CY1105892T1 - Θepαπεια του ξανθωματος με παραγωγα αζετιδινονης ως αναστολεις απορροφησης στepολης - Google Patents

Θepαπεια του ξανθωματος με παραγωγα αζετιδινονης ως αναστολεις απορροφησης στepολης

Info

Publication number
CY1105892T1
CY1105892T1 CY20061101869T CY061101869T CY1105892T1 CY 1105892 T1 CY1105892 T1 CY 1105892T1 CY 20061101869 T CY20061101869 T CY 20061101869T CY 061101869 T CY061101869 T CY 061101869T CY 1105892 T1 CY1105892 T1 CY 1105892T1
Authority
CY
Cyprus
Prior art keywords
treatment
stepolis
xanthoma
absorption inhibitors
azetidinone derivatives
Prior art date
Application number
CY20061101869T
Other languages
English (en)
Inventor
Harry R. Davis
Original Assignee
Schering Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corporation filed Critical Schering Corporation
Publication of CY1105892T1 publication Critical patent/CY1105892T1/el

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Η παρούσα εφεύρεση παρέχει θεραπευτικούς συνδυασμούς και μεθόδους που περιέχουν τουλάχιστον έναν αναστολέα απορρόφησης στερόλης ή 5α-στανόλης οι οποίοι μπορούν να είναι χρήσιμοι στη θεραπεία των ξανθωμάτων.
CY20061101869T 2001-09-21 2006-12-29 Θepαπεια του ξανθωματος με παραγωγα αζετιδινονης ως αναστολεις απορροφησης στepολης CY1105892T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32394201P 2001-09-21 2001-09-21
PCT/US2002/029652 WO2003026643A2 (en) 2001-09-21 2002-09-19 Treatment of xanthoma with azetidinone derivatives as sterol absorption inhibitors

Publications (1)

Publication Number Publication Date
CY1105892T1 true CY1105892T1 (el) 2011-02-02

Family

ID=23261375

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20061101869T CY1105892T1 (el) 2001-09-21 2006-12-29 Θepαπεια του ξανθωματος με παραγωγα αζετιδινονης ως αναστολεις απορροφησης στepολης

Country Status (13)

Country Link
US (2) US7132415B2 (el)
EP (1) EP1429756B1 (el)
JP (1) JP2005504091A (el)
AT (1) ATE345793T1 (el)
AU (1) AU2002336609B2 (el)
CA (1) CA2460340C (el)
CY (1) CY1105892T1 (el)
DE (1) DE60216300T2 (el)
DK (1) DK1429756T3 (el)
ES (1) ES2272776T3 (el)
MX (1) MXPA04002573A (el)
PT (1) PT1429756E (el)
WO (1) WO2003026643A2 (el)

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CN104023718B (zh) 2011-10-28 2017-04-05 鲁美纳医药公司 用于治疗高胆血症和胆汁淤积性肝病的胆汁酸再循环抑制剂
AU2014228850A1 (en) 2013-03-15 2015-10-29 Lumena Pharmaceuticals Llc Bile acid recycling inhibitors for treatment of primary sclerosing cholangitis and inflammatory bowel disease
AU2014229050A1 (en) 2013-03-15 2015-10-22 Lumena Pharmaceuticals Llc Bile acid recycling inhibitors for treatment of Barrett's esophagus and gastroesophageal reflux disease
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AU2002336609B2 (en) 2006-08-24
US7132415B2 (en) 2006-11-07
EP1429756B1 (en) 2006-11-22
US20030119809A1 (en) 2003-06-26
DE60216300T2 (de) 2007-06-28
ATE345793T1 (de) 2006-12-15
MXPA04002573A (es) 2004-06-18
WO2003026643A3 (en) 2003-07-03
ES2272776T3 (es) 2007-05-01
PT1429756E (pt) 2007-01-31
CA2460340A1 (en) 2003-04-03
US20060217363A1 (en) 2006-09-28
DE60216300D1 (de) 2007-01-04
WO2003026643A2 (en) 2003-04-03
JP2005504091A (ja) 2005-02-10
DK1429756T3 (da) 2007-03-19
EP1429756A2 (en) 2004-06-23

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