CY1112643T1 - Διενυδρη υδροχλωρικη ναλμεφαινη - Google Patents
Διενυδρη υδροχλωρικη ναλμεφαινηInfo
- Publication number
- CY1112643T1 CY1112643T1 CY20121100278T CY121100278T CY1112643T1 CY 1112643 T1 CY1112643 T1 CY 1112643T1 CY 20121100278 T CY20121100278 T CY 20121100278T CY 121100278 T CY121100278 T CY 121100278T CY 1112643 T1 CY1112643 T1 CY 1112643T1
- Authority
- CY
- Cyprus
- Prior art keywords
- nalmefein
- hydrochlorine
- hydrochloric
- nalmefine
- hydrochloride dihydrate
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D489/00—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
- C07D489/06—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: with a hetero atom directly attached in position 14
- C07D489/08—Oxygen atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4866—Organic macromolecular compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
- A61K9/7084—Transdermal patches having a drug layer or reservoir, and one or more separate drug-free skin-adhesive layers, e.g. between drug reservoir and skin, or surrounding the drug reservoir; Liquid-filled reservoir patches
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Neurology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Addiction (AREA)
- Dermatology (AREA)
- Epidemiology (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Steroid Compounds (AREA)
Abstract
Η παρούσα εφεύρεση αφορά σε διένυδρη υδροχλωρική Ναλμεφαίνη, μεθόδους βιομηχανικής κατασκευής διενύδρου υδροχλωρικής Ναλμεφαίνης, φαρμακευτική σύνθεση που περιλαμβάνει διένυδρη υδροχλωρική Ναλμεφαίνη και μέθοδο θεραπείας που περιλαμβάνει χορήγηση διενύδρου υδροχλωρικής Ναλμεφαίνης.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US12013208P | 2008-12-05 | 2008-12-05 | |
DKPA200801729 | 2008-12-05 | ||
EP09771286A EP2300479B1 (en) | 2008-12-05 | 2009-12-04 | Nalmefene hydrochloride dihydrate |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1112643T1 true CY1112643T1 (el) | 2016-02-10 |
Family
ID=41571731
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20121100278T CY1112643T1 (el) | 2008-12-05 | 2012-03-15 | Διενυδρη υδροχλωρικη ναλμεφαινη |
CY20141100563T CY1115381T1 (el) | 2008-12-05 | 2014-07-25 | Διενυδρη υδροχλωρικη ναλμεφαινη |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20141100563T CY1115381T1 (el) | 2008-12-05 | 2014-07-25 | Διενυδρη υδροχλωρικη ναλμεφαινη |
Country Status (31)
Country | Link |
---|---|
US (2) | US8530495B2 (el) |
EP (2) | EP2300479B1 (el) |
JP (3) | JP6055183B2 (el) |
KR (2) | KR20170008893A (el) |
CN (2) | CN102325778B (el) |
AR (1) | AR074507A1 (el) |
AT (1) | ATE546453T1 (el) |
AU (1) | AU2009321898B2 (el) |
BR (1) | BRPI0922774B8 (el) |
CA (1) | CA2744932C (el) |
CL (1) | CL2011001331A1 (el) |
CO (1) | CO6362012A2 (el) |
CY (2) | CY1112643T1 (el) |
DK (2) | DK2441766T3 (el) |
EA (1) | EA018948B1 (el) |
ES (2) | ES2488165T3 (el) |
HK (1) | HK1205108A1 (el) |
HR (2) | HRP20120247T1 (el) |
IL (1) | IL213112A (el) |
MX (1) | MX2011005865A (el) |
MY (1) | MY149028A (el) |
NZ (1) | NZ593874A (el) |
PL (2) | PL2441766T3 (el) |
PT (2) | PT2441766E (el) |
RS (2) | RS52255B (el) |
SG (1) | SG171910A1 (el) |
SI (2) | SI2300479T1 (el) |
SM (2) | SMT201200014B (el) |
TW (1) | TWI465450B (el) |
UA (1) | UA102128C2 (el) |
WO (1) | WO2010063292A1 (el) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
UA102128C2 (en) * | 2008-12-05 | 2013-06-10 | Х. Луннбек А/С | Nalmefene hydrochloride dihydrate |
JP2019031524A (ja) * | 2008-12-05 | 2019-02-28 | ハー・ルンドベック・アクチエゼルスカベット | ナルメフェン塩酸塩二水和物 |
TWI560170B (en) * | 2011-12-06 | 2016-12-01 | Lundbeck & Co As H | Process for recovery of nalmefene hydrochloride |
US20140155608A1 (en) | 2012-05-03 | 2014-06-05 | H. Lundbeck A/S | Method for the manufacturing of naltrexone |
US20140005216A1 (en) | 2012-06-27 | 2014-01-02 | H. Lundbeck A/S | Nalmefene for reduction of alcohol consumption in specific target populations |
JP6419780B2 (ja) * | 2013-04-17 | 2018-11-07 | ハー・ルンドベック・アクチエゼルスカベット | 睡眠障害患者の治療のためのナルメフェン |
US20160058754A1 (en) * | 2013-04-17 | 2016-03-03 | H. Lundbeck A/S | Nalmefene for Treatment of Patients with Anxiety Disorder |
AR096851A1 (es) * | 2013-07-11 | 2016-02-03 | H Lundbeck As | Sales que no forman hidratos ni solvatos de nalmefeno |
ES2742888T3 (es) | 2014-04-22 | 2020-02-17 | Otsuka Pharma Co Ltd | Combinación de brexpiprazol y nalmefeno y su uso para tratar trastornos relacionados con una sustancia |
TWI729644B (zh) | 2014-06-12 | 2021-06-01 | 美商西爾拉癌症醫學公司 | N-(氰基甲基)-4-(2-(4-𠰌啉基苯基胺基)嘧啶-4-基)苯甲醯胺 |
CN105646508B (zh) * | 2016-02-17 | 2018-02-27 | 南京卓康医药科技有限公司 | 一种盐酸纳美芬一水合物的制备方法 |
WO2019022274A1 (ko) * | 2017-07-28 | 2019-01-31 | 동아대학교 산학협력단 | Pauf 단백질에 특이적으로 결합하는 항체 및 이의 용도 |
US10927121B1 (en) | 2019-12-20 | 2021-02-23 | Southwest Research Institute | Technologies for removing residual solvent from nalmefene hydrochloride and producing crystalline nalmefene hydrochloride monohydrate, monosolvate, or crystalline nalmefene hydrochloride dihydrate |
CN111875530A (zh) * | 2020-08-17 | 2020-11-03 | 浙江朗华制药有限公司 | 一种普拉西坦水合物晶体及其制备方法 |
WO2022165040A1 (en) | 2021-01-28 | 2022-08-04 | Rhodes Technologies | Process for crystallizing nalmefene hydrochloride |
CN113354652A (zh) * | 2021-06-24 | 2021-09-07 | 无锡济煜山禾药业股份有限公司 | 一种盐酸纳美芬合成方法 |
CN117986261B (zh) * | 2024-04-02 | 2024-06-18 | 成都瑞尔医药科技有限公司 | 一种盐酸纳美芬母液的回收套用方法 |
Family Cites Families (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4535157A (en) | 1983-11-01 | 1985-08-13 | Key Pharmaceuticals, Inc. | Process for making 6-desoxy-6-methylenenaloxone and 6-desoxy-6-methylenenaltrexone |
US4751307A (en) | 1985-01-17 | 1988-06-14 | Mallinckrodt, Inc. | Wittig-reaction processes |
JPH07206857A (ja) * | 1993-12-28 | 1995-08-08 | Synthelabo Sa | アルフゾシン塩酸塩の二水和物 |
US6262067B1 (en) * | 1999-06-22 | 2001-07-17 | Pfizer Inc. | Polymorphs of a crystalline azo-bicyclo 2,2,2 OCT-3-yl amine dihydrochloride and their pharmaceutical compositions |
ES2177373B1 (es) * | 1999-11-26 | 2003-11-01 | Astur Pharma Sa | Preparacion de azitromicina en su forma no cristalina |
CH693586A8 (de) * | 2002-10-14 | 2003-12-15 | Roche Consumer Health Ag | Darreichungsform von Ibuprofen-Natrium. |
FR2861299B1 (fr) * | 2003-10-28 | 2006-01-27 | Pf Medicament | Compositions pharmaceutiques a base de derives d'idasoxan sous formes polymorphes |
DK1708690T3 (en) * | 2003-11-17 | 2016-11-07 | Biomarin Pharm Inc | TREATMENT OF PHENYLKETONURI WITH BH4 |
MY139797A (en) * | 2004-11-29 | 2009-10-30 | Kowa Co | (s)-(-)-1-(4-fluoroisoquinolin-5-yl)sulfonyl-2-methyl-1, 4-homopiperazine hydrochloride dihydrate |
CN100536848C (zh) * | 2005-07-13 | 2009-09-09 | 北京易明康元医药科技有限公司 | 稳定的盐酸纳美芬注射液及其制备方法 |
GB2447013A (en) | 2007-03-01 | 2008-09-03 | Reckitt Benckiser Healthcare | Analgesic composition containing buprenorphone and nalmefene |
GB2447016A (en) | 2007-03-01 | 2008-09-03 | Reckitt Benckiser Healthcare | Buprenorphine/naloxone compositions |
CA2707757C (en) | 2007-03-06 | 2017-01-03 | Peter X. Wang | Process for the preparation of quaternary n-alkyl morphinan alkaloid salts |
US8399475B2 (en) * | 2007-04-12 | 2013-03-19 | Mallinckrodt Llc | Crystalline and amorphous forms of naltrexone hydrochloride |
UA102128C2 (en) * | 2008-12-05 | 2013-06-10 | Х. Луннбек А/С | Nalmefene hydrochloride dihydrate |
-
2009
- 2009-04-12 UA UAA201108231A patent/UA102128C2/ru unknown
- 2009-12-04 JP JP2011538838A patent/JP6055183B2/ja active Active
- 2009-12-04 AU AU2009321898A patent/AU2009321898B2/en not_active Ceased
- 2009-12-04 EP EP09771286A patent/EP2300479B1/en active Active
- 2009-12-04 KR KR1020177001191A patent/KR20170008893A/ko not_active Application Discontinuation
- 2009-12-04 ES ES12150266.0T patent/ES2488165T3/es active Active
- 2009-12-04 MY MYPI2011002518A patent/MY149028A/en unknown
- 2009-12-04 MX MX2011005865A patent/MX2011005865A/es active IP Right Grant
- 2009-12-04 RS RS20120126A patent/RS52255B/en unknown
- 2009-12-04 SI SI200930215T patent/SI2300479T1/sl unknown
- 2009-12-04 PT PT121502660T patent/PT2441766E/pt unknown
- 2009-12-04 CN CN200980156373.5A patent/CN102325778B/zh active Active
- 2009-12-04 WO PCT/DK2009/050320 patent/WO2010063292A1/en active Application Filing
- 2009-12-04 PT PT09771286T patent/PT2300479E/pt unknown
- 2009-12-04 US US13/132,494 patent/US8530495B2/en active Active
- 2009-12-04 SG SG2011040102A patent/SG171910A1/en unknown
- 2009-12-04 RS RS20140376A patent/RS53415B/en unknown
- 2009-12-04 DK DK12150266.0T patent/DK2441766T3/da active
- 2009-12-04 EP EP12150266.0A patent/EP2441766B1/en active Active
- 2009-12-04 KR KR1020117012659A patent/KR20110089333A/ko active Search and Examination
- 2009-12-04 CN CN201410323051.8A patent/CN104211707B/zh active Active
- 2009-12-04 BR BRPI0922774A patent/BRPI0922774B8/pt active IP Right Grant
- 2009-12-04 AT AT09771286T patent/ATE546453T1/de active
- 2009-12-04 NZ NZ593874A patent/NZ593874A/xx unknown
- 2009-12-04 SI SI200930985T patent/SI2441766T1/sl unknown
- 2009-12-04 DK DK09771286.3T patent/DK2300479T3/da active
- 2009-12-04 ES ES09771286T patent/ES2380297T3/es active Active
- 2009-12-04 CA CA2744932A patent/CA2744932C/en active Active
- 2009-12-04 PL PL12150266T patent/PL2441766T3/pl unknown
- 2009-12-04 EA EA201170753A patent/EA018948B1/ru not_active IP Right Cessation
- 2009-12-04 PL PL09771286T patent/PL2300479T3/pl unknown
- 2009-12-07 AR ARP090104739A patent/AR074507A1/es unknown
- 2009-12-07 TW TW098141677A patent/TWI465450B/zh not_active IP Right Cessation
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2011
- 2011-05-24 IL IL213112A patent/IL213112A/en active IP Right Grant
- 2011-06-01 CO CO11067790A patent/CO6362012A2/es not_active Application Discontinuation
- 2011-06-03 CL CL2011001331A patent/CL2011001331A1/es unknown
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2012
- 2012-03-15 CY CY20121100278T patent/CY1112643T1/el unknown
- 2012-03-16 HR HRP20120247AT patent/HRP20120247T1/hr unknown
- 2012-04-04 SM SM201200014T patent/SMT201200014B/it unknown
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2013
- 2013-06-25 US US13/926,427 patent/US8754217B2/en active Active
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2014
- 2014-07-08 HR HRP20140648AT patent/HRP20140648T1/hr unknown
- 2014-07-25 CY CY20141100563T patent/CY1115381T1/el unknown
- 2014-08-18 SM SM201400113T patent/SMT201400113B/xx unknown
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2015
- 2015-02-16 JP JP2015028004A patent/JP6591759B2/ja active Active
- 2015-06-10 HK HK15105492.5A patent/HK1205108A1/xx not_active IP Right Cessation
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2016
- 2016-09-07 JP JP2016175002A patent/JP6591944B2/ja active Active
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