CY1105228T1 - Φαρμακευτικο αιωρημα πepιλαμβανον ημι-ενυδρη νεβιραπινη - Google Patents

Φαρμακευτικο αιωρημα πepιλαμβανον ημι-ενυδρη νεβιραπινη

Info

Publication number
CY1105228T1
CY1105228T1 CY20061101147T CY061101147T CY1105228T1 CY 1105228 T1 CY1105228 T1 CY 1105228T1 CY 20061101147 T CY20061101147 T CY 20061101147T CY 061101147 T CY061101147 T CY 061101147T CY 1105228 T1 CY1105228 T1 CY 1105228T1
Authority
CY
Cyprus
Prior art keywords
pepilamvanone
nebirapine
hydric
semi
pharmaceutical suspension
Prior art date
Application number
CY20061101147T
Other languages
English (en)
Inventor
Karl Georg Grozinger
Amale A. Hawi
Original Assignee
Boehringer Ingelheim Pharmaceuticals Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22006658&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY1105228(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Pharmaceuticals Inc. filed Critical Boehringer Ingelheim Pharmaceuticals Inc.
Publication of CY1105228T1 publication Critical patent/CY1105228T1/el

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A61K31/55131,4-Benzodiazepines, e.g. diazepam or clozapine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Virology (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Steroid Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Υδατικό φαρμακευτικό αιώρημα αποτελούμενο ουσιαστικώς από ημι-ένυδρη νεβιραπίνη έχουσα διάμετρο σωματιδίων μεγέθους από 1 έως 150 μm περίπου.
CY20061101147T 1997-08-25 2006-08-11 Φαρμακευτικο αιωρημα πepιλαμβανον ημι-ενυδρη νεβιραπινη CY1105228T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US5680397P 1997-08-25 1997-08-25
PCT/US1998/016581 WO1999009990A1 (en) 1997-08-25 1998-08-11 Pharmaceutical suspension comprising nevirapine hemihydrate

Publications (1)

Publication Number Publication Date
CY1105228T1 true CY1105228T1 (el) 2010-03-03

Family

ID=22006658

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20061101147T CY1105228T1 (el) 1997-08-25 2006-08-11 Φαρμακευτικο αιωρημα πepιλαμβανον ημι-ενυδρη νεβιραπινη

Country Status (38)

Country Link
US (2) US6172059B1 (el)
EP (1) EP1019058B1 (el)
JP (1) JP3472261B2 (el)
KR (1) KR100426516B1 (el)
CN (1) CN1197578C (el)
AR (2) AR016869A1 (el)
AT (1) ATE326971T1 (el)
AU (1) AU742761B2 (el)
BG (1) BG64337B1 (el)
BR (1) BR9811994B1 (el)
CA (1) CA2301646C (el)
CL (1) CL2008003111A1 (el)
CO (1) CO4970742A1 (el)
CY (1) CY1105228T1 (el)
CZ (1) CZ290667B6 (el)
DE (1) DE69834655T2 (el)
DK (1) DK1019058T3 (el)
EG (1) EG24075A (el)
ES (1) ES2265666T3 (el)
HK (1) HK1027975A1 (el)
HR (1) HRP980461B1 (el)
HU (1) HU226063B1 (el)
ID (1) ID21650A (el)
IL (1) IL134185A (el)
MY (1) MY122272A (el)
NO (1) NO326226B1 (el)
NZ (1) NZ503414A (el)
PE (1) PE105799A1 (el)
PL (1) PL192361B1 (el)
PT (1) PT1019058E (el)
RS (1) RS49808B (el)
RU (1) RU2196584C2 (el)
SA (1) SA98190680B1 (el)
TR (1) TR200000490T2 (el)
TW (1) TW450812B (el)
UA (1) UA44370C2 (el)
WO (1) WO1999009990A1 (el)
ZA (1) ZA987623B (el)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002092095A1 (en) * 2001-05-11 2002-11-21 Boehringer Ingelheim International Gmbh Use of nevirapine to treat or prevent lipid pathology in patients with hiv that is resistant to nevirapine
WO2003091290A1 (en) * 2002-04-23 2003-11-06 Boehringer Ingelheim Pharmaceuticals, Inc. Method for reduction of residual organic solvent in carbomer
ATE484284T1 (de) * 2005-08-31 2010-10-15 Cipla Ltd Pharmazeutische kombinationen mit lamivudin, stavudin und nevirapin
WO2010006697A2 (en) * 2008-06-30 2010-01-21 Tibotec Pharmaceuticals Powders for reconstitution
DE112010004065T5 (de) * 2009-11-10 2012-10-25 North West University Verfahren zur Erhöhung der Löslichkeit einer Transkriptaseinhibitor-Zusammensetzung
CN102725293A (zh) * 2009-12-17 2012-10-10 西北大学 奈韦拉平的多晶型形式及其制备

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5366972A (en) 1989-04-20 1994-11-22 Boehringer Ingelheim Pharmaceuticals, Inc. 5,11-dihydro-6H-dipyrido(3,2-B:2',3'-E)(1,4)diazepines and their use in the prevention or treatment of HIV infection
CA2030056C (en) * 1989-11-17 1995-10-17 Karl D. Hargrave 5,11-dihydro-6h-dipyrido[3,2-b:2',3'-e][1,4]diazepines and their use in the prevention or treatment of hiv infection
US5571912A (en) * 1990-10-19 1996-11-05 Boehringer Ingelheim Pharmaceuticals, Inc. Method for the preparation of 5,11-dihydro-6h-dipyrido [3,2-b:2',3'-e][1,4]diazepines
DE4403311C1 (de) * 1994-02-03 1995-04-20 Boehringer Ingelheim Kg Verfahren zur Herstellung von Nevirapine (11-Cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3,2-b:2',3'-e][1,4-diazepin]-6-on)

Also Published As

Publication number Publication date
ID21650A (id) 1999-07-08
ATE326971T1 (de) 2006-06-15
AU742761B2 (en) 2002-01-10
CZ290667B6 (cs) 2002-09-11
BR9811994B1 (pt) 2013-11-19
AR083451A2 (es) 2013-02-27
NZ503414A (en) 2002-11-26
AR016869A1 (es) 2001-08-01
PL192361B1 (pl) 2006-10-31
TW450812B (en) 2001-08-21
UA44370C2 (uk) 2002-02-15
MY122272A (en) 2006-04-29
HRP980461A2 (en) 1999-06-30
EP1019058B1 (en) 2006-05-24
YU9800A (sh) 2001-12-26
EG24075A (en) 2008-05-11
HUP0003093A2 (hu) 2001-08-28
HRP980461B1 (en) 2002-08-31
US6172059B1 (en) 2001-01-09
KR20010023257A (ko) 2001-03-26
PL338828A1 (en) 2000-11-20
RS49808B (sr) 2008-08-07
NO20000906L (no) 2000-02-24
NO20000906D0 (no) 2000-02-24
CZ2000694A3 (cs) 2000-09-13
DE69834655D1 (de) 2006-06-29
KR100426516B1 (ko) 2004-04-13
CA2301646A1 (en) 1999-03-04
CA2301646C (en) 2008-11-18
BG64337B1 (bg) 2004-10-29
HU226063B1 (hu) 2008-04-28
CO4970742A1 (es) 2000-11-07
IL134185A0 (en) 2001-04-30
SA98190680B1 (ar) 2006-04-04
RU2196584C2 (ru) 2003-01-20
NO326226B1 (no) 2008-10-20
PT1019058E (pt) 2006-08-31
CL2008003111A1 (es) 2009-09-11
PE105799A1 (es) 1999-11-16
ES2265666T3 (es) 2007-02-16
EP1019058A1 (en) 2000-07-19
WO1999009990A1 (en) 1999-03-04
US6255481B1 (en) 2001-07-03
JP2001513564A (ja) 2001-09-04
HK1027975A1 (en) 2001-02-02
EP1019058A4 (en) 2004-11-10
DE69834655T2 (de) 2006-12-14
CN1268055A (zh) 2000-09-27
ZA987623B (en) 2000-03-22
CN1197578C (zh) 2005-04-20
DK1019058T3 (da) 2006-06-12
BG104133A (en) 2000-08-31
IL134185A (en) 2005-11-20
TR200000490T2 (tr) 2000-08-21
JP3472261B2 (ja) 2003-12-02
AU8777198A (en) 1999-03-16
BR9811994A (pt) 2000-09-05

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