CU20110107A7 - Nuevo procedimiento de preparación de granulados de principios activos, y granulados tal como se los ha obtenido - Google Patents

Nuevo procedimiento de preparación de granulados de principios activos, y granulados tal como se los ha obtenido

Info

Publication number
CU20110107A7
CU20110107A7 CU20110107A CU20110107A CU20110107A7 CU 20110107 A7 CU20110107 A7 CU 20110107A7 CU 20110107 A CU20110107 A CU 20110107A CU 20110107 A CU20110107 A CU 20110107A CU 20110107 A7 CU20110107 A7 CU 20110107A7
Authority
CU
Cuba
Prior art keywords
granulates
active principles
preparation
new procedure
principles
Prior art date
Application number
CU20110107A
Other languages
English (en)
Inventor
Pascal Suplie
Christophe Lebon
Original Assignee
Debregeas Et Associes Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40348849&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CU20110107(A7) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Debregeas Et Associes Pharma filed Critical Debregeas Et Associes Pharma
Publication of CU20110107A7 publication Critical patent/CU20110107A7/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/145Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5036Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005Wall or coating material
    • A61K9/5021Organic macromolecular compounds
    • A61K9/5036Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • A61K9/5042Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
    • A61K9/5047Cellulose ethers containing no ester groups, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Medicinal Preparation (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Fertilizers (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Glanulating (AREA)
  • Seasonings (AREA)
  • Fodder In General (AREA)
  • Medicines Containing Plant Substances (AREA)

Abstract

La presente invención se refiere a un método para la preparación de un granulado de al menos dos principios activos, incluyendo una etapa de aplicación por polvificado de dichos principios activos sobre un soporte particular sólido, y dichos principios activos no son extractos de plantas.
CU20110107A 2008-11-14 2011-05-13 Nuevo procedimiento de preparación de granulados de principios activos, y granulados tal como se los ha obtenido CU20110107A7 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0857764A FR2938432B1 (fr) 2008-11-14 2008-11-14 Nouveau procede de preparation de granules de principes actifs, et granules tels qu'obtenus

Publications (1)

Publication Number Publication Date
CU20110107A7 true CU20110107A7 (es) 2012-01-31

Family

ID=40348849

Family Applications (1)

Application Number Title Priority Date Filing Date
CU20110107A CU20110107A7 (es) 2008-11-14 2011-05-13 Nuevo procedimiento de preparación de granulados de principios activos, y granulados tal como se los ha obtenido

Country Status (25)

Country Link
US (1) US20110280945A1 (es)
EP (1) EP2349226A1 (es)
JP (1) JP5608681B2 (es)
KR (1) KR101585705B1 (es)
CN (1) CN102223879A (es)
AR (1) AR074330A1 (es)
AU (1) AU2009315449B2 (es)
BR (1) BRPI0916019A2 (es)
CA (1) CA2743753A1 (es)
CL (1) CL2011001115A1 (es)
CO (1) CO6382108A2 (es)
CU (1) CU20110107A7 (es)
EA (1) EA201100757A1 (es)
FR (1) FR2938432B1 (es)
IL (1) IL212850A0 (es)
MA (1) MA32789B1 (es)
MX (1) MX2011005072A (es)
NZ (1) NZ592857A (es)
PE (1) PE20110945A1 (es)
SG (1) SG195651A1 (es)
TN (1) TN2011000235A1 (es)
TW (1) TWI522113B (es)
UA (1) UA103781C2 (es)
WO (1) WO2010055268A1 (es)
ZA (1) ZA201103543B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2971422B1 (fr) * 2011-02-11 2016-05-20 Debregeas Et Associes Pharma Granules d'acide gamma-hydroxybutyrique
US20140127296A1 (en) * 2012-11-05 2014-05-08 Kenneth John Tibbs Pharmaceutical preparation and method for treatment of diabetes
US9241956B2 (en) * 2012-11-05 2016-01-26 Kenneth John Tibbs Pharmaceutical preparation and method for treatment of diabetes
US11058635B1 (en) * 2020-10-15 2021-07-13 King Abdulaziz University Oral administration of 5-FU in a gelling nanosuspension for targeted delivery to treat colorectal cancers

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6327424A (ja) * 1986-07-17 1988-02-05 Shionogi & Co Ltd 徐放性製剤およびその製造法
JP2820829B2 (ja) * 1991-03-07 1998-11-05 武田薬品工業株式会社 有核散剤およびその製造方法
JPH08310969A (ja) * 1995-05-22 1996-11-26 Lion Corp 固形薬品組成物及びその製造方法
FR2790668B1 (fr) * 1999-03-12 2002-07-26 D B F Granules contenant une substance vegetale et leur procede de preparation
WO2000069414A2 (fr) * 1999-05-17 2000-11-23 D.B.F. Granules contenant une substance vegetale et leur procede de preparation
MY148805A (en) * 2002-10-16 2013-05-31 Takeda Pharmaceutical Controlled release preparation
US9247765B2 (en) * 2004-01-14 2016-02-02 Omniactive Health Technologies Limited Stable beadlets of lipophilic nutrients
FR2880541B1 (fr) * 2005-01-10 2008-02-22 Amalric Veret Une nouvelle formule de plantes sous forme de micro-granules de xilitol pour renforcer les effets des plantes et leurs proprietes par une meilleure assimilation
US20060182796A1 (en) * 2005-02-03 2006-08-17 Abrika Pharmaceuticals, Inc. Taste masked pharmaceutical compositions
CA2661683C (en) * 2006-08-31 2015-11-24 Eurand, Inc Drug delivery systems comprising solid solutions of weakly basic drugs
CN101611099B (zh) * 2007-02-14 2013-01-02 大日精化工业株式会社 有机颜料的分散剂及其使用
US20090004281A1 (en) * 2007-06-26 2009-01-01 Biovail Laboratories International S.R.L. Multiparticulate osmotic delivery system

Also Published As

Publication number Publication date
WO2010055268A1 (fr) 2010-05-20
JP5608681B2 (ja) 2014-10-15
IL212850A0 (en) 2011-07-31
AU2009315449A1 (en) 2010-05-20
MA32789B1 (fr) 2011-11-01
JP2012508786A (ja) 2012-04-12
US20110280945A1 (en) 2011-11-17
AR074330A1 (es) 2011-01-05
NZ592857A (en) 2013-07-26
TWI522113B (zh) 2016-02-21
BRPI0916019A2 (pt) 2015-11-10
MX2011005072A (es) 2011-10-03
TN2011000235A1 (fr) 2012-12-17
ZA201103543B (en) 2012-01-25
CA2743753A1 (fr) 2010-05-20
FR2938432B1 (fr) 2011-05-20
AU2009315449B2 (en) 2015-03-26
EP2349226A1 (fr) 2011-08-03
CO6382108A2 (es) 2012-02-15
CL2011001115A1 (es) 2011-11-11
TW201029667A (en) 2010-08-16
UA103781C2 (uk) 2013-11-25
KR101585705B1 (ko) 2016-01-15
SG195651A1 (en) 2013-12-30
KR20110095888A (ko) 2011-08-25
FR2938432A1 (fr) 2010-05-21
PE20110945A1 (es) 2012-02-01
EA201100757A1 (ru) 2011-12-30
CN102223879A (zh) 2011-10-19

Similar Documents

Publication Publication Date Title
SMT201600216B (it) Ottaidropirrolo[3,4.c]pirroli disostituiti come modulatori del recettore di orexina
CL2012002419A1 (es) Metodo para mejorar una caracteristica de una planta que comprende administrar bacillus subtilis fb17 a la planta, semilla o al suelo alrededor de la planta o semilla; y metodo para producir biocombustible.
BR112012006415A2 (pt) método para preparar vlps derivadas de plantas
BR112013011574A2 (pt) composição de fertilizante de liberação controlada, e, processo para produzir um fertilizante de liberação controlada
DK2691079T3 (da) Bionedbrydelige sammensætninger, der er egnet til kontrolleret udløsning
BRPI0912252A2 (pt) dispositivos oftálmicos para liberação controlada de agentes ativos.
BR112013004456A2 (pt) composição para tratamento de planta, e, método para o tratamento de plantas
UY34210A (es) Composiciones, métodos y sistemas para la micropropagación de plantas
BR112014006161A2 (pt) embalagem, composição, semente de planta, e, método para intensificar o crescimento de planta
BRPI1007177A2 (pt) processo para a fabricação de composições de fertilizante contendo enxofre, composição de fertilizante, e, uso de um tensoativo aniônico.
BR112012032902A2 (pt) método para controlar vegetação indesejada, composição herbicida e processo para a preparação de composições ativas herbicidas
BRPI0909198A2 (pt) composto antifolato, composto, método para preparar um composto antifolato, composição farmacêutica, método para tratar
MX350447B (es) Composicion farmaceutica de disolucion rapida.
BRPI1011888A2 (pt) processo para preparar um composto, e, composição.
BR112013008008A2 (pt) composto, composição farmacêutica e processo para preparar um composto
BRPI0917104A2 (pt) Métodos para aperfeiçoamento do crescimento de plantas
BR112013032876A2 (pt) uso de formulações, e, método para fertilizar plantas
BR112013007038A2 (pt) "derivados de 2,4-diaril-pirrolina substituída por imina como pesticidas"
DK2582673T3 (da) Fremgangsmåde til fremstilling af 2,2-difluorethylamin-derivater ved hjælp af alkylering med 2,2-difluor-1-halogenethaner
BRPI1014691A2 (pt) Composto, e, processo para a preparação de um composto.
UY33014A (es) Nuevos compuestos de diazinil-pirazolilo
CU20110107A7 (es) Nuevo procedimiento de preparación de granulados de principios activos, y granulados tal como se los ha obtenido
BRPI1012868A2 (pt) processo para a preparacao de um po para pulverizacao, e, uso do po para pulverizacao
BRPI0919774A2 (pt) Complexo cristalino, processo para prepara complexo cristalino, e, composição agrícola
BRPI1010571A2 (pt) processo para a preparação de um composto útil como um inibidor de tafla.