DE60129672T2 - Tyrosinkinase inhibitoren - Google Patents

Tyrosinkinase inhibitoren Download PDF

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Publication number
DE60129672T2
DE60129672T2 DE60129672T DE60129672T DE60129672T2 DE 60129672 T2 DE60129672 T2 DE 60129672T2 DE 60129672 T DE60129672 T DE 60129672T DE 60129672 T DE60129672 T DE 60129672T DE 60129672 T2 DE60129672 T2 DE 60129672T2
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DE
Germany
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optionally substituted
alkyl
substituents selected
aryl
alkenyl
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
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DE60129672T
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German (de)
English (en)
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DE60129672D1 (de
Inventor
Mark E. Rahway FRALEY
George D. Rahway HARTMAN
Randall W. Rahway HUNGATE
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Merck and Co Inc
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Merck and Co Inc
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Publication of DE60129672D1 publication Critical patent/DE60129672D1/de
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Publication of DE60129672T2 publication Critical patent/DE60129672T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Immunology (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DE60129672T 2000-02-25 2001-02-21 Tyrosinkinase inhibitoren Expired - Fee Related DE60129672T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US18502300P 2000-02-25 2000-02-25
US185023P 2000-02-25
PCT/US2001/005482 WO2001062251A1 (en) 2000-02-25 2001-02-21 Tyrosine kinase inhibitors

Publications (2)

Publication Number Publication Date
DE60129672D1 DE60129672D1 (de) 2007-09-13
DE60129672T2 true DE60129672T2 (de) 2008-04-30

Family

ID=22679236

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60129672T Expired - Fee Related DE60129672T2 (de) 2000-02-25 2001-02-21 Tyrosinkinase inhibitoren

Country Status (9)

Country Link
US (1) US6420382B2 (https=)
EP (1) EP1259235B1 (https=)
JP (1) JP2003523389A (https=)
AT (1) ATE368457T1 (https=)
AU (2) AU2001238575B2 (https=)
CA (1) CA2400875A1 (https=)
DE (1) DE60129672T2 (https=)
ES (1) ES2288928T3 (https=)
WO (1) WO2001062251A1 (https=)

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Also Published As

Publication number Publication date
AU2001238575B2 (en) 2005-04-07
US6420382B2 (en) 2002-07-16
AU3857501A (en) 2001-09-03
DE60129672D1 (de) 2007-09-13
ATE368457T1 (de) 2007-08-15
EP1259235A1 (en) 2002-11-27
US20010044451A1 (en) 2001-11-22
ES2288928T3 (es) 2008-02-01
CA2400875A1 (en) 2001-08-30
JP2003523389A (ja) 2003-08-05
EP1259235A4 (en) 2004-11-03
EP1259235B1 (en) 2007-08-01
WO2001062251A1 (en) 2001-08-30

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