DE2351948A1 - 4-aryl-5-aminoalkyl-4-oxazolin-2-one, verfahren zu deren herstellung und diese verbindungen enthaltende pharmazeutische zusammensetzungen - Google Patents
4-aryl-5-aminoalkyl-4-oxazolin-2-one, verfahren zu deren herstellung und diese verbindungen enthaltende pharmazeutische zusammensetzungenInfo
- Publication number
- DE2351948A1 DE2351948A1 DE19732351948 DE2351948A DE2351948A1 DE 2351948 A1 DE2351948 A1 DE 2351948A1 DE 19732351948 DE19732351948 DE 19732351948 DE 2351948 A DE2351948 A DE 2351948A DE 2351948 A1 DE2351948 A1 DE 2351948A1
- Authority
- DE
- Germany
- Prior art keywords
- group
- fluorophenyl
- oxazolin
- pharmaceutically acceptable
- acceptable salts
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/48—Nitrogen atoms not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/36—One oxygen atom
- C07D263/38—One oxygen atom attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/46—Sulfur atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT3053672 | 1972-10-16 | ||
| IT2811573A IT1056733B (it) | 1973-08-22 | 1973-08-22 | 4 aril 5 aminoalohil 4 ossazolin 2 oni loro derivati e processi per la loro preparazione |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DE2351948A1 true DE2351948A1 (de) | 1974-04-25 |
Family
ID=26328766
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE19732351948 Withdrawn DE2351948A1 (de) | 1972-10-16 | 1973-10-16 | 4-aryl-5-aminoalkyl-4-oxazolin-2-one, verfahren zu deren herstellung und diese verbindungen enthaltende pharmazeutische zusammensetzungen |
Country Status (13)
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0180136A2 (de) | 1984-11-02 | 1986-05-07 | Bayer Ag | Substituierte Azolylmethyl-cyclopropyl-carbinol-Derivate |
| US4728661A (en) * | 1985-11-13 | 1988-03-01 | Merrell Dow Pharmaceuticals Inc. | Cardiotonic phenyl oxazolones |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4123529A (en) * | 1976-04-23 | 1978-10-31 | Lilly Industries Limited | Phenylpiperazine derivatives |
| PT77428B (fr) * | 1982-10-05 | 1986-02-27 | Cortial | Procede pour preparer de nouvelles amino-2-substitue-5-oxazoli-nes-2 et des compositions les contenant |
| FR2546167B2 (fr) * | 1983-05-19 | 1985-07-12 | Cortial | Nouvelles amino-2 piperazino et piperidinomethyl-5 oxazolines-2, leur methode de preparation ainsi que leur application therapeutique |
| US6159990A (en) * | 1997-06-18 | 2000-12-12 | Synaptic Pharmaceutical Corporation | Oxazolidinones as α1A receptor antagonists |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3576808A (en) * | 1967-09-15 | 1971-04-27 | Miles Lab | N-4-phenyl-1-piperazinylalkyl-5-phenyl-oxazolidinones |
| JPS4922770A (US07655688-20100202-C00109.png) * | 1972-06-22 | 1974-02-28 |
-
1973
- 1973-10-03 US US403275A patent/US3930008A/en not_active Expired - Lifetime
- 1973-10-11 CH CH1449973A patent/CH605859A5/xx not_active IP Right Cessation
- 1973-10-12 GB GB4787573A patent/GB1429571A/en not_active Expired
- 1973-10-15 NL NL7314147.A patent/NL161154C/xx not_active IP Right Cessation
- 1973-10-15 FI FI3183/73A patent/FI57752C/fi active
- 1973-10-15 SE SE7313966A patent/SE391717B/xx unknown
- 1973-10-15 ES ES419632A patent/ES419632A1/es not_active Expired
- 1973-10-15 NO NO4002/73A patent/NO140299C/no unknown
- 1973-10-15 CA CA183,418A patent/CA1016550A/en not_active Expired
- 1973-10-16 FR FR7336838A patent/FR2202701B1/fr not_active Expired
- 1973-10-16 JP JP48116238A patent/JPS4993360A/ja active Pending
- 1973-10-16 DK DK560273AA patent/DK135122B/da unknown
- 1973-10-16 DE DE19732351948 patent/DE2351948A1/de not_active Withdrawn
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0180136A2 (de) | 1984-11-02 | 1986-05-07 | Bayer Ag | Substituierte Azolylmethyl-cyclopropyl-carbinol-Derivate |
| US4728661A (en) * | 1985-11-13 | 1988-03-01 | Merrell Dow Pharmaceuticals Inc. | Cardiotonic phenyl oxazolones |
Also Published As
| Publication number | Publication date |
|---|---|
| NL161154C (nl) | 1980-01-15 |
| NL7314147A (US07655688-20100202-C00109.png) | 1974-04-18 |
| AU6121673A (en) | 1975-04-10 |
| ES419632A1 (es) | 1976-06-16 |
| CA1016550A (en) | 1977-08-30 |
| FR2202701B1 (US07655688-20100202-C00109.png) | 1980-01-11 |
| US3930008A (en) | 1975-12-30 |
| DK135122C (US07655688-20100202-C00109.png) | 1977-08-08 |
| NL161154B (nl) | 1979-08-15 |
| SE391717B (sv) | 1977-02-28 |
| FR2202701A1 (US07655688-20100202-C00109.png) | 1974-05-10 |
| FI57752B (fi) | 1980-06-30 |
| FI57752C (fi) | 1980-10-10 |
| DK135122B (da) | 1977-03-07 |
| CH605859A5 (US07655688-20100202-C00109.png) | 1978-10-13 |
| NO140299C (no) | 1979-08-08 |
| NO140299B (no) | 1979-04-30 |
| GB1429571A (en) | 1976-03-24 |
| JPS4993360A (US07655688-20100202-C00109.png) | 1974-09-05 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 8139 | Disposal/non-payment of the annual fee |