CH577984A5 - - Google Patents

Info

Publication number
CH577984A5
CH577984A5 CH389073A CH389073A CH577984A5 CH 577984 A5 CH577984 A5 CH 577984A5 CH 389073 A CH389073 A CH 389073A CH 389073 A CH389073 A CH 389073A CH 577984 A5 CH577984 A5 CH 577984A5
Authority
CH
Switzerland
Application number
CH389073A
Original Assignee
Dainippon Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP2786572A external-priority patent/JPS5545545B2/ja
Priority claimed from JP2786672A external-priority patent/JPS5616154B2/ja
Application filed by Dainippon Pharmaceutical Co filed Critical Dainippon Pharmaceutical Co
Publication of CH577984A5 publication Critical patent/CH577984A5/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D261/00Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/20Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CH389073A 1972-03-17 1973-03-16 CH577984A5 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2786572A JPS5545545B2 (da) 1972-03-17 1972-03-17
JP2786672A JPS5616154B2 (da) 1972-03-17 1972-03-17

Publications (1)

Publication Number Publication Date
CH577984A5 true CH577984A5 (da) 1976-07-30

Family

ID=26365855

Family Applications (1)

Application Number Title Priority Date Filing Date
CH389073A CH577984A5 (da) 1972-03-17 1973-03-16

Country Status (10)

Country Link
US (1) US3948928A (da)
AU (1) AU466970B2 (da)
CA (1) CA1025857A (da)
CH (1) CH577984A5 (da)
DK (1) DK140498B (da)
ES (1) ES412813A1 (da)
FR (1) FR2181831B1 (da)
GB (1) GB1416071A (da)
NL (1) NL168833C (da)
SE (1) SE381047B (da)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4673746A (en) * 1978-10-06 1987-06-16 Hoechst-Roussel Pharmaceuticals, Inc. 1,2-benzisoxazoloxyacetic acids and related compounds
US4728662A (en) * 1977-11-21 1988-03-01 Hoechst-Roussel Pharmaceuticals Inc. 1,2-benzisoxazoloxyacetic acids and related compounds
US4610988A (en) * 1982-04-09 1986-09-09 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted)piperazines useful for alleviating pain
US4536578A (en) * 1982-04-09 1985-08-20 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted)piperazines
US4609658A (en) * 1982-04-09 1986-09-02 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted) piperazines useful for reducing blood pressure
JPS58201770A (ja) * 1982-05-18 1983-11-24 Dainippon Pharmaceut Co Ltd α−置換−1,2−ベンズイソキサゾ−ル−3−酢酸エステル類並びにその酸付加塩類及び第4級アンモニウム塩類
DE602006001511D1 (de) * 2005-02-04 2008-07-31 Ctg Pharma S R L Neue 4-aminochinolinderivate als antimalariamittel
DK2559690T3 (da) 2005-05-10 2016-04-25 Incyte Holdings Corp Modulatorer af indolamin-2,3-dioxygenase og fremgangsmåder til anvendelse deraf
EP1971583B1 (en) * 2005-12-20 2015-03-25 Incyte Corporation N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase
WO2007081335A1 (en) * 2006-01-12 2007-07-19 Merck & Co., Inc. Therapeutic compounds for treating dyslipidemic conditions
WO2008036642A2 (en) * 2006-09-19 2008-03-27 Incyte Corporation N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase
US20080146624A1 (en) * 2006-09-19 2008-06-19 Incyte Corporation Amidines as modulators of indoleamine 2,3-dioxygenase
CL2007002650A1 (es) 2006-09-19 2008-02-08 Incyte Corp Compuestos derivados de heterociclo n-hidroxiamino; composicion farmaceutica, util para tratar cancer, infecciones virales y desordenes neurodegenerativos entre otras.
US20080182882A1 (en) * 2006-11-08 2008-07-31 Incyte Corporation N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase
EP2152679A1 (en) * 2007-05-24 2010-02-17 NeuroSearch A/S Benzisoxazole derivatives as potassium channel modulators for the treatment of e.g. respiratory diseases, epilepsy and convulsions
BRPI0915692B8 (pt) 2008-07-08 2021-05-25 Incyte Corp compostos derivados de 1,2,5-oxadiazóis, sua forma sólida, sua composição, bem como seus usos
SG10201803874PA (en) 2013-11-08 2018-07-30 Incyte Holdings Corp Process for the synthesis of an indoleamine 2,3-dioxygenase inhibitor

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1670497C3 (de) * 1967-06-06 1973-12-20 Chinoin Gyogyszer- Es Vegyeszeti Termekek Gyara Rt, Budapest Isochinohnderivate und Verfahren zu deren Herstellung

Also Published As

Publication number Publication date
AU5347973A (en) 1974-09-19
NL168833B (nl) 1981-12-16
CA1025857A (en) 1978-02-07
FR2181831B1 (da) 1975-10-10
NL168833C (nl) 1982-05-17
AU466970B2 (en) 1975-11-13
DK140498B (da) 1979-09-17
ES412813A1 (es) 1976-07-01
NL7303682A (da) 1973-09-19
GB1416071A (en) 1975-12-03
FR2181831A1 (da) 1973-12-07
SE381047B (sv) 1975-11-24
DK140498C (da) 1980-03-17
US3948928A (en) 1976-04-06

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Legal Events

Date Code Title Description
PL Patent ceased