CU24476B1 - Nueva triterpenona c-3 con derivados de amida inversa c-17 como inhibidores de vih - Google Patents

Nueva triterpenona c-3 con derivados de amida inversa c-17 como inhibidores de vih

Info

Publication number
CU24476B1
CU24476B1 CU2017000102A CU20170102A CU24476B1 CU 24476 B1 CU24476 B1 CU 24476B1 CU 2017000102 A CU2017000102 A CU 2017000102A CU 20170102 A CU20170102 A CU 20170102A CU 24476 B1 CU24476 B1 CU 24476B1
Authority
CU
Cuba
Prior art keywords
triterpenone
new
amide derivatives
hiv inhibitors
inverse amide
Prior art date
Application number
CU2017000102A
Other languages
English (en)
Other versions
CU20170102A7 (es
Inventor
Reddy Kasireddy Bhaskar
Krupadanam Gazula Levi David
Reddy Adulla Panduranga
Reddy Bandi Parthasaradhi
Reddy Kura Rathnakar
Subrahmanyam Lanka Vl
Original Assignee
Dfh Therapeutics Inc
Hetero Labs Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=57153504&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CU24476(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dfh Therapeutics Inc, Hetero Labs Ltd filed Critical Dfh Therapeutics Inc
Publication of CU20170102A7 publication Critical patent/CU20170102A7/es
Publication of CU24476B1 publication Critical patent/CU24476B1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J63/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • C07J63/008—Expansion of ring D by one atom, e.g. D homo steroids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Virology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • AIDS & HIV (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

<p>La invención se refiere a una nueva triterpenona C-3 con derivados amida inversa C-17 y compuestos relacionados útiles para el tratamiento terapéutico de enfermedades virales y particularmente enfermedades mediadas por VIH. </p>
CU2017000102A 2015-02-09 2016-02-09 Nueva triterpenona c-3 con derivados de amida inversa c-17 como inhibidores de vih CU24476B1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN623CH2015 2015-02-09
PCT/IB2016/000811 WO2016178092A2 (en) 2015-02-09 2016-02-09 C-3 novel triterpenone with c-28 reverse amide derivatives as hiv inhibitors

Publications (2)

Publication Number Publication Date
CU20170102A7 CU20170102A7 (es) 2018-01-10
CU24476B1 true CU24476B1 (es) 2020-03-04

Family

ID=57153504

Family Applications (1)

Application Number Title Priority Date Filing Date
CU2017000102A CU24476B1 (es) 2015-02-09 2016-02-09 Nueva triterpenona c-3 con derivados de amida inversa c-17 como inhibidores de vih

Country Status (22)

Country Link
US (3) US10533035B2 (es)
EP (1) EP3256483B1 (es)
JP (1) JP2018505216A (es)
KR (1) KR20170110143A (es)
CN (1) CN107428797A (es)
AU (1) AU2016258274B2 (es)
BR (1) BR112017017109A2 (es)
CA (1) CA2975359A1 (es)
CL (1) CL2017002034A1 (es)
CO (1) CO2017008765A2 (es)
CU (1) CU24476B1 (es)
DK (1) DK3256483T3 (es)
EA (1) EA033264B1 (es)
ES (1) ES2780649T3 (es)
IL (1) IL253844A0 (es)
MA (1) MA40886B1 (es)
MX (1) MX2017010297A (es)
PE (1) PE20171433A1 (es)
PH (1) PH12017550077A1 (es)
SG (1) SG11201706189PA (es)
WO (1) WO2016178092A2 (es)
ZA (1) ZA201705253B (es)

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Also Published As

Publication number Publication date
WO2016178092A3 (en) 2017-01-05
WO2016178092A8 (en) 2017-09-21
EP3256483A2 (en) 2017-12-20
CL2017002034A1 (es) 2018-04-27
CA2975359A1 (en) 2016-11-10
WO2016178092A2 (en) 2016-11-10
CN107428797A (zh) 2017-12-01
ES2780649T3 (es) 2020-08-26
JP2018505216A (ja) 2018-02-22
MA40886B1 (fr) 2020-03-31
ZA201705253B (en) 2020-01-29
EA201791807A1 (ru) 2018-01-31
US10533035B2 (en) 2020-01-14
DK3256483T3 (da) 2020-03-23
EA033264B1 (ru) 2019-09-30
AU2016258274B2 (en) 2019-12-05
US20170008921A1 (en) 2017-01-12
EP3256483B1 (en) 2019-12-11
BR112017017109A2 (pt) 2018-04-03
MX2017010297A (es) 2018-11-12
PE20171433A1 (es) 2017-09-26
PH12017550077A1 (en) 2018-02-12
CO2017008765A2 (es) 2017-11-10
AU2016258274A1 (en) 2017-09-07
US20180215780A1 (en) 2018-08-02
SG11201706189PA (en) 2017-08-30
CU20170102A7 (es) 2018-01-10
KR20170110143A (ko) 2017-10-10
US20200087342A1 (en) 2020-03-19
US11034718B2 (en) 2021-06-15
IL253844A0 (en) 2017-09-28

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