CS226405B2 - Method of preparing piperidinepropoxyquinoline and piperidinepropoxycoumarin - Google Patents

Method of preparing piperidinepropoxyquinoline and piperidinepropoxycoumarin Download PDF

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Publication number
CS226405B2
CS226405B2 CS80289A CS28980A CS226405B2 CS 226405 B2 CS226405 B2 CS 226405B2 CS 80289 A CS80289 A CS 80289A CS 28980 A CS28980 A CS 28980A CS 226405 B2 CS226405 B2 CS 226405B2
Authority
CS
Czechoslovakia
Prior art keywords
group
propoxy
hydrogen
formula
compound
Prior art date
Application number
CS80289A
Other languages
Czech (cs)
English (en)
Inventor
Walter Gunar Dr Friebe
Werner Dr Winter
Max Dr Thiel
Androniki Dr Roesch
Otto Henning Dr Wilhelms
Original Assignee
Boehringer Mannheim Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Mannheim Gmbh filed Critical Boehringer Mannheim Gmbh
Publication of CS226405B2 publication Critical patent/CS226405B2/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
CS80289A 1979-01-15 1980-01-14 Method of preparing piperidinepropoxyquinoline and piperidinepropoxycoumarin CS226405B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19792901336 DE2901336A1 (de) 1979-01-15 1979-01-15 Neue arylether, verfahren zu deren herstellung sowie diese verbindungen enthaltende arzneimittel

Publications (1)

Publication Number Publication Date
CS226405B2 true CS226405B2 (en) 1984-03-19

Family

ID=6060592

Family Applications (1)

Application Number Title Priority Date Filing Date
CS80289A CS226405B2 (en) 1979-01-15 1980-01-14 Method of preparing piperidinepropoxyquinoline and piperidinepropoxycoumarin

Country Status (13)

Country Link
US (2) US4330549A (fr)
EP (1) EP0013894B1 (fr)
JP (1) JPS5598179A (fr)
AT (1) ATE645T1 (fr)
AU (1) AU529663B2 (fr)
CA (1) CA1141385A (fr)
CS (1) CS226405B2 (fr)
DD (1) DD148634A5 (fr)
DE (2) DE2901336A1 (fr)
ES (1) ES487677A1 (fr)
HU (1) HU182084B (fr)
SU (1) SU997606A3 (fr)
YU (1) YU6880A (fr)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2901336A1 (de) 1979-01-15 1980-07-24 Boehringer Mannheim Gmbh Neue arylether, verfahren zu deren herstellung sowie diese verbindungen enthaltende arzneimittel
DE3034237A1 (de) * 1979-09-18 1981-04-16 Otsuka Pharmaceutical Co. Ltd., Tokyo Carbostyrilderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende, antihistaminisch wirkende mittel
DE3025385A1 (de) * 1980-07-04 1982-01-28 Boehringer Mannheim Gmbh, 6800 Mannheim Neue tricyclische arylether, verfahren zu ihrer herstellung sowie diese verbindungen enthaltende arzneimittel
US4390541A (en) * 1980-12-19 1983-06-28 Lilly Industries Limited Quinolone derivatives and their use in a method of controlling an immediate hypersensitivity disease
DE3117389A1 (de) * 1981-05-02 1982-11-18 Boehringer Mannheim Gmbh, 6800 Mannheim Benzopyranylether, verfahren zu deren herstellung sowie diese verbindungen enthaltende arzneimittel
DE3209271A1 (de) * 1982-03-13 1983-09-15 Boehringer Mannheim Gmbh, 6800 Mannheim Bicyclische phenolether, verfahren zu deren herstellung sowie diese verbindungen enthaltende arzneimittel
JPS6013788A (ja) * 1983-07-05 1985-01-24 Yamanouchi Pharmaceut Co Ltd 新規なクマリン誘導体
US4808619A (en) * 1983-07-27 1989-02-28 Beecham Group P.L.C. Di/tetra-hydroquinolines
DE3431004A1 (de) * 1984-08-23 1986-03-06 Hoechst Ag, 6230 Frankfurt Neue 3-pyridylverbindungen und verfahren zu ihrer herstellung
US4701456A (en) * 1984-09-19 1987-10-20 Warner-Lambert Company Aminoalkoxybenzopyranones as antipsychotic and anxiolytic agents
DE3520718A1 (de) * 1985-06-10 1986-12-11 Herbert 7853 Steinen Hüttlin Fliessbettapparatur
US4704390A (en) * 1986-02-13 1987-11-03 Warner-Lambert Company Phenyl and heterocyclic tetrahydropyridyl alkoxy-benzheterocyclic compounds as antipsychotic agents
GB9018134D0 (en) * 1989-09-29 1990-10-03 Ici Plc Heterocyclic derivatives
US5082847A (en) * 1990-07-18 1992-01-21 Syntex (U.S.A.) Inc. Carbostyril compounds connected via an oxyalkyl group with a piperidine ring and having pharmaceutical utility
IL134193A0 (en) * 1997-07-31 2001-04-30 Hoffmann La Roche O-substituted hydroxycumaranone derivatives as antitumor and antimetastatic agents
CN100393716C (zh) * 2006-05-18 2008-06-11 中国药科大学 香豆素衍生物、其制备方法及作为α1受体拮抗剂的用途
CA2750047A1 (fr) 2009-01-21 2010-07-29 Basilea Pharmaceutica Ag Nouveaux antibiotiques bicycliques
EP3233077A4 (fr) 2014-12-19 2018-08-08 The Broad Institute Inc. Ligands des récepteurs dopaminergiques d2
EP3233799B1 (fr) * 2014-12-19 2021-05-19 The Broad Institute, Inc. Ligands du récepteur d2 de la dopamine
CN113816944B (zh) * 2020-06-20 2023-06-27 中山大学 抗丝状病毒化合物及其应用

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3275658A (en) * 1963-05-23 1966-09-27 Upjohn Co Tertiary-aminoalkoxy-substituted 3, 4-diphenylcoumarins
GB1058822A (en) 1963-07-30 1967-02-15 Ici Ltd 3-amino-2-hydroxypropoxy heterocyclic derivatives
DE1932384U (de) 1965-11-30 1966-02-10 Wilhelm Klein & Soehne Spezial Fraesvorrichtung fuer messerbloecke.
CH529746A (de) * 1968-08-01 1972-10-31 Spofa Vereinigte Pharma Werke Verfahren zur Herstellung von Chromanderivaten
US4029801A (en) 1970-09-03 1977-06-14 John Wyeth & Brother Limited Pharmaceutical compositions and methods of treating hypertension
DE2162721A1 (de) * 1970-12-19 1972-06-22 Dr L Zambeletti SpA, Mailand (Italien) Substituierte Cumarine und Verfahren zu ihrer Herstellung
BE884459Q (fr) 1971-05-14 1981-01-26 Boehringer Mannheim Gmbh Derives de la 4-(omega-(coumarine-7-yl-oxy)-alkyl)-piperazine et procede de preparation
GB1410783A (en) * 1972-01-20 1975-10-22 Wyeth John & Brother Ltd N-substituted 4-amidopyridines tetrahydropyridines and piperidines
US4148909A (en) * 1974-07-30 1979-04-10 Beecham Group Limited Chromans to treat depression and reduce appetite
GB1493998A (en) * 1975-06-03 1977-12-07 Beecham Group Ltd Propanolamine derivatives
CH619453A5 (fr) * 1976-03-17 1980-09-30 Otsuka Pharma Co Ltd
US4210753A (en) * 1976-03-17 1980-07-01 Otsuka Pharmaceutical Co., Ltd. Carbostyril compounds
LU75688A1 (fr) * 1976-08-31 1978-04-13
GB1524260A (en) 1976-11-23 1978-09-06 Beecham Group Ltd Aminoalkyloneoxyd substituted 4-hydroxy-3 nitrocoumarins
FI782133A (fi) * 1977-07-08 1979-01-09 Ciba Geigy Ag Piperidino-propanoler och foerfarande foer deras framstaellning
US4281132A (en) * 1977-10-29 1981-07-28 John Wyeth & Brother Limited Piperidino ureas and thioureas
DE2901336A1 (de) 1979-01-15 1980-07-24 Boehringer Mannheim Gmbh Neue arylether, verfahren zu deren herstellung sowie diese verbindungen enthaltende arzneimittel
DE2905876A1 (de) * 1979-02-16 1980-08-28 Boehringer Mannheim Gmbh Neue piperidinopropylderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE3034237A1 (de) 1979-09-18 1981-04-16 Otsuka Pharmaceutical Co. Ltd., Tokyo Carbostyrilderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende, antihistaminisch wirkende mittel

Also Published As

Publication number Publication date
DE3060160D1 (en) 1982-03-11
AU5435880A (en) 1980-07-24
HU182084B (en) 1983-12-28
EP0013894B1 (fr) 1982-02-03
JPS5598179A (en) 1980-07-25
ATE645T1 (de) 1982-02-15
ES487677A1 (es) 1980-06-16
DD148634A5 (de) 1981-06-03
YU6880A (en) 1983-01-21
AU529663B2 (en) 1983-06-16
CA1141385A (fr) 1983-02-15
DE2901336A1 (de) 1980-07-24
SU997606A3 (ru) 1983-02-15
US4427680A (en) 1984-01-24
EP0013894A1 (fr) 1980-08-06
US4330549A (en) 1982-05-18

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