DK0645389T3 - Fremgangsmåde til fremstilling af imidazopyridinderivater - Google Patents

Fremgangsmåde til fremstilling af imidazopyridinderivater

Info

Publication number
DK0645389T3
DK0645389T3 DK94114551.8T DK94114551T DK0645389T3 DK 0645389 T3 DK0645389 T3 DK 0645389T3 DK 94114551 T DK94114551 T DK 94114551T DK 0645389 T3 DK0645389 T3 DK 0645389T3
Authority
DK
Denmark
Prior art keywords
preparation
image
imidazopyridine derivatives
imidazopyridines
general formula
Prior art date
Application number
DK94114551.8T
Other languages
Danish (da)
English (en)
Inventor
Gerhard Dr Stucky
Rene Dr Imwinkelried
Original Assignee
Lonza Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lonza Ag filed Critical Lonza Ag
Application granted granted Critical
Publication of DK0645389T3 publication Critical patent/DK0645389T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK94114551.8T 1993-09-17 1994-09-15 Fremgangsmåde til fremstilling af imidazopyridinderivater DK0645389T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH281693 1993-09-17

Publications (1)

Publication Number Publication Date
DK0645389T3 true DK0645389T3 (da) 1997-03-10

Family

ID=4242236

Family Applications (1)

Application Number Title Priority Date Filing Date
DK94114551.8T DK0645389T3 (da) 1993-09-17 1994-09-15 Fremgangsmåde til fremstilling af imidazopyridinderivater

Country Status (22)

Country Link
US (1) US5446160A (cs)
EP (1) EP0645389B1 (cs)
JP (1) JP3713724B2 (cs)
KR (1) KR950008512A (cs)
AT (1) ATE148702T1 (cs)
AU (1) AU680025B2 (cs)
BR (1) BR9403594A (cs)
CA (1) CA2131680C (cs)
CZ (1) CZ285489B6 (cs)
DE (1) DE59401760D1 (cs)
DK (1) DK0645389T3 (cs)
ES (1) ES2098089T3 (cs)
GR (1) GR3022500T3 (cs)
HU (1) HU218488B (cs)
IL (1) IL110994A (cs)
PL (1) PL305067A1 (cs)
RU (1) RU94033473A (cs)
SI (1) SI0645389T1 (cs)
SK (1) SK111494A3 (cs)
TR (1) TR27788A (cs)
TW (1) TW410225B (cs)
ZA (1) ZA947189B (cs)

Families Citing this family (34)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9312853D0 (en) 1993-06-22 1993-08-04 Euro Celtique Sa Chemical compounds
US5591776A (en) 1994-06-24 1997-01-07 Euro-Celtique, S.A. Pheynl or benzyl-substituted rolipram-based compounds for and method of inhibiting phosphodiesterase IV
US5922751A (en) 1994-06-24 1999-07-13 Euro-Celtique, S.A. Aryl pyrazole compound for inhibiting phosphodiesterase IV and methods of using same
US6166041A (en) 1995-10-11 2000-12-26 Euro-Celtique, S.A. 2-heteroaryl and 2-heterocyclic benzoxazoles as PDE IV inhibitors for the treatment of asthma
US6075016A (en) 1996-04-10 2000-06-13 Euro-Celtique S.A. 6,5-fused aromatic ring systems having enhanced phosphodiesterase IV inhibitory activity
NZ502642A (en) * 1997-07-03 2002-06-28 Du Pont Pharm Co Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders
US6365589B1 (en) 1998-07-02 2002-04-02 Bristol-Myers Squibb Pharma Company Imidazo-pyridines, -pyridazines, and -triazines as corticotropin releasing factor antagonists
US6124463A (en) * 1998-07-02 2000-09-26 Dupont Pharmaceuticals Benzimidazoles as corticotropin release factor antagonists
CA2392992A1 (en) * 1999-12-17 2001-06-21 Dupont Pharmaceuticals Company Imidazopyrimidinyl and imidazopyridinyl derivatives
JP2007502293A (ja) 2003-08-12 2007-02-08 スリーエム イノベイティブ プロパティズ カンパニー ヒドロキシルアミン置換イミダゾ含有化合物
EP1658076B1 (en) 2003-08-27 2013-03-06 3M Innovative Properties Company Aryloxy and arylalkyleneoxy substituted imidazoquinolines
CA2537763A1 (en) 2003-09-05 2005-03-17 3M Innovative Properties Company Treatment for cd5+ b cell lymphoma
US7544697B2 (en) 2003-10-03 2009-06-09 Coley Pharmaceutical Group, Inc. Pyrazolopyridines and analogs thereof
AR046046A1 (es) 2003-10-03 2005-11-23 3M Innovative Properties Co Imidazoquinolinas alcoxi sustituidas. composiciones farmaceuticas.
CA2545825A1 (en) 2003-11-14 2005-06-02 3M Innovative Properties Company Hydroxylamine substituted imidazo ring compounds
CA2545774A1 (en) 2003-11-14 2005-06-02 3M Innovative Properties Company Oxime substituted imidazo ring compounds
BRPI0416936A (pt) 2003-11-25 2007-01-16 3M Innovative Properties Co sistemas de anel de imidazo substituìdos e métodos
EP1701955A1 (en) 2003-12-29 2006-09-20 3M Innovative Properties Company Arylalkenyl and arylalkynyl substituted imidazoquinolines
EP1699788A2 (en) 2003-12-30 2006-09-13 3M Innovative Properties Company Imidazoquinolinyl, imidazopyridinyl and imidazonaphthyridinyl sulfonamides
AU2005228150A1 (en) 2004-03-24 2005-10-13 3M Innovative Properties Company Amide substituted imidazopyridines, imidazoquinolines, and imidazonaphthyridines
WO2005123080A2 (en) 2004-06-15 2005-12-29 3M Innovative Properties Company Nitrogen-containing heterocyclyl substituted imidazoquinolines and imidazonaphthyridines
WO2006009826A1 (en) 2004-06-18 2006-01-26 3M Innovative Properties Company Aryloxy and arylalkyleneoxy substituted thiazoloquinolines and thiazolonaphthyridines
WO2006038923A2 (en) 2004-06-18 2006-04-13 3M Innovative Properties Company Aryl substituted imidazonaphthyridines
WO2006065280A2 (en) 2004-06-18 2006-06-22 3M Innovative Properties Company Isoxazole, dihydroisoxazole, and oxadiazole substituted imidazo ring compounds and methods
US8034938B2 (en) 2004-12-30 2011-10-11 3M Innovative Properties Company Substituted chiral fused [1,2]imidazo[4,5-c] ring compounds
JP5543068B2 (ja) 2004-12-30 2014-07-09 スリーエム イノベイティブ プロパティズ カンパニー キラル縮合[1,2]イミダゾ[4,5−c]環状化合物
US9248127B2 (en) 2005-02-04 2016-02-02 3M Innovative Properties Company Aqueous gel formulations containing immune response modifiers
EP1846405A2 (en) 2005-02-11 2007-10-24 3M Innovative Properties Company Oxime and hydroxylamine substituted imidazo 4,5-c ring compounds and methods
CA2602590A1 (en) 2005-04-01 2006-10-12 Coley Pharmaceutical Group, Inc. 1-substituted pyrazolo (3,4-c) ring compounds as modulators of cytokine biosynthesis for the treatment of viral infections and neoplastic diseases
EP1863770A4 (en) * 2005-04-01 2010-05-05 Coley Pharm Group Inc RING CLOSURE AND CORRESPONDING METHODS AND INTERMEDIATE PRODUCTS
US7943610B2 (en) 2005-04-01 2011-05-17 3M Innovative Properties Company Pyrazolopyridine-1,4-diamines and analogs thereof
AU2006292119A1 (en) * 2005-09-23 2007-03-29 3M Innovative Properties Company Method for 1H-imidazo[4,5-c]pyridines and analogs thereof
WO2008008432A2 (en) 2006-07-12 2008-01-17 Coley Pharmaceutical Group, Inc. Substituted chiral fused( 1,2) imidazo (4,5-c) ring compounds and methods
US20080139608A1 (en) * 2006-12-06 2008-06-12 Universiteit Leiden 2,6,8, Trisubstituted 1-deazapurines and their different uses

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3324115A1 (de) * 1983-07-05 1985-01-17 Dr. Karl Thomae Gmbh, 7950 Biberach Neue imidazole, ihre herstellung und diese verbindungen enthaltende arzneimittel
FR2643903A1 (fr) * 1989-03-03 1990-09-07 Union Pharma Scient Appl Nouveaux derives de benzimidazole, leurs procedes de preparation, intermediaires de synthese, compositions pharmaceutiques les contenant, utiles notamment pour le traitement des maladies cardiovasculaires, et des ulceres duodenaux
US5223499A (en) * 1989-05-30 1993-06-29 Merck & Co., Inc. 6-amino substituted imidazo[4,5-bipyridines as angiotensin II antagonists
US5240938A (en) * 1991-02-13 1993-08-31 Merck & Co., Inc. Angiotensin II antagonists incorporating a substituted pyridoimidazolyl ring
US5066654A (en) * 1990-10-22 1991-11-19 A. H. Robins Company, Incorporated 2-aryl-3-heterocyclicmethyl-3H-imidazo[4,5-b]pyridines as anxiolytics and anticonvulsants
US5128327A (en) * 1991-03-25 1992-07-07 Merck & Co., Inc. Angiotensin II antagonists incorporating a nitrogen containing six membered ring heterocycle

Also Published As

Publication number Publication date
GR3022500T3 (en) 1997-05-31
PL305067A1 (en) 1995-03-20
HU9402662D0 (en) 1994-11-28
AU680025B2 (en) 1997-07-17
IL110994A0 (en) 1994-11-28
CA2131680A1 (en) 1995-03-18
EP0645389B1 (de) 1997-02-05
BR9403594A (pt) 1995-05-16
EP0645389A1 (de) 1995-03-29
CZ226694A3 (en) 1995-04-12
JP3713724B2 (ja) 2005-11-09
IL110994A (en) 1998-02-08
TW410225B (en) 2000-11-01
HU218488B (hu) 2000-09-28
RU94033473A (ru) 1996-08-10
SK111494A3 (en) 1995-06-07
ATE148702T1 (de) 1997-02-15
HUT68250A (en) 1995-06-28
ES2098089T3 (es) 1997-04-16
SI0645389T1 (en) 1997-10-31
DE59401760D1 (de) 1997-03-20
KR950008512A (ko) 1995-04-17
AU7305894A (en) 1995-03-30
TR27788A (tr) 1995-08-29
ZA947189B (en) 1995-05-12
JPH07179465A (ja) 1995-07-18
CZ285489B6 (cs) 1999-08-11
US5446160A (en) 1995-08-29
CA2131680C (en) 2006-11-07

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