DE3520469A1 - Neue anthracycline, verfahren zu deren herstellung, zwischenverbindungen und pharmazeutische zubereitung - Google Patents

Neue anthracycline, verfahren zu deren herstellung, zwischenverbindungen und pharmazeutische zubereitung

Info

Publication number
DE3520469A1
DE3520469A1 DE19853520469 DE3520469A DE3520469A1 DE 3520469 A1 DE3520469 A1 DE 3520469A1 DE 19853520469 DE19853520469 DE 19853520469 DE 3520469 A DE3520469 A DE 3520469A DE 3520469 A1 DE3520469 A1 DE 3520469A1
Authority
DE
Germany
Prior art keywords
compound
amino
formula
pharmaceutically acceptable
group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
DE19853520469
Other languages
German (de)
English (en)
Inventor
Michele Mailand/Milano Caruso
Sergio Penco
Antonio Suarato
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Farmitalia Carlo Erba SpA Mailand/milano
Farmitalia Carlo Erba SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmitalia Carlo Erba SpA Mailand/milano, Farmitalia Carlo Erba SRL filed Critical Farmitalia Carlo Erba SpA Mailand/milano
Publication of DE3520469A1 publication Critical patent/DE3520469A1/de
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/24—Condensed ring systems having three or more rings
    • C07H15/252—Naphthacene radicals, e.g. daunomycins, adriamycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Furan Compounds (AREA)
DE19853520469 1984-06-08 1985-06-07 Neue anthracycline, verfahren zu deren herstellung, zwischenverbindungen und pharmazeutische zubereitung Ceased DE3520469A1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB848414619A GB8414619D0 (en) 1984-06-08 1984-06-08 Anthracyclines

Publications (1)

Publication Number Publication Date
DE3520469A1 true DE3520469A1 (de) 1985-12-12

Family

ID=10562109

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19853520469 Ceased DE3520469A1 (de) 1984-06-08 1985-06-07 Neue anthracycline, verfahren zu deren herstellung, zwischenverbindungen und pharmazeutische zubereitung

Country Status (4)

Country Link
JP (1) JPH0631297B2 (ja)
BE (1) BE902610A (ja)
DE (1) DE3520469A1 (ja)
GB (1) GB8414619D0 (ja)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1996007665A1 (en) * 1994-09-09 1996-03-14 Pharmacia S.P.A. Anthracycline derivatives

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9325420D0 (en) * 1993-12-13 1994-02-16 Erba Carlo Spa 4'-o-sulfonyl-anthracycline derivatives
DE10297516B4 (de) 2001-12-11 2008-08-28 Kayaba Industry Co., Ltd. Elektromagnetisches Proportional-Stromregelventil

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0030295A1 (de) * 1979-11-22 1981-06-17 FARMITALIA CARLO ERBA S.p.A. Verfahren zur Herstellung von 4'-Epidaunorubicin, 3',4'-Diepidaunorubicin, hierbei entstehende Zwischenprodukte sowie deren Verwendung
US4438105A (en) * 1982-04-19 1984-03-20 Farmaitalia Carlo Erba S.P.A 4'-Iododerivatives of anthracycline glycosides
DE3428945A1 (de) * 1983-08-11 1985-02-28 Farmitalia Carlo Erba S.p.A., Mailand/Milano 4'-halogenanthracyclinglykoside, verfahren zu deren herstellung und diese enthaltende pharmazeutische zubereitung

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0030295A1 (de) * 1979-11-22 1981-06-17 FARMITALIA CARLO ERBA S.p.A. Verfahren zur Herstellung von 4'-Epidaunorubicin, 3',4'-Diepidaunorubicin, hierbei entstehende Zwischenprodukte sowie deren Verwendung
US4438105A (en) * 1982-04-19 1984-03-20 Farmaitalia Carlo Erba S.P.A 4'-Iododerivatives of anthracycline glycosides
DE3428945A1 (de) * 1983-08-11 1985-02-28 Farmitalia Carlo Erba S.p.A., Mailand/Milano 4'-halogenanthracyclinglykoside, verfahren zu deren herstellung und diese enthaltende pharmazeutische zubereitung

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
Cancer Treat.Rep., 1978, 62, S. 375-380 *
J.Med.Chem., 1975, 18, S. 703-707 *

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1996007665A1 (en) * 1994-09-09 1996-03-14 Pharmacia S.P.A. Anthracycline derivatives

Also Published As

Publication number Publication date
GB8414619D0 (en) 1984-07-11
JPS611697A (ja) 1986-01-07
JPH0631297B2 (ja) 1994-04-27
BE902610A (fr) 1985-09-30

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Legal Events

Date Code Title Description
8127 New person/name/address of the applicant

Owner name: FARMITALIA CARLO ERBA S.R.L., MAILAND/MILANO, IT

8128 New person/name/address of the agent

Representative=s name: EITLE, W., DIPL.-ING. HOFFMANN, K., DIPL.-ING. DR.

8110 Request for examination paragraph 44
8131 Rejection