CS91591A2 - Derivatives of 2-deoxy-d-threo-pentofuranoside, method of their preparation, intermediates for their preparation and their application - Google Patents

Derivatives of 2-deoxy-d-threo-pentofuranoside, method of their preparation, intermediates for their preparation and their application Download PDF

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Publication number
CS91591A2
CS91591A2 CS91915A CS91591A CS91591A2 CS 91591 A2 CS91591 A2 CS 91591A2 CS 91915 A CS91915 A CS 91915A CS 91591 A CS91591 A CS 91591A CS 91591 A2 CS91591 A2 CS 91591A2
Authority
CS
Czechoslovakia
Prior art keywords
deoxy
group
formula
methyl
pentofuranoside
Prior art date
Application number
CS91915A
Other languages
Czech (cs)
English (en)
Inventor
Gerald Dipl Ing Saischek
Franz Fuchs
Karl Dr Dax
Gertrude Dr Billiani
Original Assignee
Chemprosa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from AT0079190A external-priority patent/AT394564B/de
Priority claimed from AT0141090A external-priority patent/AT395426B/de
Application filed by Chemprosa filed Critical Chemprosa
Publication of CS91591A2 publication Critical patent/CS91591A2/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H5/00—Compounds containing saccharide radicals in which the hetero bonds to oxygen have been replaced by the same number of hetero bonds to halogen, nitrogen, sulfur, selenium, or tellurium
    • C07H5/02—Compounds containing saccharide radicals in which the hetero bonds to oxygen have been replaced by the same number of hetero bonds to halogen, nitrogen, sulfur, selenium, or tellurium to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H3/00—Compounds containing only hydrogen atoms and saccharide radicals having only carbon, hydrogen, and oxygen atoms
    • C07H3/08—Deoxysugars; Unsaturated sugars; Osones
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H13/00—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids
    • C07H13/02—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by carboxylic acids
    • C07H13/04—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by carboxylic acids having the esterifying carboxyl radicals attached to acyclic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/02—Acyclic radicals, not substituted by cyclic structures
    • C07H15/04—Acyclic radicals, not substituted by cyclic structures attached to an oxygen atom of the saccharide radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/18—Acyclic radicals, substituted by carbocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06—Pyrimidine radicals

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CS91915A 1990-04-04 1991-04-03 Derivatives of 2-deoxy-d-threo-pentofuranoside, method of their preparation, intermediates for their preparation and their application CS91591A2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
AT0079190A AT394564B (de) 1990-04-04 1990-04-04 Verfahren zur herstellung von 2-desoxy-d-threopentose und 2,3-didesoxy-3-fluor-d-erythro-pentosesowie von substituierten und unsubstituierten 2,3-didesoxy-3-fluor-d-erythro-pentofuranosen und deren verwendung
AT0141090A AT395426B (de) 1990-07-03 1990-07-03 Verfahren zur herstellung von 3-azido-2,3didesoxy-d-erythro-pentose sowie von substituierten und unsubstituierten 3-azido-2,3- didesoxy-d-erythro-pentofuranosen und deren verwendung.

Publications (1)

Publication Number Publication Date
CS91591A2 true CS91591A2 (en) 1991-12-17

Family

ID=25593924

Family Applications (1)

Application Number Title Priority Date Filing Date
CS91915A CS91591A2 (en) 1990-04-04 1991-04-03 Derivatives of 2-deoxy-d-threo-pentofuranoside, method of their preparation, intermediates for their preparation and their application

Country Status (8)

Country Link
EP (1) EP0450585A3 (ko)
JP (1) JPH0597885A (ko)
KR (1) KR910018399A (ko)
CA (1) CA2039403A1 (ko)
CS (1) CS91591A2 (ko)
FI (1) FI911603A (ko)
HU (1) HUT57225A (ko)
IL (1) IL97772A0 (ko)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1999043678A1 (fr) * 1998-02-24 1999-09-02 Kyowa Hakko Kogyo Co., Ltd. Medicaments et prophylaxie contre la maladie de parkinson
KR100699099B1 (ko) * 2004-07-29 2007-03-22 한미약품 주식회사 1-α-할로-2,2-다이플루오로-2-데옥시-Ｄ-라이보퓨라노스유도체 및 이의 제조방법
US7858761B2 (en) 2004-07-29 2010-12-28 Hanmi Pharm. Co., Ltd 1-α-halo-2,2-difluoro-2-deoxy-D-ribofuranose derivatives and process for the preparation thereof
CN103242386B (zh) * 2013-04-11 2015-11-04 中国中化股份有限公司 一种制备alpha-1-甲氧基-2-脱氧呋喃核糖衍生物的方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4898936A (en) * 1984-09-24 1990-02-06 Pcr, Inc. 2-deoxyuridines and riboside precursors
DK161788A (da) * 1987-03-25 1988-09-26 Wellcome Found Fremgangsmaade til fremstilling af zidovudin
SE8802173D0 (sv) * 1988-06-10 1988-06-10 Astra Ab Pyrimidine derivatives
US4987224A (en) * 1988-08-02 1991-01-22 University Of Georgia Research Foundation, Inc. Method of preparation of 2',3'-dideoxynucleosides

Also Published As

Publication number Publication date
HUT57225A (en) 1991-11-28
HU911086D0 (en) 1991-10-28
EP0450585A3 (en) 1993-03-10
EP0450585A2 (en) 1991-10-09
FI911603A (fi) 1991-10-05
IL97772A0 (en) 1992-06-21
CA2039403A1 (en) 1991-10-05
JPH0597885A (ja) 1993-04-20
FI911603A0 (fi) 1991-04-03
KR910018399A (ko) 1991-11-30

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