CS228537B2 - Method for the production of methandiole bis-ester with derivates of foaming lanic acid - Google Patents

Method for the production of methandiole bis-ester with derivates of foaming lanic acid Download PDF

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Publication number
CS228537B2
CS228537B2 CS821227A CS122782A CS228537B2 CS 228537 B2 CS228537 B2 CS 228537B2 CS 821227 A CS821227 A CS 821227A CS 122782 A CS122782 A CS 122782A CS 228537 B2 CS228537 B2 CS 228537B2
Authority
CS
Czechoslovakia
Prior art keywords
acid
compounds
bis
compound
formula
Prior art date
Application number
CS821227A
Other languages
Czech (cs)
English (en)
Inventor
Thomas Ch Crawford
Constantine Sklavounos
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/246,504 external-priority patent/US4321196A/en
Application filed by Pfizer filed Critical Pfizer
Priority to CS827097A priority Critical patent/CS228545B2/cs
Publication of CS228537B2 publication Critical patent/CS228537B2/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
    • C07D499/32—Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/80—Compounds with a nitrogen-containing hetero ring, attached with the ring nitrogen atom in position 6

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
CS821227A 1981-03-23 1982-02-23 Method for the production of methandiole bis-ester with derivates of foaming lanic acid CS228537B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CS827097A CS228545B2 (cs) 1981-03-23 1982-10-05 Způsob výroby bis-esterů methandiolu s deriváty penicilanové kyseliny

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US24650381A 1981-03-23 1981-03-23
US06/246,504 US4321196A (en) 1981-03-23 1981-03-23 Bis-esters of methanediol with acetonides of ampicillin or amoxicillin and penicillanic acid 1,1-dioxide

Publications (1)

Publication Number Publication Date
CS228537B2 true CS228537B2 (en) 1984-05-14

Family

ID=26938034

Family Applications (1)

Application Number Title Priority Date Filing Date
CS821227A CS228537B2 (en) 1981-03-23 1982-02-23 Method for the production of methandiole bis-ester with derivates of foaming lanic acid

Country Status (24)

Country Link
EP (1) EP0061281B1 (OSRAM)
KR (1) KR850001630B1 (OSRAM)
AR (1) AR231297A1 (OSRAM)
AU (1) AU527916B2 (OSRAM)
BG (2) BG39297A3 (OSRAM)
CA (1) CA1178575A (OSRAM)
CS (1) CS228537B2 (OSRAM)
DD (1) DD202578A5 (OSRAM)
DE (1) DE3261166D1 (OSRAM)
DK (1) DK159159C (OSRAM)
EG (1) EG15802A (OSRAM)
ES (2) ES8305770A1 (OSRAM)
FI (1) FI74018C (OSRAM)
GB (1) GB2095249A (OSRAM)
GR (1) GR76479B (OSRAM)
IE (1) IE52653B1 (OSRAM)
IL (1) IL65305A (OSRAM)
IN (1) IN157669B (OSRAM)
NO (1) NO159660C (OSRAM)
PL (2) PL130553B1 (OSRAM)
PT (1) PT74623B (OSRAM)
RO (2) RO83699B (OSRAM)
SU (1) SU1122229A3 (OSRAM)
YU (1) YU42760B (OSRAM)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR910009271B1 (ko) * 1989-06-20 1991-11-08 김영설 1,1-디옥소페닐실라노일 옥시메틸 D-6-[α-(메틸렌아미노)페닐-아세트아미도]-페니실라네이트와 그의 파라-톨루엔술폰산염
US7838708B2 (en) 2001-06-20 2010-11-23 Grt, Inc. Hydrocarbon conversion process improvements
CA2532367C (en) 2003-07-15 2013-04-23 Grt, Inc. Hydrocarbon synthesis
US20050171393A1 (en) 2003-07-15 2005-08-04 Lorkovic Ivan M. Hydrocarbon synthesis
US20060100469A1 (en) 2004-04-16 2006-05-11 Waycuilis John J Process for converting gaseous alkanes to olefins and liquid hydrocarbons
US20080275284A1 (en) 2004-04-16 2008-11-06 Marathon Oil Company Process for converting gaseous alkanes to liquid hydrocarbons
US7674941B2 (en) 2004-04-16 2010-03-09 Marathon Gtf Technology, Ltd. Processes for converting gaseous alkanes to liquid hydrocarbons
US8173851B2 (en) 2004-04-16 2012-05-08 Marathon Gtf Technology, Ltd. Processes for converting gaseous alkanes to liquid hydrocarbons
US7244867B2 (en) 2004-04-16 2007-07-17 Marathon Oil Company Process for converting gaseous alkanes to liquid hydrocarbons
US8642822B2 (en) 2004-04-16 2014-02-04 Marathon Gtf Technology, Ltd. Processes for converting gaseous alkanes to liquid hydrocarbons using microchannel reactor
WO2007092410A2 (en) 2006-02-03 2007-08-16 Grt, Inc. Separation of light gases from halogens
EP2457887A1 (en) 2006-02-03 2012-05-30 GRT, Inc. Continuous process for converting natural gas to liquid hydrocarbons
JP2010528054A (ja) 2007-05-24 2010-08-19 ジーアールティー インコーポレイテッド 可逆的なハロゲン化水素の捕捉及び放出を組み込んだ領域反応器
US8282810B2 (en) 2008-06-13 2012-10-09 Marathon Gtf Technology, Ltd. Bromine-based method and system for converting gaseous alkanes to liquid hydrocarbons using electrolysis for bromine recovery
KR101740419B1 (ko) 2008-07-18 2017-05-26 지알티, 인코포레이티드 천연 가스를 액체 탄화수소로 변환시키는 연속 공정
US8198495B2 (en) 2010-03-02 2012-06-12 Marathon Gtf Technology, Ltd. Processes and systems for the staged synthesis of alkyl bromides
US8367884B2 (en) 2010-03-02 2013-02-05 Marathon Gtf Technology, Ltd. Processes and systems for the staged synthesis of alkyl bromides
US8815050B2 (en) 2011-03-22 2014-08-26 Marathon Gtf Technology, Ltd. Processes and systems for drying liquid bromine
US8436220B2 (en) 2011-06-10 2013-05-07 Marathon Gtf Technology, Ltd. Processes and systems for demethanization of brominated hydrocarbons
US8829256B2 (en) 2011-06-30 2014-09-09 Gtc Technology Us, Llc Processes and systems for fractionation of brominated hydrocarbons in the conversion of natural gas to liquid hydrocarbons
US8802908B2 (en) 2011-10-21 2014-08-12 Marathon Gtf Technology, Ltd. Processes and systems for separate, parallel methane and higher alkanes' bromination
US9193641B2 (en) 2011-12-16 2015-11-24 Gtc Technology Us, Llc Processes and systems for conversion of alkyl bromides to higher molecular weight hydrocarbons in circulating catalyst reactor-regenerator systems
CN111440194A (zh) * 2020-04-22 2020-07-24 华南农业大学 一种阿莫西林衍生物及其制备方法和应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE49880B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd Penicillin derivatives
US4244951A (en) * 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide

Also Published As

Publication number Publication date
AR231297A1 (es) 1984-10-31
EP0061281B1 (en) 1984-11-07
SU1122229A3 (ru) 1984-10-30
RO86859B (ro) 1985-05-31
KR830009109A (ko) 1983-12-17
FI74018C (fi) 1987-12-10
ES518997A0 (es) 1984-03-01
PT74623A (en) 1982-04-01
IN157669B (OSRAM) 1986-05-17
EP0061281A1 (en) 1982-09-29
DK159159C (da) 1991-02-11
DK126882A (da) 1982-09-24
IE820655L (en) 1982-09-23
KR850001630B1 (ko) 1985-10-31
NO159660C (no) 1989-01-25
RO83699A (ro) 1984-03-15
BG39113A3 (en) 1986-04-15
GR76479B (OSRAM) 1984-08-10
YU61782A (en) 1985-03-20
PL130553B1 (en) 1984-08-31
AU527916B2 (en) 1983-03-31
YU42760B (en) 1988-12-31
NO159660B (no) 1988-10-17
RO86859A (ro) 1985-05-20
IL65305A0 (en) 1982-05-31
FI74018B (fi) 1987-08-31
AU8176282A (en) 1982-11-04
IE52653B1 (en) 1988-01-06
BG39297A3 (en) 1986-05-15
PL131262B1 (en) 1984-10-31
PT74623B (en) 1984-11-26
ES510657A0 (es) 1983-04-16
IL65305A (en) 1985-02-28
DE3261166D1 (en) 1984-12-13
RO83699B (ro) 1984-03-30
PL235275A1 (en) 1983-04-11
NO820896L (no) 1982-09-24
FI820995L (fi) 1982-09-24
ES8403136A1 (es) 1984-03-01
PL239265A1 (en) 1983-06-06
ES8305770A1 (es) 1983-04-16
DD202578A5 (de) 1983-09-21
GB2095249A (en) 1982-09-29
CA1178575A (en) 1984-11-27
DK159159B (da) 1990-09-10
EG15802A (en) 1987-03-30

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