DK140498B - Analogifremgangsmåde til fremstilling af 3-substituerede 1,2-benzisoxazolderivater. - Google Patents

Analogifremgangsmåde til fremstilling af 3-substituerede 1,2-benzisoxazolderivater.

Info

Publication number
DK140498B
DK140498B DK145373AA DK145373A DK140498B DK 140498 B DK140498 B DK 140498B DK 145373A A DK145373A A DK 145373AA DK 145373 A DK145373 A DK 145373A DK 140498 B DK140498 B DK 140498B
Authority
DK
Denmark
Prior art keywords
substituted
preparation
analogous process
benzisoxazole derivatives
benzisoxazole
Prior art date
Application number
DK145373AA
Other languages
English (en)
Other versions
DK140498C (da
Inventor
Haruki Nishimura
Masanao Shimizu
Hitoshi Uno
Tetsuo Hirooka
Yoshinobu Masuda
Mikio Kurokawa
Original Assignee
Dainippon Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP2786672A external-priority patent/JPS5616154B2/ja
Priority claimed from JP2786572A external-priority patent/JPS5545545B2/ja
Application filed by Dainippon Pharmaceutical Co filed Critical Dainippon Pharmaceutical Co
Publication of DK140498B publication Critical patent/DK140498B/da
Application granted granted Critical
Publication of DK140498C publication Critical patent/DK140498C/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK145373AA 1972-03-17 1973-03-16 Analogifremgangsmåde til fremstilling af 3-substituerede 1,2-benzisoxazolderivater. DK140498B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2786672A JPS5616154B2 (da) 1972-03-17 1972-03-17
JP2786572A JPS5545545B2 (da) 1972-03-17 1972-03-17

Publications (2)

Publication Number Publication Date
DK140498B true DK140498B (da) 1979-09-17
DK140498C DK140498C (da) 1980-03-17

Family

ID=26365855

Family Applications (1)

Application Number Title Priority Date Filing Date
DK145373AA DK140498B (da) 1972-03-17 1973-03-16 Analogifremgangsmåde til fremstilling af 3-substituerede 1,2-benzisoxazolderivater.

Country Status (10)

Country Link
US (1) US3948928A (da)
AU (1) AU466970B2 (da)
CA (1) CA1025857A (da)
CH (1) CH577984A5 (da)
DK (1) DK140498B (da)
ES (1) ES412813A1 (da)
FR (1) FR2181831B1 (da)
GB (1) GB1416071A (da)
NL (1) NL168833C (da)
SE (1) SE381047B (da)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4673746A (en) * 1978-10-06 1987-06-16 Hoechst-Roussel Pharmaceuticals, Inc. 1,2-benzisoxazoloxyacetic acids and related compounds
US4728662A (en) * 1977-11-21 1988-03-01 Hoechst-Roussel Pharmaceuticals Inc. 1,2-benzisoxazoloxyacetic acids and related compounds
US4609658A (en) * 1982-04-09 1986-09-02 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted) piperazines useful for reducing blood pressure
US4536578A (en) * 1982-04-09 1985-08-20 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted)piperazines
US4610988A (en) * 1982-04-09 1986-09-09 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted)piperazines useful for alleviating pain
JPS58201770A (ja) * 1982-05-18 1983-11-24 Dainippon Pharmaceut Co Ltd α−置換−１，２−ベンズイソキサゾ−ル−３−酢酸エステル類並びにその酸付加塩類及び第４級アンモニウム塩類
EP1846401B1 (en) * 2005-02-04 2008-06-18 CTG Pharma S.r.l. New 4-aminoquinoline derivatives as antimalarials
EP2559690B1 (en) 2005-05-10 2016-03-30 Incyte Holdings Corporation Modulators of indoleamine 2,3-dioxygenase and methods of using the same
WO2007075598A2 (en) * 2005-12-20 2007-07-05 Incyte Corporation N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase
WO2007081335A1 (en) * 2006-01-12 2007-07-19 Merck & Co., Inc. Therapeutic compounds for treating dyslipidemic conditions
CL2007002650A1 (es) 2006-09-19 2008-02-08 Incyte Corp Compuestos derivados de heterociclo n-hidroxiamino; composicion farmaceutica, util para tratar cancer, infecciones virales y desordenes neurodegenerativos entre otras.
EP2064207B1 (en) * 2006-09-19 2013-11-06 Incyte Corporation N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase
US20080146624A1 (en) * 2006-09-19 2008-06-19 Incyte Corporation Amidines as modulators of indoleamine 2,3-dioxygenase
WO2008058178A1 (en) * 2006-11-08 2008-05-15 Incyte Corporation N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase
WO2008142134A1 (en) * 2007-05-24 2008-11-27 Neurosearch A/S Benzisoxazole derivatives as potassium channel modulators for the treatment of e.g. respiratory diseases, epilepsy and convulsions
KR101927291B1 (ko) 2008-07-08 2018-12-10 인사이트 홀딩스 코포레이션 인돌아민 ２,３-디옥시게나아제의 억제제로서의 １,２,５-옥사디아졸
DK3066085T3 (da) 2013-11-08 2020-06-02 Incyte Holdings Corp Fremgangsmåde til syntesen af en indolamin-2,3-dioxygenaseinhibitor

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1670497C3 (de) * 1967-06-06 1973-12-20 Chinoin Gyogyszer- Es Vegyeszeti Termekek Gyara Rt, Budapest Isochinohnderivate und Verfahren zu deren Herstellung

Also Published As

Publication number Publication date
CH577984A5 (da) 1976-07-30
US3948928A (en) 1976-04-06
NL168833C (nl) 1982-05-17
ES412813A1 (es) 1976-07-01
CA1025857A (en) 1978-02-07
NL7303682A (da) 1973-09-19
AU5347973A (en) 1974-09-19
DK140498C (da) 1980-03-17
GB1416071A (en) 1975-12-03
AU466970B2 (en) 1975-11-13
SE381047B (sv) 1975-11-24
FR2181831A1 (da) 1973-12-07
NL168833B (nl) 1981-12-16
FR2181831B1 (da) 1975-10-10

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