NL7303682A - - Google Patents

Info

Publication number
NL7303682A
NL7303682A NL7303682A NL7303682A NL7303682A NL 7303682 A NL7303682 A NL 7303682A NL 7303682 A NL7303682 A NL 7303682A NL 7303682 A NL7303682 A NL 7303682A NL 7303682 A NL7303682 A NL 7303682A
Authority
NL
Netherlands
Application number
NL7303682A
Other versions
NL168833C (nl
NL168833B (nl
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP2786672A external-priority patent/JPS5616154B2/ja
Priority claimed from JP2786572A external-priority patent/JPS5545545B2/ja
Application filed filed Critical
Publication of NL7303682A publication Critical patent/NL7303682A/xx
Publication of NL168833B publication Critical patent/NL168833B/xx
Application granted granted Critical
Publication of NL168833C publication Critical patent/NL168833C/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D261/00Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/20Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NLAANVRAGE7303682,A 1972-03-17 1973-03-16 Werkwijze voor het bereiden of vervaardigen van een geneesmiddel met antidepressieve werking en werkwijze voor het bereiden van een isoxazoolverbinding, die voor gebruik bij voornoemde werkwijze geschikt is. NL168833C (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2786672A JPS5616154B2 (da) 1972-03-17 1972-03-17
JP2786572A JPS5545545B2 (da) 1972-03-17 1972-03-17

Publications (3)

Publication Number Publication Date
NL7303682A true NL7303682A (da) 1973-09-19
NL168833B NL168833B (nl) 1981-12-16
NL168833C NL168833C (nl) 1982-05-17

Family

ID=26365855

Family Applications (1)

Application Number Title Priority Date Filing Date
NLAANVRAGE7303682,A NL168833C (nl) 1972-03-17 1973-03-16 Werkwijze voor het bereiden of vervaardigen van een geneesmiddel met antidepressieve werking en werkwijze voor het bereiden van een isoxazoolverbinding, die voor gebruik bij voornoemde werkwijze geschikt is.

Country Status (10)

Country Link
US (1) US3948928A (da)
AU (1) AU466970B2 (da)
CA (1) CA1025857A (da)
CH (1) CH577984A5 (da)
DK (1) DK140498B (da)
ES (1) ES412813A1 (da)
FR (1) FR2181831B1 (da)
GB (1) GB1416071A (da)
NL (1) NL168833C (da)
SE (1) SE381047B (da)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4673746A (en) * 1978-10-06 1987-06-16 Hoechst-Roussel Pharmaceuticals, Inc. 1,2-benzisoxazoloxyacetic acids and related compounds
US4728662A (en) * 1977-11-21 1988-03-01 Hoechst-Roussel Pharmaceuticals Inc. 1,2-benzisoxazoloxyacetic acids and related compounds
US4609658A (en) * 1982-04-09 1986-09-02 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted) piperazines useful for reducing blood pressure
US4536578A (en) * 1982-04-09 1985-08-20 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted)piperazines
US4610988A (en) * 1982-04-09 1986-09-09 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted)piperazines useful for alleviating pain
JPS58201770A (ja) * 1982-05-18 1983-11-24 Dainippon Pharmaceut Co Ltd α−置換−1,2−ベンズイソキサゾ−ル−3−酢酸エステル類並びにその酸付加塩類及び第4級アンモニウム塩類
EP1846401B1 (en) * 2005-02-04 2008-06-18 CTG Pharma S.r.l. New 4-aminoquinoline derivatives as antimalarials
EP2559690B1 (en) 2005-05-10 2016-03-30 Incyte Holdings Corporation Modulators of indoleamine 2,3-dioxygenase and methods of using the same
WO2007075598A2 (en) * 2005-12-20 2007-07-05 Incyte Corporation N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase
WO2007081335A1 (en) * 2006-01-12 2007-07-19 Merck & Co., Inc. Therapeutic compounds for treating dyslipidemic conditions
CL2007002650A1 (es) 2006-09-19 2008-02-08 Incyte Corp Compuestos derivados de heterociclo n-hidroxiamino; composicion farmaceutica, util para tratar cancer, infecciones virales y desordenes neurodegenerativos entre otras.
EP2064207B1 (en) * 2006-09-19 2013-11-06 Incyte Corporation N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase
US20080146624A1 (en) * 2006-09-19 2008-06-19 Incyte Corporation Amidines as modulators of indoleamine 2,3-dioxygenase
WO2008058178A1 (en) * 2006-11-08 2008-05-15 Incyte Corporation N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase
WO2008142134A1 (en) * 2007-05-24 2008-11-27 Neurosearch A/S Benzisoxazole derivatives as potassium channel modulators for the treatment of e.g. respiratory diseases, epilepsy and convulsions
KR101927291B1 (ko) 2008-07-08 2018-12-10 인사이트 홀딩스 코포레이션 인돌아민 2,3-디옥시게나아제의 억제제로서의 1,2,5-옥사디아졸
DK3066085T3 (da) 2013-11-08 2020-06-02 Incyte Holdings Corp Fremgangsmåde til syntesen af en indolamin-2,3-dioxygenaseinhibitor

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1670497C3 (de) * 1967-06-06 1973-12-20 Chinoin Gyogyszer- Es Vegyeszeti Termekek Gyara Rt, Budapest Isochinohnderivate und Verfahren zu deren Herstellung

Also Published As

Publication number Publication date
CH577984A5 (da) 1976-07-30
US3948928A (en) 1976-04-06
NL168833C (nl) 1982-05-17
ES412813A1 (es) 1976-07-01
CA1025857A (en) 1978-02-07
AU5347973A (en) 1974-09-19
DK140498C (da) 1980-03-17
GB1416071A (en) 1975-12-03
AU466970B2 (en) 1975-11-13
SE381047B (sv) 1975-11-24
FR2181831A1 (da) 1973-12-07
DK140498B (da) 1979-09-17
NL168833B (nl) 1981-12-16
FR2181831B1 (da) 1975-10-10

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Legal Events

Date Code Title Description
V1 Lapsed because of non-payment of the annual fee