CY1117390T1 - Παραγωγα καρβοξυλικων οξεων με δακτυλιο οξαζολο[4,5-β]πυριδινης - Google Patents
Παραγωγα καρβοξυλικων οξεων με δακτυλιο οξαζολο[4,5-β]πυριδινηςInfo
- Publication number
- CY1117390T1 CY1117390T1 CY20161100150T CY161100150T CY1117390T1 CY 1117390 T1 CY1117390 T1 CY 1117390T1 CY 20161100150 T CY20161100150 T CY 20161100150T CY 161100150 T CY161100150 T CY 161100150T CY 1117390 T1 CY1117390 T1 CY 1117390T1
- Authority
- CY
- Cyprus
- Prior art keywords
- oxazol
- carboxylic acid
- pyridine ring
- acid producers
- producers
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/424—Oxazoles condensed with heterocyclic ring systems, e.g. clavulanic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Diabetes (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Obesity (AREA)
- Epidemiology (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Heart & Thoracic Surgery (AREA)
- Dermatology (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicinal Preparation (AREA)
Abstract
Η εφεύρεση αφορά ενώσεις του τύπου όπου οι Χ, Υ, R1, R2 και R3 έχουν τις διδόμενες σημασίες. Οι ενώσεις του τύπου I είναι κατάλληλες π.χ., για την επούλωση πληγών.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP11305877 | 2011-07-07 | ||
| EP12305525 | 2012-05-11 | ||
| EP12733131.2A EP2729473B1 (de) | 2011-07-07 | 2012-07-06 | Carbonsäurederivate mit einem oxazolo[5,4-b]pyridinring |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CY1117390T1 true CY1117390T1 (el) | 2017-04-26 |
Family
ID=46466551
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CY20161100150T CY1117390T1 (el) | 2011-07-07 | 2016-02-24 | Παραγωγα καρβοξυλικων οξεων με δακτυλιο οξαζολο[4,5-β]πυριδινης |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US8580816B2 (el) |
| EP (1) | EP2729473B1 (el) |
| JP (1) | JP5984925B2 (el) |
| KR (1) | KR20140061384A (el) |
| CN (1) | CN103781790B (el) |
| AU (1) | AU2012280206B2 (el) |
| BR (1) | BR112014000100A2 (el) |
| CA (1) | CA2841220C (el) |
| CY (1) | CY1117390T1 (el) |
| DK (1) | DK2729473T3 (el) |
| ES (1) | ES2562852T3 (el) |
| HK (1) | HK1192239A1 (el) |
| HR (1) | HRP20160167T1 (el) |
| HU (1) | HUE026432T2 (el) |
| MX (1) | MX365931B (el) |
| MY (1) | MY164133A (el) |
| PL (1) | PL2729473T3 (el) |
| PT (1) | PT2729473E (el) |
| RU (1) | RU2609002C2 (el) |
| SI (1) | SI2729473T1 (el) |
| WO (1) | WO2013004826A1 (el) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8907093B2 (en) * | 2011-07-07 | 2014-12-09 | Sanofi | Carboxylic acid derivatives having an oxazolo[4,5-c]pyridine ring |
| US9321787B2 (en) | 2011-07-07 | 2016-04-26 | Sanofi | Carboxylic acid derivatives having an oxazolo[5,4-d]pyrimidine ring |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NO143535C (no) * | 1972-06-14 | 1981-03-04 | Merck & Co Inc | Analogifremgangsmaate ved fremstilling av terapeutisk aktive oxazolopyridiner |
| BR0209645A (pt) * | 2001-05-14 | 2004-07-06 | Novartis Ag | Oxazolo- e furopirimidinas e seu uso como medicamentos |
| CA2524054C (en) * | 2003-05-19 | 2012-04-24 | Irm Llc | Immunosuppressant compounds and compositions |
| JP2009520688A (ja) * | 2005-11-23 | 2009-05-28 | エピックス デラウェア， インコーポレイテッド | Ｓ１ｐ受容体調節化合物およびそれらの使用 |
| EP1900729A1 (en) * | 2006-09-15 | 2008-03-19 | Novartis AG | Benzoxazoles and oxazolopyridines being useful as Janus kinases inhibitors |
| AU2007227278B2 (en) | 2007-03-21 | 2014-09-11 | Epix Pharmaceuticals, Inc. | SIP receptor modulating compounds and use thereof |
| WO2009155017A2 (en) | 2008-05-30 | 2009-12-23 | Merck & Co., Inc. | Novel substituted azabenzoxazoles |
| TW201000099A (en) | 2008-06-20 | 2010-01-01 | Amgen Inc | S1P1 receptor agonists and use thereof |
| AU2009270511B2 (en) | 2008-07-15 | 2013-07-18 | Sanofi | Oxazolopyrimidines as Edg-1 receptor agonists |
| US8907093B2 (en) * | 2011-07-07 | 2014-12-09 | Sanofi | Carboxylic acid derivatives having an oxazolo[4,5-c]pyridine ring |
-
2012
- 2012-06-25 US US13/532,255 patent/US8580816B2/en active Active
- 2012-07-06 PL PL12733131T patent/PL2729473T3/pl unknown
- 2012-07-06 CN CN201280043621.7A patent/CN103781790B/zh active Active
- 2012-07-06 ES ES12733131.2T patent/ES2562852T3/es active Active
- 2012-07-06 WO PCT/EP2012/063297 patent/WO2013004826A1/de active Application Filing
- 2012-07-06 BR BR112014000100A patent/BR112014000100A2/pt not_active IP Right Cessation
- 2012-07-06 AU AU2012280206A patent/AU2012280206B2/en not_active Ceased
- 2012-07-06 HU HUE12733131A patent/HUE026432T2/en unknown
- 2012-07-06 KR KR1020147003226A patent/KR20140061384A/ko not_active Application Discontinuation
- 2012-07-06 PT PT127331312T patent/PT2729473E/pt unknown
- 2012-07-06 RU RU2014104232A patent/RU2609002C2/ru not_active IP Right Cessation
- 2012-07-06 MY MYPI2014000006A patent/MY164133A/en unknown
- 2012-07-06 MX MX2014000024A patent/MX365931B/es active IP Right Grant
- 2012-07-06 CA CA2841220A patent/CA2841220C/en not_active Expired - Fee Related
- 2012-07-06 SI SI201230458T patent/SI2729473T1/sl unknown
- 2012-07-06 DK DK12733131.2T patent/DK2729473T3/en active
- 2012-07-06 EP EP12733131.2A patent/EP2729473B1/de active Active
- 2012-07-06 JP JP2014517829A patent/JP5984925B2/ja active Active
-
2014
- 2014-06-13 HK HK14105591.6A patent/HK1192239A1/zh not_active IP Right Cessation
-
2016
- 2016-02-16 HR HRP20160167TT patent/HRP20160167T1/hr unknown
- 2016-02-24 CY CY20161100150T patent/CY1117390T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| MX2014000024A (es) | 2014-02-27 |
| KR20140061384A (ko) | 2014-05-21 |
| EP2729473B1 (de) | 2015-11-25 |
| AU2012280206A1 (en) | 2014-01-23 |
| RU2014104232A (ru) | 2015-08-20 |
| CA2841220A1 (en) | 2013-01-10 |
| HRP20160167T1 (hr) | 2016-03-11 |
| AU2012280206B2 (en) | 2016-07-28 |
| EP2729473A1 (de) | 2014-05-14 |
| WO2013004826A1 (de) | 2013-01-10 |
| CN103781790A (zh) | 2014-05-07 |
| US20130023557A1 (en) | 2013-01-24 |
| CA2841220C (en) | 2019-07-30 |
| HK1192239A1 (zh) | 2014-08-15 |
| JP2014518247A (ja) | 2014-07-28 |
| HUE026432T2 (en) | 2016-05-30 |
| MX365931B (es) | 2019-06-20 |
| CN103781790B (zh) | 2016-04-27 |
| ES2562852T3 (es) | 2016-03-08 |
| PT2729473E (pt) | 2016-03-22 |
| RU2609002C2 (ru) | 2017-01-30 |
| DK2729473T3 (en) | 2016-02-29 |
| US8580816B2 (en) | 2013-11-12 |
| BR112014000100A2 (pt) | 2017-01-10 |
| JP5984925B2 (ja) | 2016-09-06 |
| SI2729473T1 (sl) | 2016-03-31 |
| PL2729473T3 (pl) | 2016-05-31 |
| MY164133A (en) | 2017-11-30 |
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