IL110994A - PROCESS FOR PREPARING 2-SUBSTITUTED-3H-IMIDAZO £4, 5-b| PYRIDINE DERIVATIVES - Google Patents

PROCESS FOR PREPARING 2-SUBSTITUTED-3H-IMIDAZO £4, 5-b| PYRIDINE DERIVATIVES

Info

Publication number
IL110994A
IL110994A IL110994A IL11099494A IL110994A IL 110994 A IL110994 A IL 110994A IL 110994 A IL110994 A IL 110994A IL 11099494 A IL11099494 A IL 11099494A IL 110994 A IL110994 A IL 110994A
Authority
IL
Israel
Prior art keywords
general formula
alkyl
aryl
groups
preparing
Prior art date
Application number
IL110994A
Other languages
English (en)
Other versions
IL110994A0 (en
Original Assignee
Lonza Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lonza Ag filed Critical Lonza Ag
Publication of IL110994A0 publication Critical patent/IL110994A0/xx
Publication of IL110994A publication Critical patent/IL110994A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IL110994A 1993-09-17 1994-09-18 PROCESS FOR PREPARING 2-SUBSTITUTED-3H-IMIDAZO £4, 5-b| PYRIDINE DERIVATIVES IL110994A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH281693 1993-09-17

Publications (2)

Publication Number Publication Date
IL110994A0 IL110994A0 (en) 1994-11-28
IL110994A true IL110994A (en) 1998-02-08

Family

ID=4242236

Family Applications (1)

Application Number Title Priority Date Filing Date
IL110994A IL110994A (en) 1993-09-17 1994-09-18 PROCESS FOR PREPARING 2-SUBSTITUTED-3H-IMIDAZO £4, 5-b| PYRIDINE DERIVATIVES

Country Status (22)

Country Link
US (1) US5446160A (cs)
EP (1) EP0645389B1 (cs)
JP (1) JP3713724B2 (cs)
KR (1) KR950008512A (cs)
AT (1) ATE148702T1 (cs)
AU (1) AU680025B2 (cs)
BR (1) BR9403594A (cs)
CA (1) CA2131680C (cs)
CZ (1) CZ285489B6 (cs)
DE (1) DE59401760D1 (cs)
DK (1) DK0645389T3 (cs)
ES (1) ES2098089T3 (cs)
GR (1) GR3022500T3 (cs)
HU (1) HU218488B (cs)
IL (1) IL110994A (cs)
PL (1) PL305067A1 (cs)
RU (1) RU94033473A (cs)
SI (1) SI0645389T1 (cs)
SK (1) SK111494A3 (cs)
TR (1) TR27788A (cs)
TW (1) TW410225B (cs)
ZA (1) ZA947189B (cs)

Families Citing this family (34)

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GB9312853D0 (en) 1993-06-22 1993-08-04 Euro Celtique Sa Chemical compounds
US5922751A (en) 1994-06-24 1999-07-13 Euro-Celtique, S.A. Aryl pyrazole compound for inhibiting phosphodiesterase IV and methods of using same
US5591776A (en) 1994-06-24 1997-01-07 Euro-Celtique, S.A. Pheynl or benzyl-substituted rolipram-based compounds for and method of inhibiting phosphodiesterase IV
US6166041A (en) 1995-10-11 2000-12-26 Euro-Celtique, S.A. 2-heteroaryl and 2-heterocyclic benzoxazoles as PDE IV inhibitors for the treatment of asthma
US6075016A (en) 1996-04-10 2000-06-13 Euro-Celtique S.A. 6,5-fused aromatic ring systems having enhanced phosphodiesterase IV inhibitory activity
AU746706B2 (en) * 1997-07-03 2002-05-02 Du Pont Pharmaceuticals Company Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders
US6365589B1 (en) 1998-07-02 2002-04-02 Bristol-Myers Squibb Pharma Company Imidazo-pyridines, -pyridazines, and -triazines as corticotropin releasing factor antagonists
US6124463A (en) * 1998-07-02 2000-09-26 Dupont Pharmaceuticals Benzimidazoles as corticotropin release factor antagonists
JP2003516992A (ja) * 1999-12-17 2003-05-20 デュポン ファーマシューティカルズ カンパニー イミダゾピリミジニル誘導体およびイミダゾピリジニル誘導体
BRPI0413558A (pt) 2003-08-12 2006-10-17 3M Innovative Properties Co compostos contendo imidazo substituìdo por hidroxilamina
RU2006105101A (ru) 2003-08-27 2007-10-10 3М Инновейтив Пропертиз Компани (US) Арилокси и арилалкиленокси замещенные имидазохинолины
CA2537763A1 (en) 2003-09-05 2005-03-17 3M Innovative Properties Company Treatment for cd5+ b cell lymphoma
US7544697B2 (en) 2003-10-03 2009-06-09 Coley Pharmaceutical Group, Inc. Pyrazolopyridines and analogs thereof
JP5043435B2 (ja) 2003-10-03 2012-10-10 スリーエム イノベイティブ プロパティズ カンパニー アルコキシ置換イミダゾキノリン
JP2007511527A (ja) 2003-11-14 2007-05-10 スリーエム イノベイティブ プロパティズ カンパニー オキシム置換イミダゾ環化合物
CN1906192A (zh) 2003-11-14 2007-01-31 3M创新有限公司 羟胺取代的咪唑环化合物
NZ547467A (en) 2003-11-25 2010-06-25 3M Innovative Properties Co Substituted imidazo ring system and methods
WO2005066170A1 (en) 2003-12-29 2005-07-21 3M Innovative Properties Company Arylalkenyl and arylalkynyl substituted imidazoquinolines
JP2007517044A (ja) 2003-12-30 2007-06-28 スリーエム イノベイティブ プロパティズ カンパニー イミダゾキノリニル、イミダゾピリジニル、およびイミダゾナフチリジニルスルホンアミド
TW200612932A (en) 2004-03-24 2006-05-01 3M Innovative Properties Co Amide substituted imidazopyridines, imidazoquinolines, and imidazonaphthyridines
WO2005123080A2 (en) 2004-06-15 2005-12-29 3M Innovative Properties Company Nitrogen-containing heterocyclyl substituted imidazoquinolines and imidazonaphthyridines
WO2006009826A1 (en) 2004-06-18 2006-01-26 3M Innovative Properties Company Aryloxy and arylalkyleneoxy substituted thiazoloquinolines and thiazolonaphthyridines
WO2006038923A2 (en) 2004-06-18 2006-04-13 3M Innovative Properties Company Aryl substituted imidazonaphthyridines
WO2006065280A2 (en) 2004-06-18 2006-06-22 3M Innovative Properties Company Isoxazole, dihydroisoxazole, and oxadiazole substituted imidazo ring compounds and methods
JP5313502B2 (ja) 2004-12-30 2013-10-09 スリーエム イノベイティブ プロパティズ カンパニー 置換キラル縮合［１，２］イミダゾ［４，５−ｃ］環状化合物
CA2592904C (en) 2004-12-30 2015-04-07 3M Innovative Properties Company Chiral fused [1,2]imidazo[4,5-c] ring compounds
AU2006210392A1 (en) 2005-02-04 2006-08-10 Coley Pharmaceutical Group, Inc. Aqueous gel formulations containing immune response modifiers
US7968563B2 (en) 2005-02-11 2011-06-28 3M Innovative Properties Company Oxime and hydroxylamine substituted imidazo[4,5-c] ring compounds and methods
EP1863814A1 (en) 2005-04-01 2007-12-12 Coley Pharmaceutical Group, Inc. 1-substituted pyrazolo (3,4-c) ring compounds as modulators of cytokine biosynthesis for the treatment of viral infections and neoplastic diseases
EP1863770A4 (en) * 2005-04-01 2010-05-05 Coley Pharm Group Inc RING CLOSURE AND CORRESPONDING METHODS AND INTERMEDIATE PRODUCTS
JP2008535832A (ja) 2005-04-01 2008-09-04 コーリー ファーマシューティカル グループ，インコーポレイテッド ピラゾロピリジン−１，４−ジアミン、およびそのアナログ
KR20080048551A (ko) * 2005-09-23 2008-06-02 콜레이 파마시티컬 그룹, 인코포레이티드 1Ｈ-이미다조[4,5-ｃ]피리딘 및 그의 유사체의 제조법
US7906506B2 (en) 2006-07-12 2011-03-15 3M Innovative Properties Company Substituted chiral fused [1,2] imidazo [4,5-c] ring compounds and methods
US20080139608A1 (en) * 2006-12-06 2008-06-12 Universiteit Leiden 2,6,8, Trisubstituted 1-deazapurines and their different uses

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3324115A1 (de) * 1983-07-05 1985-01-17 Dr. Karl Thomae Gmbh, 7950 Biberach Neue imidazole, ihre herstellung und diese verbindungen enthaltende arzneimittel
FR2643903A1 (fr) * 1989-03-03 1990-09-07 Union Pharma Scient Appl Nouveaux derives de benzimidazole, leurs procedes de preparation, intermediaires de synthese, compositions pharmaceutiques les contenant, utiles notamment pour le traitement des maladies cardiovasculaires, et des ulceres duodenaux
US5223499A (en) * 1989-05-30 1993-06-29 Merck & Co., Inc. 6-amino substituted imidazo[4,5-bipyridines as angiotensin II antagonists
US5240938A (en) * 1991-02-13 1993-08-31 Merck & Co., Inc. Angiotensin II antagonists incorporating a substituted pyridoimidazolyl ring
US5066654A (en) * 1990-10-22 1991-11-19 A. H. Robins Company, Incorporated 2-aryl-3-heterocyclicmethyl-3H-imidazo[4,5-b]pyridines as anxiolytics and anticonvulsants
US5128327A (en) * 1991-03-25 1992-07-07 Merck & Co., Inc. Angiotensin II antagonists incorporating a nitrogen containing six membered ring heterocycle

Also Published As

Publication number Publication date
EP0645389B1 (de) 1997-02-05
SK111494A3 (en) 1995-06-07
HU9402662D0 (en) 1994-11-28
IL110994A0 (en) 1994-11-28
BR9403594A (pt) 1995-05-16
ATE148702T1 (de) 1997-02-15
JPH07179465A (ja) 1995-07-18
ZA947189B (en) 1995-05-12
HUT68250A (en) 1995-06-28
EP0645389A1 (de) 1995-03-29
AU7305894A (en) 1995-03-30
JP3713724B2 (ja) 2005-11-09
ES2098089T3 (es) 1997-04-16
CA2131680C (en) 2006-11-07
GR3022500T3 (en) 1997-05-31
AU680025B2 (en) 1997-07-17
HU218488B (hu) 2000-09-28
SI0645389T1 (en) 1997-10-31
PL305067A1 (en) 1995-03-20
RU94033473A (ru) 1996-08-10
DK0645389T3 (da) 1997-03-10
DE59401760D1 (de) 1997-03-20
US5446160A (en) 1995-08-29
CA2131680A1 (en) 1995-03-18
KR950008512A (ko) 1995-04-17
CZ226694A3 (en) 1995-04-12
CZ285489B6 (cs) 1999-08-11
TR27788A (tr) 1995-08-29
TW410225B (en) 2000-11-01

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