DE2647496A1 - Neue cephalosporinderivate - Google Patents
Neue cephalosporinderivateInfo
- Publication number
- DE2647496A1 DE2647496A1 DE19762647496 DE2647496A DE2647496A1 DE 2647496 A1 DE2647496 A1 DE 2647496A1 DE 19762647496 DE19762647496 DE 19762647496 DE 2647496 A DE2647496 A DE 2647496A DE 2647496 A1 DE2647496 A1 DE 2647496A1
- Authority
- DE
- Germany
- Prior art keywords
- deep
- acid
- radical
- amino
- compound according
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
- C07D295/21—Radicals derived from sulfur analogues of carbonic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C57/00—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
- C07C57/52—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms containing halogen
- C07C57/58—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms containing halogen containing six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C57/00—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
- C07C57/64—Acyl halides
- C07C57/76—Acyl halides containing halogen outside the carbonyl halide groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/24—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cephalosporin Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US05/625,541 US4031083A (en) | 1975-10-24 | 1975-10-24 | Cephalosporin antibiotics |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DE2647496A1 true DE2647496A1 (de) | 1977-04-28 |
Family
ID=24506570
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE19762647496 Withdrawn DE2647496A1 (de) | 1975-10-24 | 1976-10-21 | Neue cephalosporinderivate |
Country Status (16)
| Country | Link |
|---|---|
| US (2) | US4031083A (enExample) |
| JP (1) | JPS5251390A (enExample) |
| AU (1) | AU503927B2 (enExample) |
| BE (1) | BE847551A (enExample) |
| CA (1) | CA1073900A (enExample) |
| DE (1) | DE2647496A1 (enExample) |
| DK (1) | DK480076A (enExample) |
| ES (1) | ES452637A1 (enExample) |
| FR (1) | FR2328472A1 (enExample) |
| GB (1) | GB1510417A (enExample) |
| IE (1) | IE43965B1 (enExample) |
| NL (1) | NL7611707A (enExample) |
| NO (1) | NO763600L (enExample) |
| NZ (1) | NZ182400A (enExample) |
| SE (1) | SE7611777L (enExample) |
| ZA (1) | ZA766308B (enExample) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4031083A (en) * | 1975-10-24 | 1977-06-21 | Yeda Research And Development Co., Ltd. | Cephalosporin antibiotics |
| US4180571A (en) * | 1976-03-25 | 1979-12-25 | Shionogi & Co., Ltd. | Arylmalonamido-1-oxadethiacephalosporins |
| JPS609718B2 (ja) * | 1977-08-25 | 1985-03-12 | 塩野義製薬株式会社 | チアジアゾリルチオセフアロスポリン類縁抗生物質 |
| US4236002A (en) * | 1977-12-23 | 1980-11-25 | Yeda Research & Development Co., Ltd. | Cephalosporin derivatives |
| JPS5690088A (en) * | 1979-11-02 | 1981-07-21 | Meiji Seika Kaisha Ltd | Novel cephalosporin analog compound |
| GB2162537A (en) * | 1984-08-01 | 1986-02-05 | Albright & Wilson | Suspension culture of plant tissue |
| AU3052300A (en) * | 1999-01-15 | 2000-08-01 | Elf Atochem S.A. | Polymerisation using a compound which is both an initiator and a surfactant |
| EP2958889B1 (en) | 2013-02-25 | 2017-03-22 | The Scripps Research Institute | Neoseptins: small molecule adjuvants |
Citations (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA892580A (en) | 1972-02-08 | Patchornik Avraham | Polymer acylation of penicillins | |
| US3655658A (en) | 1968-01-30 | 1972-04-11 | Leo Pharm Prod Ltd | 7(alpha-amino-alpha-phenylacetamido)-cephalosporanate esters |
| US3657232A (en) | 1970-06-19 | 1972-04-18 | R & L Molecular Research Ltd | 7-((o-aminomethylphenylthio)-acetamido) cephalosporanic acid |
| DE2236620A1 (de) | 1972-07-26 | 1973-08-02 | Werner Selzer | Fussboden- bzw. sockelleiste |
| US3778432A (en) | 1971-12-13 | 1973-12-11 | Merck & Co Inc | Isocyanates and carbamates of penicillins and 3-cephem-4-carboxylic acids |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3341531A (en) * | 1967-02-15 | 1967-09-12 | American Cyanamid Co | Substituted 7-acetylamino cephalosporanic acids |
| DE2118635A1 (de) * | 1971-04-17 | 1972-11-02 | Farbwerke Hoechst AG, vormals Meister Lucius & Brüning, 6000 Frankfurt | Acylaminocephalosporansäuren und Verfahren zu ihrer Herstellung |
| NL7305936A (enExample) * | 1972-05-05 | 1973-11-07 | ||
| US3919206A (en) * | 1973-09-25 | 1975-11-11 | Yeda Res & Dev | 7-(Halomethylaryl)acetamidocephalosporin derivatives |
| US3919208A (en) * | 1973-10-09 | 1975-11-11 | Yeda Res & Dev | 7-(Cyanomethylaryl)acetamide-cephalosporin derivatives |
| US4031083A (en) * | 1975-10-24 | 1977-06-21 | Yeda Research And Development Co., Ltd. | Cephalosporin antibiotics |
| US4026887A (en) * | 1975-10-24 | 1977-05-31 | Yeda Research & Development Co. Ltd. | Cephalosporin antibiotics |
-
1975
- 1975-10-24 US US05/625,541 patent/US4031083A/en not_active Expired - Lifetime
-
1976
- 1976-10-18 CA CA263,626A patent/CA1073900A/en not_active Expired
- 1976-10-21 DE DE19762647496 patent/DE2647496A1/de not_active Withdrawn
- 1976-10-22 NL NL7611707A patent/NL7611707A/xx not_active Application Discontinuation
- 1976-10-22 BE BE171718A patent/BE847551A/xx unknown
- 1976-10-22 NZ NZ182400A patent/NZ182400A/xx unknown
- 1976-10-22 IE IE2328/76A patent/IE43965B1/en unknown
- 1976-10-22 AU AU18920/76A patent/AU503927B2/en not_active Expired
- 1976-10-22 ES ES452637A patent/ES452637A1/es not_active Expired
- 1976-10-22 ZA ZA766308A patent/ZA766308B/xx unknown
- 1976-10-22 FR FR7631921A patent/FR2328472A1/fr active Granted
- 1976-10-22 DK DK480076A patent/DK480076A/da not_active Application Discontinuation
- 1976-10-22 SE SE7611777A patent/SE7611777L/xx not_active Application Discontinuation
- 1976-10-22 NO NO763600A patent/NO763600L/no unknown
- 1976-10-23 JP JP51126822A patent/JPS5251390A/ja active Pending
- 1976-10-25 GB GB44199/76A patent/GB1510417A/en not_active Expired
-
1977
- 1977-01-14 US US05/759,276 patent/US4093802A/en not_active Expired - Lifetime
Patent Citations (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA892580A (en) | 1972-02-08 | Patchornik Avraham | Polymer acylation of penicillins | |
| US3655658A (en) | 1968-01-30 | 1972-04-11 | Leo Pharm Prod Ltd | 7(alpha-amino-alpha-phenylacetamido)-cephalosporanate esters |
| US3657232A (en) | 1970-06-19 | 1972-04-18 | R & L Molecular Research Ltd | 7-((o-aminomethylphenylthio)-acetamido) cephalosporanic acid |
| US3778432A (en) | 1971-12-13 | 1973-12-11 | Merck & Co Inc | Isocyanates and carbamates of penicillins and 3-cephem-4-carboxylic acids |
| DE2236620A1 (de) | 1972-07-26 | 1973-08-02 | Werner Selzer | Fussboden- bzw. sockelleiste |
Non-Patent Citations (3)
| Title |
|---|
| B. Reichert, et al., Pharmazie 5, 10 (1950) |
| E. Emmet Reid, Organic Chemistry of Bi-Valent Sulfur, Chemical Publishing, Co., New York, 1962, Bd. IV, S. 196 |
| J. Parrod, Compt. rend, 234, 1062 (1952) |
Also Published As
| Publication number | Publication date |
|---|---|
| GB1510417A (en) | 1978-05-10 |
| FR2328472B1 (enExample) | 1980-04-18 |
| AU503927B2 (en) | 1979-09-27 |
| AU1892076A (en) | 1978-04-27 |
| NO763600L (enExample) | 1977-04-26 |
| US4093802A (en) | 1978-06-06 |
| CA1073900A (en) | 1980-03-18 |
| IE43965B1 (en) | 1981-07-15 |
| ZA766308B (en) | 1977-09-28 |
| IE43965L (en) | 1977-04-24 |
| JPS5251390A (en) | 1977-04-25 |
| NZ182400A (en) | 1978-12-18 |
| FR2328472A1 (fr) | 1977-05-20 |
| DK480076A (da) | 1977-04-25 |
| SE7611777L (sv) | 1977-04-25 |
| NL7611707A (nl) | 1977-04-26 |
| US4031083A (en) | 1977-06-21 |
| BE847551A (fr) | 1977-02-14 |
| ES452637A1 (es) | 1977-10-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 8139 | Disposal/non-payment of the annual fee |