DE1670392A1 - Neue Pyrimidine und Verfahren zu ihrer Herstellung - Google Patents

Neue Pyrimidine und Verfahren zu ihrer Herstellung

Info

Publication number
DE1670392A1
DE1670392A1 DE19661670392 DE1670392A DE1670392A1 DE 1670392 A1 DE1670392 A1 DE 1670392A1 DE 19661670392 DE19661670392 DE 19661670392 DE 1670392 A DE1670392 A DE 1670392A DE 1670392 A1 DE1670392 A1 DE 1670392A1
Authority
DE
Germany
Prior art keywords
amino
piperazine
pyrimidyl
radicals
carbon atoms
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE19661670392
Other languages
German (de)
English (en)
Inventor
Dr-Chem Ernst Schweizer
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
BASF Schweiz AG
Original Assignee
Ciba Geigy AG
Ciba AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG, Ciba AG filed Critical Ciba Geigy AG
Publication of DE1670392A1 publication Critical patent/DE1670392A1/de
Pending legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/50Three nitrogen atoms
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DE19661670392 1965-10-22 1966-10-14 Neue Pyrimidine und Verfahren zu ihrer Herstellung Pending DE1670392A1 (de)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
CH506368A CH478817A (de) 1965-10-22 1965-10-22 Verfahren zur Herstellung neuer N,N'-Di-(pyrimidyl-(4)-aminoalkyl)-diazacycloalkanen
CH1751468A CH499528A (de) 1965-10-22 1965-10-22 Verfahren zur Herstellung neuer Pyrimidine
CH506468A CH478818A (de) 1965-10-22 1965-10-22 Verfahren zur Herstellung neuer N,N'-Di-(pyrimidyl-(4)-aminoalkyl)-diazacycloalkanen
CH506568A CH478819A (de) 1965-10-22 1965-10-22 Verfahren zur Herstellung neuer N,N'-Di-(pyrimidyl-(4)-aminoalkyl)-diazacycloalkanen
CH1463065A CH478816A (de) 1965-10-22 1965-10-22 Verfahren zur Herstellung neuer N,N'-Di-(pyrimidyl-(4)-aminoalkyl)-diazacycloalkanen
CH1133066 1966-08-05

Publications (1)

Publication Number Publication Date
DE1670392A1 true DE1670392A1 (de) 1970-07-16

Family

ID=27543760

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19661670392 Pending DE1670392A1 (de) 1965-10-22 1966-10-14 Neue Pyrimidine und Verfahren zu ihrer Herstellung

Country Status (11)

Country Link
US (1) US3503963A (US20030199744A1-20031023-C00003.png)
BE (1) BE688660A (US20030199744A1-20031023-C00003.png)
BR (1) BR6683919D0 (US20030199744A1-20031023-C00003.png)
CH (5) CH478818A (US20030199744A1-20031023-C00003.png)
DE (1) DE1670392A1 (US20030199744A1-20031023-C00003.png)
FR (3) FR1500479A (US20030199744A1-20031023-C00003.png)
GB (1) GB1135259A (US20030199744A1-20031023-C00003.png)
IL (1) IL26473A (US20030199744A1-20031023-C00003.png)
NL (1) NL6614961A (US20030199744A1-20031023-C00003.png)
SE (1) SE345273B (US20030199744A1-20031023-C00003.png)
SU (2) SU436494A3 (US20030199744A1-20031023-C00003.png)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH485754A (de) * 1966-07-28 1970-02-15 Ciba Geigy Verfahren zur Herstellung neuer Aminopyrimidine
PT1599468E (pt) 2003-01-14 2008-01-14 Arena Pharm Inc Derivados de arilo e heteroarilo 1,2,3.-trissubstituídos comomoduladores do metabolismo, e profilaxia e tratamento dedesordens relacionadas tais como diabetes e hiperglicemia
US20070066590A1 (en) * 2003-02-24 2007-03-22 Jones Robert M Phenyl-and pyridylpiperidine-derivatives as modulators of glucose metabolism
AR045047A1 (es) 2003-07-11 2005-10-12 Arena Pharm Inc Derivados arilo y heteroarilo trisustituidos como moduladores del metabolismo y de la profilaxis y tratamiento de desordenes relacionados con los mismos
CN101870690A (zh) * 2004-06-04 2010-10-27 艾尼纳制药公司 作为代谢调节剂的经取代芳基和杂芳基衍生物及其相关病症的预防和治疗
HN2005000795A (es) * 2004-10-15 2010-08-19 Aventis Pharma Inc Pirimidinas como antagonistas del receptor de prostaglandina d2
MY148521A (en) * 2005-01-10 2013-04-30 Arena Pharm Inc Substituted pyridinyl and pyrimidinyl derivatives as modulators of metabolism and the treatment of disorders related thereto
DOP2006000010A (es) 2005-01-10 2006-07-31 Arena Pharm Inc Procedimiento para preparar eteres aromáticos
MX2008003634A (es) * 2005-09-16 2009-10-08 Arena Pharm Inc Moduladores del metabolismo y tratamiento de los trastornos metabolicos.
TW200811147A (en) * 2006-07-06 2008-03-01 Arena Pharm Inc Modulators of metabolism and the treatment of disorders related thereto
TW200811140A (en) * 2006-07-06 2008-03-01 Arena Pharm Inc Modulators of metabolism and the treatment of disorders related thereto
SG10201500639TA (en) 2010-01-27 2015-03-30 Arena Pharm Inc Processes for the preparation of (r)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid and salts thereof
CN103221410B (zh) 2010-09-22 2017-09-15 艾尼纳制药公司 Gpr119受体调节剂和对与其相关的障碍的治疗
EP3242666A1 (en) 2015-01-06 2017-11-15 Arena Pharmaceuticals, Inc. Methods of treating conditions related to the s1p1 receptor
DK3310760T3 (da) 2015-06-22 2022-10-24 Arena Pharm Inc Krystallinsk L-argininsalt af (R)-2-(7-(4-cyclopentyl-3-(trifluormethyl)benzyloxy)-1,2,3,4-tetrahydrocyclopenta[b]indol-3- yl)eddikesyre til anvendelse ved S1P1-receptor-associerede lidelser
CA3053418A1 (en) 2017-02-16 2018-08-23 Arena Pharmaceuticals, Inc. Compounds and methods for treatment of primary biliary cholangitis

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB944443A (US20030199744A1-20031023-C00003.png) * 1959-09-25 1900-01-01

Also Published As

Publication number Publication date
GB1135259A (en) 1968-12-04
FR6083M (US20030199744A1-20031023-C00003.png) 1968-06-04
BE688660A (US20030199744A1-20031023-C00003.png) 1967-04-21
IL26473A (en) 1971-08-25
SU436494A3 (ru) 1974-07-15
CH478817A (de) 1969-09-30
CH478819A (de) 1969-09-30
SE345273B (US20030199744A1-20031023-C00003.png) 1972-05-23
FR1500479A (fr) 1967-11-03
NL6614961A (US20030199744A1-20031023-C00003.png) 1967-04-24
BR6683919D0 (pt) 1973-12-04
SU427513A3 (ru) 1974-05-05
US3503963A (en) 1970-03-31
FR6084M (US20030199744A1-20031023-C00003.png) 1968-06-04
CH478818A (de) 1969-09-30
CH478816A (de) 1969-09-30
CH499528A (de) 1970-11-30

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