CZ20031860A3 - Derivát benzoylpyridazinu, způsob jeho přípravy, jeho použití a farmaceutický prostředek, který ho obsahuje - Google Patents

Info

Publication number

CZ20031860A3

CZ20031860A3 CZ20031860A CZ20031860A CZ20031860A3 CZ 20031860 A3 CZ20031860 A3 CZ 20031860A3 CZ 20031860 A CZ20031860 A CZ 20031860A CZ 20031860 A CZ20031860 A CZ 20031860A CZ 20031860 A3 CZ20031860 A3 CZ 20031860A3

Authority

CZ

Czechia

Prior art keywords

och

formula

compounds

asthma

inhibitors

Prior art date

2000-12-23

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• 238000002360 preparation method Methods 0.000 title claims description 29
• 238000000034 method Methods 0.000 title claims description 17
• VDWSVBMVZLRATD-UHFFFAOYSA-N phenyl(pyridazin-3-yl)methanone Chemical class C=1C=CN=NC=1C(=O)C1=CC=CC=C1 VDWSVBMVZLRATD-UHFFFAOYSA-N 0.000 title claims description 8
• 230000008569 process Effects 0.000 title claims description 6
• 239000000825 pharmaceutical preparation Substances 0.000 title description 2
• 150000001875 compounds Chemical class 0.000 claims abstract description 218
• 239000002587 phosphodiesterase IV inhibitor Substances 0.000 claims abstract description 11
• -1 COOA 1 Chemical group 0.000 claims description 111
• 239000000203 mixture Substances 0.000 claims description 68
• 239000004480 active ingredient Substances 0.000 claims description 63
• 239000000460 chlorine Substances 0.000 claims description 61
• 239000008194 pharmaceutical composition Substances 0.000 claims description 58
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• ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical compound [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 claims description 15
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