DK138797B - Analogifremgangsmåde til fremstilling af 1,4-benzodiazepin-derivater eller N-oxider eller salte deraf. - Google Patents

Analogifremgangsmåde til fremstilling af 1,4-benzodiazepin-derivater eller N-oxider eller salte deraf.

Info

Publication number
DK138797B
DK138797B DK487071AA DK487071A DK138797B DK 138797 B DK138797 B DK 138797B DK 487071A A DK487071A A DK 487071AA DK 487071 A DK487071 A DK 487071A DK 138797 B DK138797 B DK 138797B
Authority
DK
Denmark
Prior art keywords
oxides
salts
preparation
benzodiazepine derivatives
analogous process
Prior art date
Application number
DK487071AA
Other languages
English (en)
Other versions
DK138797C (da
Inventor
Roland Jaunin
Joseph Hellerbach
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of DK138797B publication Critical patent/DK138797B/da
Application granted granted Critical
Publication of DK138797C publication Critical patent/DK138797C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
DK487071AA 1970-10-07 1971-10-06 Analogifremgangsmåde til fremstilling af 1,4-benzodiazepin-derivater eller N-oxider eller salte deraf. DK138797B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH1490570A CH538492A (de) 1970-10-07 1970-10-07 Verfahren zur Herstellung von Benzodiazepin-Derivaten

Publications (2)

Publication Number Publication Date
DK138797B true DK138797B (da) 1978-10-30
DK138797C DK138797C (da) 1979-04-09

Family

ID=4404720

Family Applications (1)

Application Number Title Priority Date Filing Date
DK487071AA DK138797B (da) 1970-10-07 1971-10-06 Analogifremgangsmåde til fremstilling af 1,4-benzodiazepin-derivater eller N-oxider eller salte deraf.

Country Status (26)

Country Link
US (1) US3757008A (da)
JP (1) JPS5614667B1 (da)
AT (6) AT317902B (da)
AU (1) AU456526B2 (da)
BE (1) BE773547A (da)
BG (6) BG20111A3 (da)
BR (1) BR7106395D0 (da)
CA (1) CA972754A (da)
CH (1) CH538492A (da)
CS (1) CS174165B2 (da)
DE (1) DE2150075A1 (da)
DK (1) DK138797B (da)
ES (1) ES395762A1 (da)
FR (1) FR2110275B1 (da)
GB (2) GB1357548A (da)
HU (1) HU164060B (da)
IE (1) IE35685B1 (da)
IL (1) IL37645A (da)
MY (1) MY7500047A (da)
NL (1) NL7113023A (da)
PH (1) PH10182A (da)
PL (1) PL82734B1 (da)
RO (1) RO71264A (da)
SE (2) SE388611B (da)
SU (1) SU520917A3 (da)
ZA (1) ZA715787B (da)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT314541B (de) * 1970-10-19 1974-04-10 Sumitomo Chemical Co Verfahren zur Herstellung von neuen Benzodiazepinen und ihren Salzen
HU171033B (hu) * 1974-05-29 1977-10-28 Richter Gedeon Vegyeszet Sposob poluchenija proizvodnykh benzodiazepina
ES2084577T3 (es) * 1986-10-24 1996-05-16 Abbott Lab Ensayo, trazadores, inmunogenos y anticuerpos para benzodiazepinas.
FR2630109B1 (fr) * 1988-04-19 1991-11-29 Synthelabo Derives de ((n-(amino-2 oxo-2 ethyl)methylamino)-2 ethyl)-5 hydroxy-3 (methoxy-4 phenyl)-2 dihydro-2,3 5h-benzothiazepine-1,5 one-4, leur preparation et leur application en therapeutique
FR2653122B1 (fr) * 1989-10-17 1994-04-15 Synthelabo Derives de 5-[2-[[2-amino-2-oxoethyl]methylamino]ethyl]-2,3-dihydro-3-hydroxy-2-(4-methoxyphenyl)-1,5(5h)-benzothiazepine-4-one, leur preparation et leur application en therapeutique.
US5302715A (en) * 1992-04-06 1994-04-12 Biosite Diagnostics, Inc. Benzodiazepine derivatives
HU227319B1 (en) * 2005-12-08 2011-03-28 Egis Gyogyszergyar Nyrt Process for the production of (2-chloro-ethoxy)-acetic acid-n,n-dimethylamide and its intermediate and the novel intermediate

Also Published As

Publication number Publication date
DK138797C (da) 1979-04-09
CS174165B2 (da) 1977-03-31
IE35685B1 (en) 1976-04-28
SE388611B (sv) 1976-10-11
BE773547A (fr) 1972-04-06
AT317900B (de) 1974-09-25
BG20597A3 (da) 1975-12-05
BR7106395D0 (pt) 1973-04-12
ES395762A1 (es) 1974-10-16
AT315859B (de) 1974-06-10
AT315180B (de) 1974-05-10
CH538492A (de) 1973-06-30
GB1357548A (en) 1974-06-26
BG21030A3 (da) 1976-01-20
AU456526B2 (en) 1974-12-19
PL82734B1 (da) 1975-10-31
IL37645A (en) 1974-11-29
ZA715787B (en) 1972-05-31
HU164060B (da) 1973-12-28
SU520917A3 (ru) 1976-07-05
BG20799A3 (da) 1975-12-20
JPS5614667B1 (da) 1981-04-06
PH10182A (en) 1976-09-23
AT317902B (de) 1974-09-25
CA972754A (en) 1975-08-12
IE35685L (en) 1972-04-07
MY7500047A (en) 1975-12-31
AT317901B (de) 1974-09-25
NL7113023A (da) 1972-04-11
AU3296671A (en) 1973-03-08
BG20111A3 (da) 1975-10-30
GB1357547A (en) 1974-06-26
FR2110275A1 (da) 1972-06-02
SE7513089L (sv) 1975-11-20
RO71264A (ro) 1980-07-15
BG19599A3 (da) 1975-06-25
IL37645A0 (en) 1971-11-29
DE2150075A1 (de) 1972-04-13
FR2110275B1 (da) 1974-11-15
BG20598A3 (da) 1975-12-05
AT315860B (de) 1974-06-10
US3757008A (en) 1973-09-04

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