DK134991B - Analogifremgangsmåde til fremstilling af (4'-(3''-indolyl)-piperidino)-alkylarylketoner eller salte deraf. - Google Patents

Analogifremgangsmåde til fremstilling af (4'-(3''-indolyl)-piperidino)-alkylarylketoner eller salte deraf.

Info

Publication number
DK134991B
DK134991B DK414673AA DK414673A DK134991B DK 134991 B DK134991 B DK 134991B DK 414673A A DK414673A A DK 414673AA DK 414673 A DK414673 A DK 414673A DK 134991 B DK134991 B DK 134991B
Authority
DK
Denmark
Prior art keywords
piperidino
indolyl
salts
preparation
analogous process
Prior art date
Application number
DK414673AA
Other languages
Danish (da)
English (en)
Other versions
DK134991C (ja
Inventor
Pierre Henri Derible
Jean-Paul Lavaux
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of DK134991B publication Critical patent/DK134991B/da
Application granted granted Critical
Publication of DK134991C publication Critical patent/DK134991C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Indole Compounds (AREA)
DK414673AA 1972-07-28 1973-07-27 Analogifremgangsmåde til fremstilling af (4'-(3''-indolyl)-piperidino)-alkylarylketoner eller salte deraf. DK134991B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7227263A FR2193584B1 (ja) 1972-07-28 1972-07-28

Publications (2)

Publication Number Publication Date
DK134991B true DK134991B (da) 1977-02-21
DK134991C DK134991C (ja) 1977-09-26

Family

ID=9102514

Family Applications (1)

Application Number Title Priority Date Filing Date
DK414673AA DK134991B (da) 1972-07-28 1973-07-27 Analogifremgangsmåde til fremstilling af (4'-(3''-indolyl)-piperidino)-alkylarylketoner eller salte deraf.

Country Status (15)

Country Link
US (1) US3850938A (ja)
JP (1) JPS562555B2 (ja)
AU (1) AU472530B2 (ja)
BE (1) BE802912A (ja)
CA (1) CA1013748A (ja)
CH (1) CH571500A5 (ja)
DE (1) DE2365967C3 (ja)
DK (1) DK134991B (ja)
ES (1) ES417333A1 (ja)
FR (1) FR2193584B1 (ja)
GB (1) GB1382782A (ja)
IL (1) IL42781A (ja)
NL (1) NL7310268A (ja)
SE (1) SE406589B (ja)
ZA (1) ZA734998B (ja)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2322470A1 (de) * 1973-05-04 1974-11-21 Boehringer Sohn Ingelheim Neue indolyl-piperidino-(bzw. 1,2,5,6tetrahydro-pyridyl-)butyrophenone und verfahren zu ihrer herstellung
IL48508A (en) * 1974-12-09 1979-10-31 Roussel Uclaf Pharmaceutical compositions comprising piperidylindole derivatives
US4046900A (en) * 1975-08-08 1977-09-06 American Hoechst Corporation Benzoylpiperidylalkylindoles
DE2708913A1 (de) * 1976-03-04 1977-09-08 Hoechst Ag Benzoylpiperidyalkyl-indole und verwandte verbindungen
FR2349331A1 (fr) * 1976-04-30 1977-11-25 Roussel Uclaf Nouveaux derives de 2,3 dihydro a/4-(3-indolyl) 1-piperidinyl/methyl 1,4-benzodioxin-2-methanol, un procede pour leur preparation et leur application comme medicaments
FR2362628A1 (fr) * 1976-08-26 1978-03-24 Roussel Uclaf Nouveaux derives du piperidyl-indole et leurs sels, procede de preparation et application a titre de medicaments
FR2420536A1 (fr) * 1978-03-22 1979-10-19 Roussel Uclaf Nouveaux derives de 1,3-dihydro 3-/1-/2-(2,3-dihydro 1,4-benzodioxin-2-yl)2-hydroxyethyl/piperidin-4-yl/2h-indol-2-one, procede pour leur preparation et application comme medicaments
US4166120A (en) * 1978-04-14 1979-08-28 American Hoechst Corporation Analgesic and tranquilizing benzoylpropyl-spiro[dihydrobenzofuran]piperidines and pyrrolidines
FR2444678A2 (fr) * 1978-12-22 1980-07-18 Roussel Uclaf Nouveau procede de preparation de derives du piperidyl-indole et de leurs sels
FR2460947A1 (fr) * 1979-07-13 1981-01-30 Roussel Uclaf Nouveau derives n-substitues du tetrahydropyridinyl-indole, leurs sels, procede de preparation, application a titre de medicaments et compositions les renfermant
IE58370B1 (en) * 1985-04-10 1993-09-08 Lundbeck & Co As H Indole derivatives
US4742057A (en) * 1985-12-05 1988-05-03 Fujisawa Pharmaceutical Co., Ltd. Antiallergic thiazole compounds
DK733788A (da) * 1988-01-14 1989-07-15 Fujisawa Pharmaceutical Co Indolylpiperidinderivater og fremgangsmaade til fremstilling deraf
US5521196A (en) * 1994-10-05 1996-05-28 Eli Lilly And Company 5-HT1F agonists for the treatment of migraine
US5521197A (en) * 1994-12-01 1996-05-28 Eli Lilly And Company 3-<1-alkylenearyl>-4-<1,2,3,6-tetrahydropyridinyl>-and 3-<1-alkylenearyl>-4-piperidinyl-1h-indoles: new 5-HT1F agonists
CN1184425A (zh) * 1995-03-20 1998-06-10 伊莱利利公司 5-取代-3-(1,2,3,6-四氢吡啶-4-基)-和3-(哌啶-4-基)-1h-吲哚:新型5-ht1f激动剂
AR013669A1 (es) * 1997-10-07 2001-01-10 Smithkline Beecham Corp Compuestos y metodos
JP2008076126A (ja) * 2006-09-20 2008-04-03 Oputo System:Kk 測光装置及び測光方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB925429A (en) * 1960-04-01 1963-05-08 Irwin Neisler & Co Indole derivatives
US3462440A (en) * 1965-12-03 1969-08-19 American Home Prod 1,4-bis(2-indol-3-ylethyl)piperidines

Also Published As

Publication number Publication date
ES417333A1 (es) 1976-02-16
SE406589B (sv) 1979-02-19
DE2338283B2 (de) 1977-06-02
DE2365967A1 (de) 1977-02-10
US3850938A (en) 1974-11-26
ZA734998B (en) 1974-09-25
NL7310268A (ja) 1974-01-30
DK134991C (ja) 1977-09-26
IL42781A (en) 1976-07-30
CH571500A5 (ja) 1976-01-15
JPS562555B2 (ja) 1981-01-20
AU5862973A (en) 1975-01-30
JPS4962481A (ja) 1974-06-17
FR2193584B1 (ja) 1975-08-08
DE2365967C3 (de) 1978-08-31
FR2193584A1 (ja) 1974-02-22
BE802912A (fr) 1974-01-28
AU472530B2 (en) 1976-05-27
IL42781A0 (en) 1973-10-25
CA1013748A (fr) 1977-07-12
GB1382782A (en) 1975-02-05
DE2365967B2 (de) 1977-12-22
DE2338283A1 (de) 1974-02-07

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