FR2181831B1 - - Google Patents

Info

Publication number
FR2181831B1
FR2181831B1 FR7309763A FR7309763A FR2181831B1 FR 2181831 B1 FR2181831 B1 FR 2181831B1 FR 7309763 A FR7309763 A FR 7309763A FR 7309763 A FR7309763 A FR 7309763A FR 2181831 B1 FR2181831 B1 FR 2181831B1
Authority
FR
France
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
FR7309763A
Other versions
FR2181831A1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Dainippon Pharmaceutical Co Ltd
Original Assignee
Dainippon Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP2786672A external-priority patent/JPS5616154B2/ja
Priority claimed from JP2786572A external-priority patent/JPS5545545B2/ja
Application filed by Dainippon Pharmaceutical Co Ltd filed Critical Dainippon Pharmaceutical Co Ltd
Publication of FR2181831A1 publication Critical patent/FR2181831A1/fr
Application granted granted Critical
Publication of FR2181831B1 publication Critical patent/FR2181831B1/fr
Expired legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D261/00Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/20Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR7309763A 1972-03-17 1973-03-19 Expired FR2181831B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2786672A JPS5616154B2 (fr) 1972-03-17 1972-03-17
JP2786572A JPS5545545B2 (fr) 1972-03-17 1972-03-17

Publications (2)

Publication Number Publication Date
FR2181831A1 FR2181831A1 (fr) 1973-12-07
FR2181831B1 true FR2181831B1 (fr) 1975-10-10

Family

ID=26365855

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7309763A Expired FR2181831B1 (fr) 1972-03-17 1973-03-19

Country Status (10)

Country Link
US (1) US3948928A (fr)
AU (1) AU466970B2 (fr)
CA (1) CA1025857A (fr)
CH (1) CH577984A5 (fr)
DK (1) DK140498B (fr)
ES (1) ES412813A1 (fr)
FR (1) FR2181831B1 (fr)
GB (1) GB1416071A (fr)
NL (1) NL168833C (fr)
SE (1) SE381047B (fr)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4673746A (en) * 1978-10-06 1987-06-16 Hoechst-Roussel Pharmaceuticals, Inc. 1,2-benzisoxazoloxyacetic acids and related compounds
US4728662A (en) * 1977-11-21 1988-03-01 Hoechst-Roussel Pharmaceuticals Inc. 1,2-benzisoxazoloxyacetic acids and related compounds
US4609658A (en) * 1982-04-09 1986-09-02 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted) piperazines useful for reducing blood pressure
US4536578A (en) * 1982-04-09 1985-08-20 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-Fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted)piperazines
US4610988A (en) * 1982-04-09 1986-09-09 Hoechst-Roussel Pharmaceuticals Inc. 1-[3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl]-4-(substituted)piperazines useful for alleviating pain
JPS58201770A (ja) * 1982-05-18 1983-11-24 Dainippon Pharmaceut Co Ltd α−置換−1,2−ベンズイソキサゾ−ル−3−酢酸エステル類並びにその酸付加塩類及び第4級アンモニウム塩類
EP1846401B1 (fr) * 2005-02-04 2008-06-18 CTG Pharma S.r.l. Nouveaux dérivés de 4-aminoquinoléine comme composés antimalaria
EP2559690B1 (fr) 2005-05-10 2016-03-30 Incyte Holdings Corporation Modulateurs de l'indolamine 2,3-dioxygenase et leurs procedes d'utilisation
WO2007075598A2 (fr) * 2005-12-20 2007-07-05 Incyte Corporation N-hydroxyamidinoheterocycles en tant que modulateurs d'indoleamine 2,3-dioxygenase
WO2007081335A1 (fr) * 2006-01-12 2007-07-19 Merck & Co., Inc. Composes therapeutiques pour traiter des troubles dyslipidemiques
CL2007002650A1 (es) 2006-09-19 2008-02-08 Incyte Corp Compuestos derivados de heterociclo n-hidroxiamino; composicion farmaceutica, util para tratar cancer, infecciones virales y desordenes neurodegenerativos entre otras.
EP2064207B1 (fr) * 2006-09-19 2013-11-06 Incyte Corporation N-hydroxyamidinohétérocycles en tant que modulateurs d'indoléamine 2,3-dioxygénase
US20080146624A1 (en) * 2006-09-19 2008-06-19 Incyte Corporation Amidines as modulators of indoleamine 2,3-dioxygenase
WO2008058178A1 (fr) * 2006-11-08 2008-05-15 Incyte Corporation N-hydroxyamidinohétérocycles utilisés comme modulateurs de l'indoleamine 2,3-dioxygénase
WO2008142134A1 (fr) * 2007-05-24 2008-11-27 Neurosearch A/S Nouveaux dérivés de benzisoxazole utiles comme modulateurs des canaux potassiques
KR101927291B1 (ko) 2008-07-08 2018-12-10 인사이트 홀딩스 코포레이션 인돌아민 2,3-디옥시게나아제의 억제제로서의 1,2,5-옥사디아졸
DK3066085T3 (da) 2013-11-08 2020-06-02 Incyte Holdings Corp Fremgangsmåde til syntesen af en indolamin-2,3-dioxygenaseinhibitor

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1670497C3 (de) * 1967-06-06 1973-12-20 Chinoin Gyogyszer- Es Vegyeszeti Termekek Gyara Rt, Budapest Isochinohnderivate und Verfahren zu deren Herstellung

Also Published As

Publication number Publication date
CH577984A5 (fr) 1976-07-30
US3948928A (en) 1976-04-06
NL168833C (nl) 1982-05-17
ES412813A1 (es) 1976-07-01
CA1025857A (fr) 1978-02-07
NL7303682A (fr) 1973-09-19
AU5347973A (en) 1974-09-19
DK140498C (fr) 1980-03-17
GB1416071A (en) 1975-12-03
AU466970B2 (en) 1975-11-13
SE381047B (sv) 1975-11-24
FR2181831A1 (fr) 1973-12-07
DK140498B (da) 1979-09-17
NL168833B (nl) 1981-12-16

Similar Documents

Publication Publication Date Title
FR2181831B1 (fr)
JPS5244885Y2 (fr)
JPS57249B2 (fr)
JPS4888240U (fr)
JPS5316835Y2 (fr)
JPS5218888Y2 (fr)
JPS4930813A (fr)
JPS4883286U (fr)
CS150342B1 (fr)
CH575879A5 (fr)
CH569108A5 (fr)
CH607068A5 (fr)
CH595385A5 (fr)
CH591857A5 (fr)
CH586498A5 (fr)
CH581621A5 (fr)
CH579551A5 (fr)
CH579257A5 (fr)
CH579003A5 (fr)
CH578464A5 (fr)
CH577134A5 (fr)
CH577057B5 (fr)
CH569165A5 (fr)
CH573880A5 (fr)
CH573646A5 (fr)

Legal Events

Date Code Title Description
ST Notification of lapse