DK0656888T3 - Sulfonylalkanoylaminohydroxyethylaminosulfonamider, anvendelige som retrovirale protease-inhibitorer - Google Patents

Sulfonylalkanoylaminohydroxyethylaminosulfonamider, anvendelige som retrovirale protease-inhibitorer

Info

Publication number
DK0656888T3
DK0656888T3 DK93920214.9T DK93920214T DK0656888T3 DK 0656888 T3 DK0656888 T3 DK 0656888T3 DK 93920214 T DK93920214 T DK 93920214T DK 0656888 T3 DK0656888 T3 DK 0656888T3
Authority
DK
Denmark
Prior art keywords
useful
protease inhibitors
retroviral protease
inhibitors
retroviral
Prior art date
Application number
DK93920214.9T
Other languages
Danish (da)
English (en)
Inventor
Michael L Vazquez
Richard A Mueller
John J Talley
Daniel Getman
Gary A Decrescenzo
John N Freskos
Original Assignee
Searle & Co
Monsanto Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Searle & Co, Monsanto Co filed Critical Searle & Co
Application granted granted Critical
Publication of DK0656888T3 publication Critical patent/DK0656888T3/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/63—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/18—Sulfonamides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/44—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
DK93920214.9T 1992-08-25 1993-08-24 Sulfonylalkanoylaminohydroxyethylaminosulfonamider, anvendelige som retrovirale protease-inhibitorer DK0656888T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US93507192A 1992-08-25 1992-08-25

Publications (1)

Publication Number Publication Date
DK0656888T3 true DK0656888T3 (da) 1998-02-09

Family

ID=25466549

Family Applications (1)

Application Number Title Priority Date Filing Date
DK93920214.9T DK0656888T3 (da) 1992-08-25 1993-08-24 Sulfonylalkanoylaminohydroxyethylaminosulfonamider, anvendelige som retrovirale protease-inhibitorer

Country Status (15)

Country Link
US (7) US5521219A (no)
EP (1) EP0656888B1 (no)
JP (1) JP4091654B2 (no)
KR (1) KR100296462B1 (no)
AT (1) ATE161828T1 (no)
AU (1) AU669223B2 (no)
CA (1) CA2140928C (no)
DE (1) DE69316223T2 (no)
DK (1) DK0656888T3 (no)
ES (1) ES2112430T3 (no)
FI (1) FI120343B (no)
GR (1) GR3025958T3 (no)
NO (1) NO303540B1 (no)
RU (1) RU2146668C1 (no)
WO (1) WO1994004493A1 (no)

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Also Published As

Publication number Publication date
NO303540B1 (no) 1998-07-27
EP0656888A1 (en) 1995-06-14
CA2140928A1 (en) 1994-02-26
FI950651A0 (fi) 1995-02-14
WO1994004493A1 (en) 1994-03-03
JP4091654B2 (ja) 2008-05-28
US6147117A (en) 2000-11-14
AU5082093A (en) 1994-03-15
ATE161828T1 (de) 1998-01-15
US5639769A (en) 1997-06-17
US5508294A (en) 1996-04-16
US5760064A (en) 1998-06-02
EP0656888B1 (en) 1998-01-07
AU669223B2 (en) 1996-05-30
CA2140928C (en) 2008-01-29
RU2146668C1 (ru) 2000-03-20
FI120343B (fi) 2009-09-30
NO950550D0 (no) 1995-02-14
RU95106996A (ru) 1996-11-20
KR100296462B1 (ko) 2001-10-24
GR3025958T3 (en) 1998-04-30
JPH08500825A (ja) 1996-01-30
DE69316223T2 (de) 1998-05-28
ES2112430T3 (es) 1998-04-01
US5521219A (en) 1996-05-28
FI950651A (fi) 1995-02-14
DE69316223D1 (de) 1998-02-12
KR950702961A (ko) 1995-08-23
NO950550L (no) 1995-02-14
US5510388A (en) 1996-04-23
US5965588A (en) 1999-10-12

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