CZ297342B6 - Lécivo pro lécení maniodepresivních bipolárních poruch u savcu - Google Patents

Lécivo pro lécení maniodepresivních bipolárních poruch u savcu

Info

Publication number
CZ297342B6
CZ297342B6 CZ0427798A CZ427798A CZ297342B6 CZ 297342 B6 CZ297342 B6 CZ 297342B6 CZ 0427798 A CZ0427798 A CZ 0427798A CZ 427798 A CZ427798 A CZ 427798A CZ 297342 B6 CZ297342 B6 CZ 297342B6
Authority
CZ
Czechia
Prior art keywords
mammals
carbon atoms
general formula
bipolar disorders
medicament
Prior art date
Application number
CZ0427798A
Other languages
English (en)
Other versions
CZ427798A3 (cs
Inventor
P. Shank@Richard
Original Assignee
Ortho-Mcneil Pharmaceutical, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/US1997/009178 external-priority patent/WO1997047135A1/en
Application filed by Ortho-Mcneil Pharmaceutical, Inc. filed Critical Ortho-Mcneil Pharmaceutical, Inc.
Publication of CZ427798A3 publication Critical patent/CZ427798A3/cs
Publication of CZ297342B6 publication Critical patent/CZ297342B6/cs

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/18—Sulfonamides
    • H—ELECTRICITY
    • H04—ELECTRIC COMMUNICATION TECHNIQUE
    • H04N—PICTORIAL COMMUNICATION, e.g. TELEVISION
    • H04N21/00—Selective content distribution, e.g. interactive television or video on demand [VOD]
    • H04N21/40—Client devices specifically adapted for the reception of or interaction with content, e.g. set-top-box [STB]; Operations thereof
    • H04N21/43—Processing of content or additional data, e.g. demultiplexing additional data from a digital video stream; Elementary client operations, e.g. monitoring of home network or synchronising decoder's clock; Client middleware
    • H04N21/442—Monitoring of processes or resources, e.g. detecting the failure of a recording device, monitoring the downstream bandwidth, the number of times a movie has been viewed, the storage space available from the internal hard disk
    • H04N21/44213—Monitoring of end-user related data
    • H04N21/44222—Analytics of user selections, e.g. selection of programs or purchase activity
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/255—Esters, e.g. nitroglycerine, selenocyanates of sulfoxy acids or sulfur analogues thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Social Psychology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Signal Processing (AREA)
  • Computer Networks & Wireless Communication (AREA)
  • Databases & Information Systems (AREA)
  • Multimedia (AREA)
  • Emergency Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyrane Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

Pouzití sulfamátových sloucenin obecného vzorce I, kde X predstavuje skupinu CH.sub.2.n. nebo atom kyslíku; R.sub.1.n. predstavuje atom vodíku nebo alkylskupinu s 1 az 4 atomy uhlíku; a R.sub.2.n., R.sub.3.n., R.sub.4.n., R.sub.5.n. predstavuje nezávisle vzdy atom vodíku nebo nizsí alkylskupinu s 1az 3 atomy uhlíku a kdyz X je atom kyslíku, R.sub.2.n. a R.sub.3.n. a/nebo R.sub.4.n. a R.sub.5.n. mohou spolecne predstavovat methylendioxyskupinu obecného vzorce II, kde R.sub.6.n. a R.sub.7.n. jsou stejné nebo odlisné a kazdý predstavuje atom vodíku nebo nizsí alkylskupinu s 1 az 3 atomy uhlíku nebo R.sub.6.n. a R.sub.7.n. predstavují alkylskupiny, které jsou spolu spojeny za vzniku cyklopentylového nebo cyklohexylového kruhu; zejména topiramatu, pro výrobu léciva pro lécení maniodepresivních bipolárních poruch u savcu.
CZ0427798A 1996-06-28 1997-06-24 Lécivo pro lécení maniodepresivních bipolárních poruch u savcu CZ297342B6 (cs)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US2085096P 1996-06-28 1996-06-28
PCT/US1997/009178 WO1997047135A1 (en) 1996-06-06 1997-06-04 Method and apparatus for automatically determining and dynamically updating user preferences in an entertainment system
US08/881,008 US5753693A (en) 1996-06-28 1997-06-23 Anticonvulsant derivatives useful in treating manic-depressive bipolar disorder

Publications (2)

Publication Number Publication Date
CZ427798A3 CZ427798A3 (cs) 1999-08-11
CZ297342B6 true CZ297342B6 (cs) 2006-11-15

Family

ID=26693960

Family Applications (1)

Application Number Title Priority Date Filing Date
CZ0427798A CZ297342B6 (cs) 1996-06-28 1997-06-24 Lécivo pro lécení maniodepresivních bipolárních poruch u savcu

Country Status (21)

Country Link
US (1) US5753693A (cs)
EP (1) EP0932398B1 (cs)
JP (1) JP2002515875A (cs)
KR (1) KR20000022233A (cs)
CN (1) CN1224350A (cs)
AP (1) AP1401A (cs)
AT (1) ATE330593T1 (cs)
AU (1) AU739363B2 (cs)
BR (1) BR9712783A (cs)
CA (1) CA2258895C (cs)
CZ (1) CZ297342B6 (cs)
DE (1) DE69736183T2 (cs)
ES (1) ES2267144T3 (cs)
HU (1) HUP0003381A3 (cs)
IL (1) IL127714A (cs)
NO (1) NO317641B1 (cs)
NZ (1) NZ333565A (cs)
RU (1) RU2185824C2 (cs)
SK (1) SK180498A3 (cs)
WO (1) WO1998000123A1 (cs)
ZA (1) ZA975773B (cs)

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WO2000032183A1 (en) * 1998-12-03 2000-06-08 Ortho-Mcneil Pharmaceutical, Inc. Topiramate and related derivatives for treating schizophrenia
ES2244411T3 (es) 1999-02-08 2005-12-16 Ortho-Mcneil Pharmaceutical, Inc. Derivados de agente anti-convulsivo utilizados en el tratamiento del autismo.
BR0008477A (pt) 1999-02-24 2002-01-22 Univ Cincinnati Método para tratar um distúrbio de controle do impulso
NZ514813A (en) 1999-04-08 2004-12-24 Ortho Mcneil Pharm Inc Anticonvulsant derivatives useful in treating chronic neurodegenerative disorders
US6420369B1 (en) 1999-05-24 2002-07-16 Ortho-Mcneil Pharmaceutical, Inc. Anticonvulsant derivatives useful in treating dementia
US20080255093A1 (en) * 1999-06-14 2008-10-16 Tam Peter Y Compositions and methods for treating obesity and related disorders
US20080103179A1 (en) * 2006-10-27 2008-05-01 Tam Peter Y Combination Therapy
US7659256B2 (en) * 1999-06-14 2010-02-09 Vivus, Inc. Combination therapy for effecting weight loss and treating obesity
EP2308481B1 (en) 1999-06-14 2015-05-06 Vivus, Inc. Combination therapy for the treatment of hypertension associated with obesity
US7553818B2 (en) * 1999-06-14 2009-06-30 Vivus, Inc. Combination therapy for effecting weight loss and treating obesity
US7674776B2 (en) * 1999-06-14 2010-03-09 Vivus, Inc. Combination therapy for effecting weight loss and treating obesity
US7056890B2 (en) 1999-06-14 2006-06-06 Vivus, Inc. Combination therapy for effecting weight loss and treating obesity
US6191117B1 (en) * 2000-07-10 2001-02-20 Walter E. Kozachuk Methods of producing weight loss and treatment of obesity
JP2004505043A (ja) * 2000-08-02 2004-02-19 オーソ−マクニール・フアーマシユーチカル・インコーポレーテツド うつ病の治療で用いるに有用な抗痙攣性誘導体
AU2002227052A1 (en) 2000-11-30 2002-06-11 University Of Florida Treatments for neurogenetic disorders, impulse control disorders, and wound healing
CA2459146A1 (en) * 2001-08-30 2003-03-13 Ortho-Mcneil Pharmaceutical, Inc. Treatment of dementia and memory disorders with anticonvulsants and acetylcholinesterase inhibitors
US20040235957A1 (en) * 2001-10-12 2004-11-25 David Bleakman Use of sulfonamide derivatives as pharmaceuticals compounds
US20090088443A1 (en) * 2002-02-15 2009-04-02 Julius Remenar Novel crystalline forms of conazoles and methods of making and using the same
US6559293B1 (en) * 2002-02-15 2003-05-06 Transform Pharmaceuticals, Inc. Topiramate sodium trihydrate
US7790905B2 (en) * 2002-02-15 2010-09-07 Mcneil-Ppc, Inc. Pharmaceutical propylene glycol solvate compositions
US7927613B2 (en) 2002-02-15 2011-04-19 University Of South Florida Pharmaceutical co-crystal compositions
US20100311701A1 (en) * 2002-02-15 2010-12-09 Transform Pharmaceuticals, Inc Pharmaceutical Co-Crystal Compositions
JP4906233B2 (ja) 2002-03-01 2012-03-28 ユニバーシティー オブ サウス フロリダ 少なくとも１種の有効薬剤成分を含有する多構成要素固相
US20070059356A1 (en) * 2002-05-31 2007-03-15 Almarsson Oern Pharmaceutical co-crystal compositions of drugs such as carbamazepine, celecoxib, olanzapine, itraconazole, topiramate, modafinil, 5-fluorouracil, hydrochlorothiazide, acetaminophen, aspirin, flurbiprofen, phenytoin and ibuprofen
MXPA05000232A (es) * 2002-06-21 2005-06-17 Transform Pharmaceuticals Inc Composiciones farmaceuticas con disolucion mejorada.
US20040115262A1 (en) * 2002-07-29 2004-06-17 Frank Jao Formulations and dosage forms for controlled delivery of topiramate
US8183290B2 (en) 2002-12-30 2012-05-22 Mcneil-Ppc, Inc. Pharmaceutically acceptable propylene glycol solvate of naproxen
WO2005000294A1 (en) * 2003-06-06 2005-01-06 Pharmacia Corporation Selective inhibitor and an anticonvulsant agent for the treatment of central nervous system disorders
WO2005065648A2 (en) * 2003-12-29 2005-07-21 Alza Corporation, Inc., Novel drug compositions and dosage forms of topiramate
MY147767A (en) * 2004-06-16 2013-01-31 Janssen Pharmaceutica Nv Novel sulfamate and sulfamide derivatives useful for the treatment of epilepsy and related disorders
AR049646A1 (es) * 2004-06-16 2006-08-23 Janssen Pharmaceutica Nv Derivados de sulfamato y sulfamida utiles para el tratamiento de la epilepsia y trastornos relacionados
MX2007002309A (es) * 2004-08-24 2007-10-08 Johnson & Johnson Novedosos derivados de heteroarilsulfamida benzofusionados utiles como agentes anticonvulsivos.
CA2609185A1 (en) * 2005-05-20 2006-11-30 Ahmed F. Abdel-Magid Process for preparation of sulfamide derivatives
US8937096B2 (en) * 2005-12-19 2015-01-20 Janssen Pharmaceutica Nv Use of benzo-fused heterocyle sulfamide derivatives for the treatment of mania and bipolar disorder
US8497298B2 (en) * 2005-12-19 2013-07-30 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels
US8691867B2 (en) * 2005-12-19 2014-04-08 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for the treatment of substance abuse and addiction
AR058389A1 (es) * 2005-12-19 2008-01-30 Janssen Pharmaceutica Nv Uso de derivados heterociclicos benzo-fusionados de sulfamida para el tratamiento de la obesidad
US20070155827A1 (en) * 2005-12-19 2007-07-05 Smith-Swintosky Virginia L Use of benzo-fused heterocycle sulfamide derivatives for the treatment of depression
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Also Published As

Publication number Publication date
BR9712783A (pt) 2000-10-24
CA2258895A1 (en) 1998-01-08
IL127714A0 (en) 1999-10-28
DE69736183T2 (de) 2007-04-26
IL127714A (en) 2004-08-31
JP2002515875A (ja) 2002-05-28
HUP0003381A3 (en) 2001-12-28
KR20000022233A (ko) 2000-04-25
CA2258895C (en) 2006-06-06
ES2267144T3 (es) 2007-03-01
AU739363B2 (en) 2001-10-11
NO986051D0 (no) 1998-12-22
AP1401A (en) 2005-04-29
NO317641B1 (no) 2004-11-29
RU2185824C2 (ru) 2002-07-27
DE69736183D1 (de) 2006-08-03
NZ333565A (en) 2000-07-28
WO1998000123A1 (en) 1998-01-08
AP9801427A0 (en) 1998-12-31
CZ427798A3 (cs) 1999-08-11
US5753693A (en) 1998-05-19
EP0932398A1 (en) 1999-08-04
CN1224350A (zh) 1999-07-28
EP0932398B1 (en) 2006-06-21
AU3409697A (en) 1998-01-21
SK180498A3 (en) 2000-03-13
HUP0003381A2 (hu) 2001-05-28
ZA975773B (en) 1998-12-28
ATE330593T1 (de) 2006-07-15
NO986051L (no) 1999-02-23

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Legal Events

Date Code Title Description
PD00 Pending as of 2000-06-30 in czech republic
MM4A Patent lapsed due to non-payment of fee

Effective date: 20070624