DK1106179T3 - Anvendelse af östrogenantagonister og östrogenagonister til hæmning af patologiske tilstande - Google Patents

Anvendelse af östrogenantagonister og östrogenagonister til hæmning af patologiske tilstande

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Publication number
DK1106179T3
DK1106179T3 DK01101953T DK01101953T DK1106179T3 DK 1106179 T3 DK1106179 T3 DK 1106179T3 DK 01101953 T DK01101953 T DK 01101953T DK 01101953 T DK01101953 T DK 01101953T DK 1106179 T3 DK1106179 T3 DK 1106179T3
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DK
Denmark
Prior art keywords
estrogen
pathological conditions
agonists
antagonists
inhibit pathological
Prior art date
Application number
DK01101953T
Other languages
Danish (da)
English (en)
Inventor
David D Thompson
David B Maclean
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of DK1106179T3 publication Critical patent/DK1106179T3/da

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/472Non-condensed isoquinolines, e.g. papaverine
    • A61K31/4725Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4453Non condensed piperidines, e.g. piperocaine only substituted in position 1, e.g. propipocaine, diperodon
    • AHUMAN NECESSITIES
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    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
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    • A61P25/34Tobacco-abuse
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30Oestrogens
    • AHUMAN NECESSITIES
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/32Antioestrogens

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  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Addiction (AREA)
  • Gynecology & Obstetrics (AREA)
  • Dermatology (AREA)
  • Emergency Medicine (AREA)
  • Pregnancy & Childbirth (AREA)
  • Psychiatry (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Pulmonology (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
DK01101953T 1996-02-28 1997-02-21 Anvendelse af östrogenantagonister og östrogenagonister til hæmning af patologiske tilstande DK1106179T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US1321296P 1996-02-28 1996-02-28

Publications (1)

Publication Number Publication Date
DK1106179T3 true DK1106179T3 (da) 2008-08-18

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ID=21758830

Family Applications (2)

Application Number Title Priority Date Filing Date
DK01101953T DK1106179T3 (da) 1996-02-28 1997-02-21 Anvendelse af östrogenantagonister og östrogenagonister til hæmning af patologiske tilstande
DK97301147T DK0792641T3 (da) 1996-02-28 1997-02-21 Anvendelse af estrogenantagonister og estrogenagonister til hæmning af patologiske tilstande

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK97301147T DK0792641T3 (da) 1996-02-28 1997-02-21 Anvendelse af estrogenantagonister og estrogenagonister til hæmning af patologiske tilstande

Country Status (17)

Country Link
US (8) US6107331A (es)
EP (2) EP0792641B1 (es)
JP (1) JPH107563A (es)
KR (1) KR970061254A (es)
CN (2) CN1515256A (es)
AT (2) ATE396728T1 (es)
AU (1) AU703473B2 (es)
CA (1) CA2198578C (es)
DE (2) DE69738740D1 (es)
DK (2) DK1106179T3 (es)
ES (2) ES2159811T3 (es)
GR (1) GR3036583T3 (es)
HK (1) HK1001963A1 (es)
IL (2) IL120266A (es)
MY (1) MY125602A (es)
PT (2) PT792641E (es)
ZA (1) ZA971714B (es)

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ZA971714B (en) 1997-08-27
US6613796B2 (en) 2003-09-02
US20040009994A1 (en) 2004-01-15
ES2159811T3 (es) 2001-10-16
IL120266A0 (en) 1997-06-10
DE69738740D1 (de) 2008-07-10
DK0792641T3 (da) 2001-10-08
IL164967A0 (en) 2005-12-18
US20020091121A1 (en) 2002-07-11
MX9701530A (es) 1998-06-30
CN1167617A (zh) 1997-12-17
US20050148625A1 (en) 2005-07-07
EP1106179A3 (en) 2004-01-07
MY125602A (en) 2006-08-30
US20010018451A1 (en) 2001-08-30
US6274618B1 (en) 2001-08-14
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US6911456B2 (en) 2005-06-28
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US6403611B2 (en) 2002-06-11
DE69705874D1 (de) 2001-09-06
AU703473B2 (en) 1999-03-25
PT1106179E (pt) 2008-07-28
ATE203670T1 (de) 2001-08-15
CA2198578C (en) 2002-06-11
JPH107563A (ja) 1998-01-13
IL120266A (en) 2005-05-17
ATE396728T1 (de) 2008-06-15
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US6355670B1 (en) 2002-03-12
US20030220349A1 (en) 2003-11-27
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US6107331A (en) 2000-08-22
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HK1001963A1 (en) 1998-07-24

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