DK120848B - Fremgangsmåde til fremstilling af 1,7-disubstituerede 5-phenyl-1,3-dihydro-2H-1,4-benzodiazepin-2-oner eller syreadditionssalte deraf. - Google Patents

Fremgangsmåde til fremstilling af 1,7-disubstituerede 5-phenyl-1,3-dihydro-2H-1,4-benzodiazepin-2-oner eller syreadditionssalte deraf.

Info

Publication number
DK120848B
DK120848B DK411265AA DK411265A DK120848B DK 120848 B DK120848 B DK 120848B DK 411265A A DK411265A A DK 411265AA DK 411265 A DK411265 A DK 411265A DK 120848 B DK120848 B DK 120848B
Authority
DK
Denmark
Prior art keywords
benzodiazepin
disubstituted
dihydro
ones
phenyl
Prior art date
Application number
DK411265AA
Other languages
English (en)
Inventor
G Archer
L Sternbach
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of DK120848B publication Critical patent/DK120848B/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK411265AA 1964-08-13 1965-08-11 Fremgangsmåde til fremstilling af 1,7-disubstituerede 5-phenyl-1,3-dihydro-2H-1,4-benzodiazepin-2-oner eller syreadditionssalte deraf. DK120848B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US38946964A 1964-08-13 1964-08-13
US474159A US3391138A (en) 1964-08-13 1965-07-22 Certain 1-substituted-benzodiazepin-2-one compounds

Publications (1)

Publication Number Publication Date
DK120848B true DK120848B (da) 1971-07-26

Family

ID=27012718

Family Applications (2)

Application Number Title Priority Date Filing Date
DK411265AA DK120848B (da) 1964-08-13 1965-08-11 Fremgangsmåde til fremstilling af 1,7-disubstituerede 5-phenyl-1,3-dihydro-2H-1,4-benzodiazepin-2-oner eller syreadditionssalte deraf.
DK411365AA DK125554B (da) 1964-08-13 1965-08-11 Analogifremgangsmåde til fremstilling af 1,5,7-trisubstituerede 1,3-dihydro-2H-1,4-benzodiazepin-2-oner eller syreadditionssalte deraf.

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK411365AA DK125554B (da) 1964-08-13 1965-08-11 Analogifremgangsmåde til fremstilling af 1,5,7-trisubstituerede 1,3-dihydro-2H-1,4-benzodiazepin-2-oner eller syreadditionssalte deraf.

Country Status (12)

Country Link
US (1) US3391138A (da)
BE (2) BE668189A (da)
BR (2) BR6571654D0 (da)
CH (1) CH462831A (da)
DE (2) DE1545952C3 (da)
DK (2) DK120848B (da)
FR (1) FR135F (da)
GB (2) GB1102934A (da)
IL (2) IL23999A (da)
NL (2) NL6510539A (da)
NO (2) NO118914B (da)
SE (2) SE310687B (da)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL33961A (en) * 1969-03-13 1973-03-30 Sparamedica Ag Benzodiazepine aminoalkyl carboxylates,their preparation and pharmaceutical compositions containing them
US3989829A (en) * 1969-04-18 1976-11-02 Sumitomo Chemical Company, Limited 1,4-Benzodiazepines
USRE28972E (en) * 1969-07-10 1976-09-21 Boehringer Ingelheim Gmbh 5-Aryl-1H-1,5-benzodiazepine-2,4-diones
US3867372A (en) * 1970-02-03 1975-02-18 Sumitomo Chemical Co Benzodiazepine process
US3691157A (en) * 1970-08-12 1972-09-12 Rodney Ian Fryer Preparation of 7-substituted-1-(2-diethylaminoethyl)-5-(2-halophenyl)-1,3-dihydro-2h-1,4-benzodiazepin-2-ones
DE2166504B2 (de) * 1970-08-31 1980-01-17 Sumitomo Chemical Co., Ltd., Osaka (Japan) 1 -Alkoxyalkoxyalkyl^-halogen-Sphenyl-13-dihydro-2H-l,4-benzodiazepin-2-one und ihre Salze sowie Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
AT314541B (de) * 1970-10-19 1974-04-10 Sumitomo Chemical Co Verfahren zur Herstellung von neuen Benzodiazepinen und ihren Salzen
US4065451A (en) * 1971-03-30 1977-12-27 American Home Products 1,3-Dihydro-3-hydroxy-5-phenyl-2H-1,4-benzodiazepin-2-one, substituted diamino acetate esters and their acid salts
US3886276A (en) * 1971-03-30 1975-05-27 American Home Prod 1,3-Dihydro-3 -hydroxy-5-phenyl-2H-1,4-benzodiazepin-2-one, substituted diamino acetate esters and their acid salts in compositions and methods for inducing a calming effect
US3872089A (en) * 1971-05-14 1975-03-18 Hoffmann La Roche Substituted thienodiazepines
US3966943A (en) * 1971-09-13 1976-06-29 The Upjohn Company 6-Pyridyl benzodiazepines antidepressants
US3926952A (en) * 1972-10-03 1975-12-16 American Home Prod 1,4-Benzodiazepin-2-ones and their synthesis
US4012413A (en) * 1973-05-17 1977-03-15 The Upjohn Company Organic compounds and process
US3865815A (en) * 1973-11-29 1975-02-11 Hoffmann La Roche 7-Hydroxyamino-1,4-benzodiazepines
US4006135A (en) * 1974-06-19 1977-02-01 Ddsa Pharmaceuticals Hydroxymethyl benzodiazepine derivatives
US3969504A (en) * 1975-02-14 1976-07-13 The Upjohn Co. 6-Phenyl benzodiazepine antidepressants
FI783743A (fi) * 1977-12-14 1979-06-15 Gerot Pharmazeutika Foerfarande foer framstaellning av 3-di-n-propyl-acetoxi-benzodiazepin-2-oner
AT361492B (de) * 1978-12-18 1981-03-10 Gerot Pharmazeutika Verfahren zur herstellung von neuen 3-hydroxy- 1,4-benzodiazepin-2-onen

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3236838A (en) * 1964-06-09 1966-02-22 Hoffmann La Roche Certain 1-substituted-benzodiazepin-2-one compounds

Also Published As

Publication number Publication date
DE1545952A1 (de) 1969-12-18
CH462831A (de) 1968-09-30
BR6571654D0 (pt) 1973-08-14
NO118914B (da) 1970-03-02
BE668189A (da) 1965-12-01
SE310687B (da) 1969-05-12
NL6510539A (da) 1966-02-14
NO119588B (da) 1970-06-08
NL6510538A (da) 1966-02-14
DK125554B (da) 1973-03-05
FR135F (da)
BR6571653D0 (pt) 1973-08-14
DE1545952C3 (de) 1975-03-06
GB1102934A (en) 1968-02-14
IL23998A (en) 1969-02-27
BE668188A (da) 1966-02-14
IL23999A (en) 1969-05-28
SE312558B (da) 1969-07-21
US3391138A (en) 1968-07-02
DE1545953A1 (de) 1969-11-20
GB1106040A (en) 1968-03-13
DE1545952B2 (de) 1974-07-04

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