SG11201706189PA - C-3 novel triterpenone with c-17 reverse amide derivatives as hiv inhibitors - Google Patents

C-3 novel triterpenone with c-17 reverse amide derivatives as hiv inhibitors

Info

Publication number
SG11201706189PA
SG11201706189PA SG11201706189PA SG11201706189PA SG11201706189PA SG 11201706189P A SG11201706189P A SG 11201706189PA SG 11201706189P A SG11201706189P A SG 11201706189PA SG 11201706189P A SG11201706189P A SG 11201706189PA SG 11201706189P A SG11201706189P A SG 11201706189PA
Authority
SG
Singapore
Prior art keywords
amide derivatives
hiv inhibitors
reverse amide
triterpenone
novel
Prior art date
Application number
SG11201706189PA
Other languages
English (en)
Inventor
Reddy Bandi Parthasaradhi
Krupadanam Gazula Levi David
Reddy Adulla Panduranga
Reddy Kasireddy Bhaskar
Subrahmanyam Lanka Vl
Reddy Kura Rathnakar
Original Assignee
Hetero Labs Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=57153504&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG11201706189P(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hetero Labs Ltd filed Critical Hetero Labs Ltd
Publication of SG11201706189PA publication Critical patent/SG11201706189PA/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J63/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • C07J63/008—Expansion of ring D by one atom, e.g. D homo steroids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Virology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • AIDS & HIV (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SG11201706189PA 2015-02-09 2016-02-09 C-3 novel triterpenone with c-17 reverse amide derivatives as hiv inhibitors SG11201706189PA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN623CH2015 2015-02-09
PCT/IB2016/000811 WO2016178092A2 (en) 2015-02-09 2016-02-09 C-3 novel triterpenone with c-28 reverse amide derivatives as hiv inhibitors

Publications (1)

Publication Number Publication Date
SG11201706189PA true SG11201706189PA (en) 2017-08-30

Family

ID=57153504

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201706189PA SG11201706189PA (en) 2015-02-09 2016-02-09 C-3 novel triterpenone with c-17 reverse amide derivatives as hiv inhibitors

Country Status (22)

Country Link
US (3) US10533035B2 (es)
EP (1) EP3256483B1 (es)
JP (1) JP2018505216A (es)
KR (1) KR20170110143A (es)
CN (1) CN107428797A (es)
AU (1) AU2016258274B2 (es)
BR (1) BR112017017109A2 (es)
CA (1) CA2975359A1 (es)
CL (1) CL2017002034A1 (es)
CO (1) CO2017008765A2 (es)
CU (1) CU24476B1 (es)
DK (1) DK3256483T3 (es)
EA (1) EA033264B1 (es)
ES (1) ES2780649T3 (es)
IL (1) IL253844A0 (es)
MA (1) MA40886B1 (es)
MX (1) MX2017010297A (es)
PE (1) PE20171433A1 (es)
PH (1) PH12017550077A1 (es)
SG (1) SG11201706189PA (es)
WO (1) WO2016178092A2 (es)
ZA (1) ZA201705253B (es)

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* Cited by examiner, † Cited by third party
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US20170129916A1 (en) 2014-06-26 2017-05-11 Hetero Research Foundation Novel betulinic proline imidazole derivatives as hiv inhibitors
MA40886B1 (fr) 2015-02-09 2020-03-31 Hetero Research Foundation Nouveau triterpénone en c-3 avec des dérivés d'amide inverse en c-28 en tant qu'inhibiteurs du vih
WO2016147099A2 (en) * 2015-03-16 2016-09-22 Hetero Research Foundation C-3 novel triterpenone with c-28 amide derivatives as hiv inhibitors
AR107512A1 (es) 2016-02-04 2018-05-09 VIIV HEALTHCARE UK Nº 5 LTD Triterpenoides modificados en c-3 y c-17 como inhibidores del vih-1
WO2018029604A1 (en) * 2016-08-08 2018-02-15 Hetero Labs Limited C-3 novel triterpenone with c-17 reverse amide derivatives as hiv inhibitors
WO2019150300A1 (en) 2018-02-02 2019-08-08 Glaxosmithkline Intellectual Property (No.2) Limited Crystalline forms of 4-(((3ar,5ar,5br,7ar,9s,11ar,11br,13as)-3a-((r)-2-((4-chlorobenzyl)(2-(dimethylamino)ethyl)amino)-1-hydroxyethyl)-1-isopropyl-5a,5b,8,8,11a-pentamethyl-2-oxo-3,3a,4,5,5a,5b,6,7,7a,8,9,10,11,11a,11b,12,13,13a-octadecahydro-2h-cyclopenta[a]chrysen-9-yl)oxy)-2,2-dimethyl-4-oxobutanoic acid
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Also Published As

Publication number Publication date
MA40886B1 (fr) 2020-03-31
PE20171433A1 (es) 2017-09-26
IL253844A0 (en) 2017-09-28
US11034718B2 (en) 2021-06-15
BR112017017109A2 (pt) 2018-04-03
US20180215780A1 (en) 2018-08-02
CU24476B1 (es) 2020-03-04
EA201791807A1 (ru) 2018-01-31
CO2017008765A2 (es) 2017-11-10
WO2016178092A3 (en) 2017-01-05
CL2017002034A1 (es) 2018-04-27
KR20170110143A (ko) 2017-10-10
AU2016258274B2 (en) 2019-12-05
PH12017550077A1 (en) 2018-02-12
EP3256483B1 (en) 2019-12-11
US20200087342A1 (en) 2020-03-19
US20170008921A1 (en) 2017-01-12
EP3256483A2 (en) 2017-12-20
WO2016178092A2 (en) 2016-11-10
CA2975359A1 (en) 2016-11-10
EA033264B1 (ru) 2019-09-30
JP2018505216A (ja) 2018-02-22
MX2017010297A (es) 2018-11-12
WO2016178092A8 (en) 2017-09-21
CN107428797A (zh) 2017-12-01
ZA201705253B (en) 2020-01-29
AU2016258274A1 (en) 2017-09-07
CU20170102A7 (es) 2018-01-10
DK3256483T3 (da) 2020-03-23
ES2780649T3 (es) 2020-08-26
US10533035B2 (en) 2020-01-14

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