
PL93755B1 (en) 1977-06-30
DK138327C (pl) 1979-01-22
AU6670474A (en) 1975-09-18
DK138327B (da) 1978-08-14
NL7403901A (pl) 1974-10-02
GB1454312A (en) 1976-11-03
DE2414751A1 (de) 1974-10-10
BE813021A (fr) 1974-07-15
NO140821B (no) 1979-08-13
FR2223036B1 (pl) 1977-05-06
JPS505396A (pl) 1975-01-21
FI57949B (fi) 1980-07-31
SU566524A3 (ru) 1977-07-25

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