DE2310329A1 - Arabinofuranosylcytosine und verfahren zu ihrer herstellung - Google Patents

Arabinofuranosylcytosine und verfahren zu ihrer herstellung

Info

Publication number
DE2310329A1
DE2310329A1 DE19732310329 DE2310329A DE2310329A1 DE 2310329 A1 DE2310329 A1 DE 2310329A1 DE 19732310329 DE19732310329 DE 19732310329 DE 2310329 A DE2310329 A DE 2310329A DE 2310329 A1 DE2310329 A1 DE 2310329A1
Authority
DE
Germany
Prior art keywords
arabinofuranosyl
cytosine
pharmaceutically acceptable
anhydro
chloride
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE19732310329
Other languages
German (de)
English (en)
Inventor
John G Moffat
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Roche Palo Alto LLC
Original Assignee
Roche Palo Alto LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roche Palo Alto LLC filed Critical Roche Palo Alto LLC
Publication of DE2310329A1 publication Critical patent/DE2310329A1/de
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06—Pyrimidine radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/12—Triazine radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DE19732310329 1972-03-03 1973-03-01 Arabinofuranosylcytosine und verfahren zu ihrer herstellung Pending DE2310329A1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/231,754 US3998807A (en) 1972-03-03 1972-03-03 Arabinofuranosyl cytosines and methods of making

Publications (1)

Publication Number Publication Date
DE2310329A1 true DE2310329A1 (de) 1973-09-20

Family

ID=22870525

Family Applications (2)

Application Number Title Priority Date Filing Date
DE19732310329 Pending DE2310329A1 (de) 1972-03-03 1973-03-01 Arabinofuranosylcytosine und verfahren zu ihrer herstellung
DE2365719*A Pending DE2365719A1 (de) 1972-03-03 1973-03-01 Arabinofuranosyl-6-azacytosine und verfahren zu ihrer herstellung

Family Applications After (1)

Application Number Title Priority Date Filing Date
DE2365719*A Pending DE2365719A1 (de) 1972-03-03 1973-03-01 Arabinofuranosyl-6-azacytosine und verfahren zu ihrer herstellung

Country Status (9)

Country Link
US (1) US3998807A (enExample)
JP (1) JPS4992078A (enExample)
CH (2) CH583249A5 (enExample)
DE (2) DE2310329A1 (enExample)
ES (2) ES412270A1 (enExample)
FR (1) FR2181780B1 (enExample)
GB (2) GB1427572A (enExample)
NL (1) NL7303000A (enExample)
SE (2) SE399560B (enExample)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5159880A (en) * 1974-11-22 1976-05-25 Asahi Chemical Ind N44 ashirunukureoshidojikarubonsanesuteruno seiho
US4267171A (en) * 1979-07-02 1981-05-12 The Regents Of The University Of California C-5 Substituted cytosine nucleosides
JPS5639019A (en) * 1979-09-05 1981-04-14 Yamasa Shoyu Co Ltd Antiviral agent
US4684630A (en) * 1983-08-24 1987-08-04 Repta Arnold J Method of parenterally delivering drugs and related compositions
GB9307043D0 (en) * 1993-04-05 1993-05-26 Norsk Hydro As Chemical compounds
US6551210B2 (en) * 2000-10-24 2003-04-22 Motion Technologies, Llc. Continuously variable transmission
TWI332507B (en) * 2002-11-19 2010-11-01 Hoffmann La Roche Antiviral nucleoside derivatives
AU2003296601A1 (en) * 2002-12-10 2004-06-30 F. Hoffmann-La Roche Ag Antiviral nucleoside derivatives
UA99836C2 (en) * 2007-09-26 2012-10-10 Маунт Синай Скул Оф Медсин Azacytidine analogue and using thereof
ATE547419T1 (de) * 2008-11-05 2012-03-15 Cognis Ip Man Gmbh Verfahren zur herstellung von acyclovir-prodrugs

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3155646A (en) * 1960-08-23 1964-11-03 Upjohn Co 1-arabinofuranosyl-5-halouracil and process for the preparation thereof
GB1070413A (en) * 1962-11-15 1967-06-01 Sankyo Co A process for preparing purine and pyrimidine nucleosides
US3328388A (en) * 1964-09-02 1967-06-27 Merck & Co Inc Arabinofuranosyl pyrimidines and methods of preparing same
US3338882A (en) * 1965-06-28 1967-08-29 Upjohn Co 2'-and 3'-phosphates of 1-beta-d-arabinofuranosylcytosine
US3463850A (en) * 1967-01-03 1969-08-26 Merck & Co Inc Arabinofuranosyl 2-thiopyrimidines and pharmaceutical compositions thereof
US3658788A (en) * 1969-06-06 1972-04-25 Salk Inst For Biological Studi Aminooxazolines and products thereof and processes for synthesizing same
US3755296A (en) * 1969-07-24 1973-08-28 Kohjin Co Process for preparing 1-{62 -d-arabinofuranosyl-cytosine and 2,2{40 -cyclocytidine
US3709874A (en) * 1970-03-19 1973-01-09 Syntex Corp 1-beta-d-arabinofuranosyl cytosine derivatives and methods of preparing
GB1322136A (en) * 1971-01-27 1973-07-04 Upjohn Co Ara-cytidine derivatives
US3894000A (en) * 1971-01-27 1975-07-08 Upjohn Co Ara-cytidine derivatives and process of preparation

Also Published As

Publication number Publication date
AU5274373A (en) 1974-09-05
ES412270A1 (es) 1976-10-16
CH583249A5 (enExample) 1976-12-31
FR2181780B1 (enExample) 1977-07-01
NL7303000A (enExample) 1973-09-06
ES441538A1 (es) 1977-04-01
JPS4992078A (enExample) 1974-09-03
GB1427571A (en) 1976-03-10
GB1427572A (en) 1976-03-10
DE2365719A1 (de) 1976-01-29
FR2181780A1 (enExample) 1973-12-07
US3998807A (en) 1976-12-21
CH585766A5 (enExample) 1977-03-15
SE7604155L (sv) 1976-04-08
SE399560B (sv) 1978-02-20

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