DE69839821D1 - Neue sulfonamid-substituierte chroman-derivate verwendbar als beta 3 adrenorezeptor agonisten - Google Patents
Neue sulfonamid-substituierte chroman-derivate verwendbar als beta 3 adrenorezeptor agonistenInfo
- Publication number
- DE69839821D1 DE69839821D1 DE69839821T DE69839821T DE69839821D1 DE 69839821 D1 DE69839821 D1 DE 69839821D1 DE 69839821 T DE69839821 T DE 69839821T DE 69839821 T DE69839821 T DE 69839821T DE 69839821 D1 DE69839821 D1 DE 69839821D1
- Authority
- DE
- Germany
- Prior art keywords
- adrene
- beta
- receptor agonists
- chroman derivatives
- substituted chroman
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
- C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Diabetes (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Emergency Medicine (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Endocrinology (AREA)
- Neurology (AREA)
- Vascular Medicine (AREA)
- Child & Adolescent Psychology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Cardiology (AREA)
- Urology & Nephrology (AREA)
- Heart & Thoracic Surgery (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyrane Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US99458597A | 1997-12-19 | 1997-12-19 | |
PCT/US1998/024627 WO1999032475A1 (en) | 1997-12-19 | 1998-11-17 | Novel sulfonamide substituted chroman derivatives useful as beta-3 adrenoreceptor agonists |
Publications (1)
Publication Number | Publication Date |
---|---|
DE69839821D1 true DE69839821D1 (de) | 2008-09-11 |
Family
ID=25540825
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE69839821T Expired - Fee Related DE69839821D1 (de) | 1997-12-19 | 1998-11-17 | Neue sulfonamid-substituierte chroman-derivate verwendbar als beta 3 adrenorezeptor agonisten |
Country Status (12)
Country | Link |
---|---|
EP (1) | EP1054881B1 (de) |
JP (1) | JP2001526281A (de) |
AR (1) | AR016691A1 (de) |
AT (1) | ATE402933T1 (de) |
AU (1) | AU751015B2 (de) |
CA (1) | CA2314925A1 (de) |
CO (1) | CO4990952A1 (de) |
DE (1) | DE69839821D1 (de) |
IL (1) | IL136688A0 (de) |
TW (1) | TW502032B (de) |
WO (1) | WO1999032475A1 (de) |
ZA (1) | ZA9810489B (de) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2000256331A (ja) * | 1999-01-08 | 2000-09-19 | Nippon Bayer Agrochem Co Ltd | テトラゾリノン誘導体および除草剤としてのその用途 |
DE60015036T2 (de) * | 1999-07-23 | 2006-03-02 | Pfizer Products Inc., Groton | Zwischenprodukte und ein Verfahren zur Herstellung von beta3-Adrenergischer Rezeptor-Agoniste |
BR0112409A (pt) * | 2000-07-13 | 2003-07-22 | Lilly Co Eli | Agonistas para beta3 adrenérgico |
CZ20013076A3 (cs) | 2000-08-29 | 2002-04-17 | Kuraray Co., Ltd. | Způsob výroby chromankarboxylové kyseliny |
JP2005505586A (ja) | 2001-10-04 | 2005-02-24 | ワイス | 5−ヒドロキシトリプタミン−6リガンドとしてのクロマン誘導体 |
US7323462B2 (en) | 2002-12-10 | 2008-01-29 | Pfizer Inc. | Morpholine dopamine agonists |
US7034051B2 (en) | 2003-08-28 | 2006-04-25 | Adolor Corporation | Fused bicyclic carboxamide derivatives and methods of their use |
US20050222247A1 (en) * | 2003-12-13 | 2005-10-06 | Bayer Healthcare Ag | Chroman derivatives |
US20120135997A1 (en) | 2009-07-17 | 2012-05-31 | Shionogi & Co., Ltd. | Pharmaceutical composition comprising a lactam or benzenesulfonamide compound |
EP2536693A4 (de) * | 2010-02-17 | 2014-08-06 | UNIVERSITé LAVAL | Substituierte 2-imidazolidone und analoga |
CN108218845B (zh) * | 2016-12-21 | 2022-11-29 | 江苏柯菲平医药股份有限公司 | 一类色满-6-磺酰胺RORγ调节剂及其用途 |
CN112107583A (zh) * | 2020-07-31 | 2020-12-22 | 东南大学 | 一种色满-6-磺酰胺RORγ调节剂的A晶型化合物的组合物及其制备方法和应用 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0091749A3 (de) * | 1982-04-08 | 1984-12-05 | Beecham Group Plc | Ethanolamin-Derivate, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Zusammensetzungen |
US5451677A (en) * | 1993-02-09 | 1995-09-19 | Merck & Co., Inc. | Substituted phenyl sulfonamides as selective β 3 agonists for the treatment of diabetes and obesity |
IL113410A (en) * | 1994-04-26 | 1999-11-30 | Merck & Co Inc | Substituted sulfonamides having an asymmetric center and pharmaceutical compositions containing them |
US5663194A (en) * | 1995-07-25 | 1997-09-02 | Mewshaw; Richard E. | Chroman-2-ylmethylamino derivatives |
FR2746395B1 (fr) * | 1996-03-22 | 1998-04-17 | Adir | Nouveaux derives d'arylethanolamine et d'aryloxypropanolamine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
EP0801060A1 (de) * | 1996-04-09 | 1997-10-15 | Pfizer Inc. | Heterocyclische Beta-3 adrenergische Angonisten |
-
1998
- 1998-11-17 CA CA002314925A patent/CA2314925A1/en not_active Abandoned
- 1998-11-17 TW TW087118968A patent/TW502032B/zh not_active IP Right Cessation
- 1998-11-17 IL IL13668898A patent/IL136688A0/xx unknown
- 1998-11-17 ZA ZA9810489A patent/ZA9810489B/xx unknown
- 1998-11-17 JP JP2000525412A patent/JP2001526281A/ja not_active Withdrawn
- 1998-11-17 AU AU14183/99A patent/AU751015B2/en not_active Ceased
- 1998-11-17 DE DE69839821T patent/DE69839821D1/de not_active Expired - Fee Related
- 1998-11-17 WO PCT/US1998/024627 patent/WO1999032475A1/en active IP Right Grant
- 1998-11-17 AT AT98958070T patent/ATE402933T1/de not_active IP Right Cessation
- 1998-11-17 EP EP98958070A patent/EP1054881B1/de not_active Expired - Lifetime
- 1998-11-18 AR ARP980105846A patent/AR016691A1/es not_active Application Discontinuation
- 1998-11-18 CO CO98067870A patent/CO4990952A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
EP1054881A1 (de) | 2000-11-29 |
ZA9810489B (en) | 1999-05-20 |
EP1054881B1 (de) | 2008-07-30 |
AR016691A1 (es) | 2001-07-25 |
ATE402933T1 (de) | 2008-08-15 |
TW502032B (en) | 2002-09-11 |
CA2314925A1 (en) | 1999-07-01 |
JP2001526281A (ja) | 2001-12-18 |
AU1418399A (en) | 1999-07-12 |
WO1999032475A1 (en) | 1999-07-01 |
CO4990952A1 (es) | 2000-12-26 |
AU751015B2 (en) | 2002-08-08 |
IL136688A0 (en) | 2001-06-14 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition | ||
8339 | Ceased/non-payment of the annual fee |