DE1470060A1 - 2,5-Diazabicyclo-[2,2,1]-heptane und octane und Verfahren zu ihrer Herstellung - Google Patents

2,5-Diazabicyclo-[2,2,1]-heptane und octane und Verfahren zu ihrer Herstellung

Info

Publication number
DE1470060A1
DE1470060A1 DE19641470060 DE1470060A DE1470060A1 DE 1470060 A1 DE1470060 A1 DE 1470060A1 DE 19641470060 DE19641470060 DE 19641470060 DE 1470060 A DE1470060 A DE 1470060A DE 1470060 A1 DE1470060 A1 DE 1470060A1
Authority
DE
Germany
Prior art keywords
compound
formula
general formula
coor
meaning
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE19641470060
Other languages
German (de)
English (en)
Inventor
Sarett Lewis Hastings
Matzuk Alexander Richard
Tsung-Ying Shen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of DE1470060A1 publication Critical patent/DE1470060A1/de
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44—Iso-indoles; Hydrogenated iso-indoles
    • C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
    • C07C51/347—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups
    • C07C51/363—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups by introduction of halogen; by substitution of halogen atoms by other halogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
    • C07C51/58—Preparation of carboxylic acid halides
    • C07C51/60—Preparation of carboxylic acid halides by conversion of carboxylic acids or their anhydrides or esters, lactones, salts into halides with the same carboxylic acid part
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08—Bridged systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06—Peri-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
DE19641470060 1963-02-05 1964-01-27 2,5-Diazabicyclo-[2,2,1]-heptane und octane und Verfahren zu ihrer Herstellung Pending DE1470060A1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US256240A US3167561A (en) 1963-02-05 1963-02-05 2, 5-diazabicyclo-[2,2,1]heptanes and [2,2,2]octanes

Publications (1)

Publication Number Publication Date
DE1470060A1 true DE1470060A1 (de) 1969-07-17

Family

ID=22971515

Family Applications (2)

Application Number Title Priority Date Filing Date
DE19641795538 Pending DE1795538A1 (de) 1963-02-05 1964-01-27 2,5-Diaza-3-monoxo- und 3,6-Dioxobicyclo-[2,2,1]-heptane und [2,2,2]-octane und Verfahren zu ihrer Herstellung
DE19641470060 Pending DE1470060A1 (de) 1963-02-05 1964-01-27 2,5-Diazabicyclo-[2,2,1]-heptane und octane und Verfahren zu ihrer Herstellung

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DE19641795538 Pending DE1795538A1 (de) 1963-02-05 1964-01-27 2,5-Diaza-3-monoxo- und 3,6-Dioxobicyclo-[2,2,1]-heptane und [2,2,2]-octane und Verfahren zu ihrer Herstellung

Country Status (8)

Country Link
US (1) US3167561A (enExample)
BR (1) BR6456585D0 (enExample)
DE (2) DE1795538A1 (enExample)
DK (2) DK114206B (enExample)
FR (1) FR1559560A (enExample)
GB (1) GB1041863A (enExample)
NL (2) NL6400946A (enExample)
SE (1) SE311661B (enExample)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0397351A1 (en) * 1989-05-11 1990-11-14 Pfizer Inc. Preparation of diazabicyclic intermediates
US5196548A (en) * 1989-05-11 1993-03-23 Pfizer Inc. Preparation of diazabicyclic Intermediates

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3318876A (en) * 1962-12-11 1967-05-09 Lepetit Spa Substituted piperazines and process for preparing same
US3281423A (en) * 1964-02-03 1966-10-25 Merck & Co Inc 1, 3-ethanopiperazines and process
DE1620230A1 (de) * 1966-11-19 1970-02-12 Roehm & Haas Gmbh Verfahren zur Herstellung von 2,5-Diketopiperazinen
DE2428792A1 (de) * 1974-06-14 1976-01-02 Knoll Ag Neue antiarrhythmika
WO1997017961A1 (en) * 1995-11-13 1997-05-22 Smithkline Beecham Corporation Hemoregulatory compounds
WO2011121633A1 (ja) * 2010-03-29 2011-10-06 株式会社 東芝 酸性ガス吸収剤、酸性ガス除去装置および酸性ガス除去方法
US10231970B2 (en) 2014-09-30 2019-03-19 NV Heterocycles Methods of producing heteropolycycles via bis-epoxidation

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2832784A (en) * 1958-04-29 Comparison of activities of piperazine
US2744086A (en) * 1949-11-26 1956-05-01 Chemstrand Corp Dyeable acrylonitrile fiber forming compositions
US2872476A (en) * 1955-05-25 1959-02-03 Zyma Sa New meta-dialkylaminoethoxybenzoic acid esters, their hydrochlorides, and process for their preparation
US2905706A (en) * 1957-08-09 1959-09-22 Dow Chemical Co 2-nitro-3, 4, 6-trichlorophenyl benzoates
US3068233A (en) * 1960-06-14 1962-12-11 Jefferson Chem Co Inc Method for preparing n, n'-dimethyltriethylenediamonim dinitrate and homologues thereof

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0397351A1 (en) * 1989-05-11 1990-11-14 Pfizer Inc. Preparation of diazabicyclic intermediates
US5196548A (en) * 1989-05-11 1993-03-23 Pfizer Inc. Preparation of diazabicyclic Intermediates
AU637099B2 (en) * 1989-05-11 1993-05-20 Pfizer Inc. 2,5-Diazabicyclo-(2.2.1) heptane derivatives

Also Published As

Publication number Publication date
DK114206B (da) 1969-06-09
NL124628C (enExample)
DK114558B (da) 1969-07-14
GB1041863A (en) 1966-09-07
DE1795538A1 (de) 1972-01-13
NL6400946A (enExample) 1964-08-06
SE311661B (enExample) 1969-06-23
US3167561A (en) 1965-01-26
FR1559560A (enExample) 1969-03-14
BR6456585D0 (pt) 1973-08-16

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Legal Events

Date Code Title Description
SH Request for examination between 03.10.1968 and 22.04.1971