DE1795254A1 - Verfahren zur Herstellung von Benzodiazepinderivaten - Google Patents

Verfahren zur Herstellung von Benzodiazepinderivaten

Info

Publication number
DE1795254A1
DE1795254A1 DE19681795254 DE1795254A DE1795254A1 DE 1795254 A1 DE1795254 A1 DE 1795254A1 DE 19681795254 DE19681795254 DE 19681795254 DE 1795254 A DE1795254 A DE 1795254A DE 1795254 A1 DE1795254 A1 DE 1795254A1
Authority
DE
Germany
Prior art keywords
methyl
compound
benzodiazepine
formula
reaction
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE19681795254
Other languages
German (de)
English (en)
Inventor
Field George Francis
Sternbach Leo Henryk
Zally William Joseph
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of DE1795254A1 publication Critical patent/DE1795254A1/de
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/20—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DE19681795254 1967-09-06 1968-08-29 Verfahren zur Herstellung von Benzodiazepinderivaten Pending DE1795254A1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US66571667A 1967-09-06 1967-09-06
US71825968A 1968-04-02 1968-04-02

Publications (1)

Publication Number Publication Date
DE1795254A1 true DE1795254A1 (de) 1972-02-17

Family

ID=27099271

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19681795254 Pending DE1795254A1 (de) 1967-09-06 1968-08-29 Verfahren zur Herstellung von Benzodiazepinderivaten

Country Status (12)

Country Link
US (1) US3624073A (enExample)
AT (1) AT280295B (enExample)
CH (1) CH503040A (enExample)
DE (1) DE1795254A1 (enExample)
DK (2) DK119166B (enExample)
ES (1) ES357870A1 (enExample)
FI (1) FI50977C (enExample)
IE (1) IE32814B1 (enExample)
NL (1) NL6812560A (enExample)
NO (2) NO129795B (enExample)
SE (2) SE365517B (enExample)
YU (1) YU32233B (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4002610A (en) * 1975-09-22 1977-01-11 Mcneil Laboratories, Incorporated 2-Aminobenzodiazepine-5-ones
US4022767A (en) * 1975-09-22 1977-05-10 Mcneil Laboratories, Incorporated 2-Aminobenzodiazepine-5-ones
US5308430A (en) * 1990-01-30 1994-05-03 Makoto Saito Reinforcing fiber sheet, method of manufacturing the same, and the method of reinforcing structure with the reinforcing fiber sheet
US5962337A (en) * 1995-06-29 1999-10-05 Pharmacopeia, Inc. Combinatorial 1,4-benzodiazepin-2,5-dione library
NZ601238A (en) * 2010-01-25 2014-07-25 Jacob Kobelt Apparatus and method for distributing fluid

Also Published As

Publication number Publication date
DK119166B (da) 1970-11-23
DK122726B (da) 1972-04-04
IE32814L (en) 1969-03-06
CH503040A (de) 1971-02-15
NL6812560A (enExample) 1969-03-10
ES357870A1 (es) 1970-04-01
NO129744B (enExample) 1974-05-20
AT280295B (de) 1970-04-10
US3624073A (en) 1971-11-30
SE339477B (enExample) 1971-10-11
FI50977B (enExample) 1976-05-31
IE32814B1 (en) 1973-12-12
SE365517B (enExample) 1974-03-25
YU205168A (en) 1973-12-31
YU32233B (en) 1974-06-30
NO129795B (enExample) 1974-05-27
FI50977C (fi) 1976-09-10

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