DE60331437D1 - Nachspaltige sulfurentschützung zur konvergenten proteinherstellung beim verfahren von chemischer ligation - Google Patents

Nachspaltige sulfurentschützung zur konvergenten proteinherstellung beim verfahren von chemischer ligation

Info

Publication number
DE60331437D1
DE60331437D1 DE60331437T DE60331437T DE60331437D1 DE 60331437 D1 DE60331437 D1 DE 60331437D1 DE 60331437 T DE60331437 T DE 60331437T DE 60331437 T DE60331437 T DE 60331437T DE 60331437 D1 DE60331437 D1 DE 60331437D1
Authority
DE
Germany
Prior art keywords
chemical ligation
oligopeptide
convergent
present
sulphide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60331437T
Other languages
German (de)
English (en)
Inventor
Paolo Botti
Matteo Villain
Sonia Manganiello
Hubert Gaertner
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Amylin Pharmaceuticals LLC
Original Assignee
Amylin Pharmaceuticals LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Amylin Pharmaceuticals LLC filed Critical Amylin Pharmaceuticals LLC
Application granted granted Critical
Publication of DE60331437D1 publication Critical patent/DE60331437D1/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/107General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides
    • C07K1/1072General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides by covalent attachment of residues or functional groups
    • C07K1/1077General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides by covalent attachment of residues or functional groups by covalent attachment of residues other than amino acids or peptide residues, e.g. sugars, polyols, fatty acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/02General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length in solution
    • C07K1/026General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length in solution by fragment condensation in solution
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/04General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/46Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • C07K14/47Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/06Linear peptides containing only normal peptide links having 5 to 11 amino acids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Analytical Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Toxicology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Peptides Or Proteins (AREA)
DE60331437T 2002-06-10 2003-06-09 Nachspaltige sulfurentschützung zur konvergenten proteinherstellung beim verfahren von chemischer ligation Expired - Lifetime DE60331437D1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US38780302P 2002-06-10 2002-06-10
US40753002P 2002-08-30 2002-08-30
PCT/IB2003/005087 WO2003106615A2 (en) 2002-06-10 2003-06-09 Post-cleavage sulfur deprotection for convergent protein synthesis by chemical ligation

Publications (1)

Publication Number Publication Date
DE60331437D1 true DE60331437D1 (de) 2010-04-08

Family

ID=29739962

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60331437T Expired - Lifetime DE60331437D1 (de) 2002-06-10 2003-06-09 Nachspaltige sulfurentschützung zur konvergenten proteinherstellung beim verfahren von chemischer ligation

Country Status (9)

Country Link
US (1) US7781488B2 (https=)
EP (1) EP1529056B1 (https=)
JP (1) JP4559219B2 (https=)
AT (1) ATE458745T1 (https=)
AU (1) AU2003276286A1 (https=)
CA (1) CA2487342A1 (https=)
DE (1) DE60331437D1 (https=)
ES (1) ES2340376T3 (https=)
WO (1) WO2003106615A2 (https=)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2877946B1 (fr) * 2004-11-12 2011-02-11 Commissariat Energie Atomique Peptides derives de la maurocalcine utilisables comme vecteurs pour l'adressage intracellulaire de molecules d'interet
EP1904515B1 (en) * 2005-06-16 2010-12-08 Amylin Pharmaceuticals, Inc. Side-chain extended ligation
EP1770099A1 (en) * 2005-09-28 2007-04-04 University of Geneva Method of producing a modified (poly)peptide
US7674881B2 (en) * 2005-10-07 2010-03-09 The University Of Chicago Convergent synthesis of proteins by kinetically controlled ligation
JP2010537984A (ja) * 2007-08-28 2010-12-09 イプセン ファルマ ソシエテ パール アクシオン サンプリフィエ ポリペプチドおよび蛋白質の化学合成のための方法および中間体
EP2197895A4 (en) * 2007-09-04 2012-12-26 Ipsen Pharma Sas METHODS AND INTERMEDIATES FOR CHEMICAL SYNTHESIS OF POLYPEPTIDES AND PROTEINS
US9175053B2 (en) 2010-02-09 2015-11-03 Ben-Gurion University Of The Negev Research And Development Authority Chemical preparation of ubiquitin thioesters and modifications thereof
PL3317390T3 (pl) 2015-07-02 2021-04-19 Novus International Inc. Anionowe środki powierzchniowo czynne
US10584306B2 (en) 2017-08-11 2020-03-10 Board Of Regents Of The University Of Oklahoma Surfactant microemulsions
US20240076311A1 (en) * 2020-12-28 2024-03-07 Jiangsu Genscript Biotech Co., Ltd. Method for synthesizing peptide thioesters and head-to-tail amide cyclic peptide thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE285415T1 (de) * 1997-06-13 2005-01-15 Gryphon Therapeutics Inc Festphasige native chemische ligation von ungeschützten oder n-cystein-geschützten peptiden in wässrigen lösungen
KR20030046389A (ko) * 2000-09-01 2003-06-12 그리폰 테라퓨틱스, 인코포레이티드 친핵체에 안정한 티오에스테르 발생 화합물, 제조 및 사용방법
BR0113579A (pt) * 2000-09-08 2003-06-17 Gryphon Therapeutics Inc Proteìnas sintéticas modificadas por polìmero
EE200300089A (et) * 2000-09-08 2005-02-15 Gryphon Therapeutics, Inc. Sünteetilised erütropoeesi stimuleerivad valgud, nende valmistamismeetodid ning kasutamine
GB0113657D0 (en) * 2001-06-05 2001-07-25 Geneprot Inc Improved native chemical ligation with three or more components

Also Published As

Publication number Publication date
AU2003276286A1 (en) 2003-12-31
EP1529056B1 (en) 2010-02-24
WO2003106615A2 (en) 2003-12-24
ES2340376T3 (es) 2010-06-02
ATE458745T1 (de) 2010-03-15
EP1529056A2 (en) 2005-05-11
JP4559219B2 (ja) 2010-10-06
US7781488B2 (en) 2010-08-24
CA2487342A1 (en) 2003-12-24
WO2003106615A3 (en) 2004-09-16
US20070059792A1 (en) 2007-03-15
JP2005529186A (ja) 2005-09-29

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