DE2314040A1 - Verfahren zur herstellung von 3-desacetoxycephalosporinderivaten - Google Patents

Verfahren zur herstellung von 3-desacetoxycephalosporinderivaten

Info

Publication number
DE2314040A1
DE2314040A1 DE19732314040 DE2314040A DE2314040A1 DE 2314040 A1 DE2314040 A1 DE 2314040A1 DE 19732314040 DE19732314040 DE 19732314040 DE 2314040 A DE2314040 A DE 2314040A DE 2314040 A1 DE2314040 A1 DE 2314040A1
Authority
DE
Germany
Prior art keywords
sulfide
acid
ester
reaction
penicillin
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE19732314040
Other languages
German (de)
English (en)
Inventor
Shoichiro Fujii
Masayasu Kato
Kenzo Naito
Michiyuki Sendai
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Takeda Pharmaceutical Co Ltd
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of DE2314040A1 publication Critical patent/DE2314040A1/de
Pending legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
DE19732314040 1972-03-23 1973-03-21 Verfahren zur herstellung von 3-desacetoxycephalosporinderivaten Pending DE2314040A1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2945972A JPS536158B2 (US06248540-20010619-C00021.png) 1972-03-23 1972-03-23

Publications (1)

Publication Number Publication Date
DE2314040A1 true DE2314040A1 (de) 1973-09-27

Family

ID=12276671

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19732314040 Pending DE2314040A1 (de) 1972-03-23 1973-03-21 Verfahren zur herstellung von 3-desacetoxycephalosporinderivaten

Country Status (13)

Country Link
US (1) US4122258A (US06248540-20010619-C00021.png)
JP (1) JPS536158B2 (US06248540-20010619-C00021.png)
AT (1) AT322105B (US06248540-20010619-C00021.png)
BE (1) BE797214A (US06248540-20010619-C00021.png)
CA (1) CA1034115A (US06248540-20010619-C00021.png)
CH (1) CH585757A5 (US06248540-20010619-C00021.png)
DE (1) DE2314040A1 (US06248540-20010619-C00021.png)
DK (1) DK136724B (US06248540-20010619-C00021.png)
ES (1) ES412910A1 (US06248540-20010619-C00021.png)
FR (1) FR2177071B1 (US06248540-20010619-C00021.png)
GB (1) GB1359451A (US06248540-20010619-C00021.png)
HU (1) HU166027B (US06248540-20010619-C00021.png)
NL (1) NL7304152A (US06248540-20010619-C00021.png)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2555183A1 (de) * 1974-12-13 1976-06-16 Lilly Co Eli Verfahren zur herstellung von 7-acylamido-3-methyl-3-cephem-4-carbonsaeureestern

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0115770B2 (en) * 1983-01-07 1996-06-19 Takeda Chemical Industries, Ltd. Thiazole Derivatives

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK136480B (da) * 1969-03-11 1977-10-17 Glaxo Lab Ltd Fremgangsmåde til fremstilling af 7beta-acylamido-3-metylceph-3-em-4-karboxylsyreestere ved omlejring af en 6beta-acylamidopenicillansyre-1-oxydester.
US3632850A (en) * 1969-03-18 1972-01-04 Lilly Co Eli Cephalexin synthesis
GB1312233A (en) * 1969-12-05 1973-04-04 Glaxo Lab Ltd Cephalosporin compounds
US3852281A (en) * 1970-02-18 1974-12-03 Koninklijke Gist Spiritus Process for the preparation of 7-substituted amino-desacetoxycephalosporanic acid compounds
US3852295A (en) * 1970-03-10 1974-12-03 Glaxo Lab Ltd Salts of mono-o-substituted and o,o-diaryl substituted phosphoric acids and a nitrogen base
US3862181A (en) * 1970-10-28 1975-01-21 Squibb & Sons Inc Process for preparing cephalosporins
US3843637A (en) * 1971-05-11 1974-10-22 Bristol Myers Co Process for rearranging 6-acylamidopenicillanic acid-1-oxides to 7-acyla mido-3-methyl-ceph-3-em-4-carboxylic acids
GB1431174A (en) * 1972-06-30 1976-04-07 Clin Midy Process for the conversion of a penicillin s-oxide into a corresponding desacetoxycephalosporin
JPS4943999A (US06248540-20010619-C00021.png) * 1972-09-01 1974-04-25

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2555183A1 (de) * 1974-12-13 1976-06-16 Lilly Co Eli Verfahren zur herstellung von 7-acylamido-3-methyl-3-cephem-4-carbonsaeureestern

Also Published As

Publication number Publication date
ES412910A1 (es) 1975-12-16
JPS4897892A (US06248540-20010619-C00021.png) 1973-12-13
FR2177071A1 (US06248540-20010619-C00021.png) 1973-11-02
DK136724B (da) 1977-11-14
BE797214A (fr) 1973-09-24
CH585757A5 (US06248540-20010619-C00021.png) 1977-03-15
US4122258A (en) 1978-10-24
AT322105B (de) 1975-05-12
HU166027B (US06248540-20010619-C00021.png) 1974-12-28
JPS536158B2 (US06248540-20010619-C00021.png) 1978-03-04
DK136724C (US06248540-20010619-C00021.png) 1978-04-24
NL7304152A (US06248540-20010619-C00021.png) 1973-09-25
GB1359451A (en) 1974-07-10
FR2177071B1 (US06248540-20010619-C00021.png) 1978-06-09
CA1034115A (en) 1978-07-04

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Legal Events

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OHA Expiration of time for request for examination