CS207753B2 - Method of making the 11 beta-hydroxysteroids - Google Patents
Method of making the 11 beta-hydroxysteroids Download PDFInfo
- Publication number
- CS207753B2 CS207753B2 CS79568A CS56879A CS207753B2 CS 207753 B2 CS207753 B2 CS 207753B2 CS 79568 A CS79568 A CS 79568A CS 56879 A CS56879 A CS 56879A CS 207753 B2 CS207753 B2 CS 207753B2
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- dione
- pregnene
- hydroxy
- hours
- methyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
- C07J5/0046—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa
- C07J5/0053—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa not substituted in position 16
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
- C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
- C07J5/0046—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa
- C07J5/0061—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa substituted in position 16
- C07J5/0069—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa substituted in position 16 by a saturated or unsaturated hydrocarbon group
- C07J5/0076—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa substituted in position 16 by a saturated or unsaturated hydrocarbon group by an alkyl group
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
- C07J5/0046—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa
- C07J5/0061—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa substituted in position 16
- C07J5/0069—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa substituted in position 16 by a saturated or unsaturated hydrocarbon group
- C07J5/0084—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa substituted in position 16 by a saturated or unsaturated hydrocarbon group by an alkylene group
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J7/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
- C07J7/0005—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21
- C07J7/001—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group
- C07J7/004—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group substituted in position 17 alfa
- C07J7/0045—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group substituted in position 17 alfa not substituted in position 16
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J7/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
- C07J7/008—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms substituted in position 21
- C07J7/0085—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms substituted in position 21 by an halogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
- C07J71/001—Oxiranes
- C07J71/0015—Oxiranes at position 9(11)
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10S435/00—Chemistry: molecular biology and microbiology
- Y10S435/8215—Microorganisms
- Y10S435/911—Microorganisms using fungi
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Priority Applications (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CS80374A CS207756B2 (cs) | 1978-12-19 | 1980-01-18 | Způsob výroby v poloze 17 substituovaných 11β-bydroxysteroidů pregnanové řady |
| CS80376A CS207758B2 (cs) | 1978-12-19 | 1980-01-18 | Způsob výroby v poloze pregnanové řady 17 substituovaných 11/3-hydroxysteroidů |
| CS80373A CS207755B2 (cs) | 1978-12-19 | 1980-01-18 | Způsob výroby v poloze 17 substituovaných 11ᵝ-hydroxysteroidů pregnanové řady |
| CS80375A CS207757B2 (cs) | 1978-12-19 | 1980-01-18 | Způsob výroby v poloze 17 substituovaných llβ-hydroxysteroidů pregnanové řady |
| CS80372A CS207754B2 (cs) | 1978-12-19 | 1980-01-18 | Způsob výroby v poloze 17 substituovaných lljS-hydroxystcroidů substituovaných lljS-hydroxystcroidů |
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19782803661 DE2803661A1 (de) | 1978-01-25 | 1978-01-25 | Neue in 17-position substituierte 11beta-hydroxysteroide der pregnanreihe, ihre herstellung und verwendung |
| DE19782855465 DE2855465A1 (de) | 1978-12-19 | 1978-12-19 | Neue kortikoide, verfahren zu ihrer herstellung, ihre verwendung und diese kortikoide enthaltende pharmazeutische praeparate |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CS207753B2 true CS207753B2 (en) | 1981-08-31 |
Family
ID=25773724
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CS79568A CS207753B2 (en) | 1978-01-25 | 1979-01-25 | Method of making the 11 beta-hydroxysteroids |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US4207316A (ro) |
| EP (1) | EP0003341B1 (ro) |
| AU (1) | AU529292B2 (ro) |
| BG (3) | BG33737A3 (ro) |
| CS (1) | CS207753B2 (ro) |
| DD (2) | DD150749A5 (ro) |
| DE (1) | DE2967070D1 (ro) |
| DK (1) | DK28779A (ro) |
| EG (1) | EG14273A (ro) |
| ES (1) | ES477162A1 (ro) |
| FI (1) | FI66023C (ro) |
| FR (1) | FR2422689A1 (ro) |
| GB (1) | GB2014150B (ro) |
| IE (1) | IE47729B1 (ro) |
| IL (1) | IL56494A (ro) |
| NO (1) | NO154583C (ro) |
| NZ (1) | NZ189460A (ro) |
| PH (1) | PH18164A (ro) |
| PT (1) | PT69126A (ro) |
| RO (2) | RO76163A (ro) |
| SU (6) | SU876059A3 (ro) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2952003A1 (de) * | 1979-12-21 | 1981-07-02 | Schering Ag Berlin Und Bergkamen, 1000 Berlin | Neue kortikoid-17-thioacetale, ihre herstellung und verwendung |
| DE3038855A1 (de) * | 1980-10-10 | 1982-05-27 | Schering Ag, 1000 Berlin Und 4619 Bergkamen | Neue d-homo-kortikoide, ihre herstellung und verwendung |
| HU221584B (hu) * | 1993-01-08 | 2002-11-28 | Aktiebolaget Astra | Új vastagbél- (colon) vagy csípőbél- (ileum) specifikus, cukortartalmú szteroidszármazékok, ezeket tartalmazó gyógyszerkészítmények és előállításuk |
| US5502222A (en) * | 1994-06-01 | 1996-03-26 | Schering Corporation | Process for preparing delta 9,11 and 21-chloro corticosteroids |
| US8729108B2 (en) * | 2008-06-17 | 2014-05-20 | Christopher J Dannaker | Waterborne topical compositions for the delivery of active ingredients such as azelaic acid |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR6682287D0 (pt) * | 1965-08-30 | 1973-12-04 | Merck & Co Inc | Processo para preparar 17-alcoxi-progesteronas |
| NL6605514A (ro) * | 1966-04-25 | 1967-10-26 | ||
| US3453297A (en) * | 1968-07-24 | 1969-07-01 | Merck & Co Inc | 17alpha-lower alkoxy-pregna-4,6-diene-3,20-dione steroids |
-
1979
- 1979-01-22 EP EP79100176A patent/EP0003341B1/de not_active Expired
- 1979-01-22 BG BG7943567A patent/BG33737A3/xx unknown
- 1979-01-22 BG BG7943566A patent/BG33736A3/xx unknown
- 1979-01-22 BG BG7943568A patent/BG33738A3/xx unknown
- 1979-01-22 DE DE7979100176T patent/DE2967070D1/de not_active Expired
- 1979-01-23 DD DD79220600A patent/DD150749A5/de unknown
- 1979-01-23 DD DD79210595A patent/DD141523A5/de unknown
- 1979-01-23 DK DK28779A patent/DK28779A/da not_active Application Discontinuation
- 1979-01-23 EG EG44/79A patent/EG14273A/xx active
- 1979-01-23 RO RO7996365A patent/RO76163A/ro unknown
- 1979-01-23 RO RO79102257A patent/RO81116A/ro unknown
- 1979-01-24 NO NO790229A patent/NO154583C/no unknown
- 1979-01-24 NZ NZ189460A patent/NZ189460A/xx unknown
- 1979-01-25 SU SU792715602A patent/SU876059A3/ru active
- 1979-01-25 PH PH22112A patent/PH18164A/en unknown
- 1979-01-25 IL IL56494A patent/IL56494A/xx unknown
- 1979-01-25 AU AU43657/79A patent/AU529292B2/en not_active Ceased
- 1979-01-25 PT PT7969126A patent/PT69126A/pt unknown
- 1979-01-25 FR FR7901876A patent/FR2422689A1/fr not_active Withdrawn
- 1979-01-25 FI FI790240A patent/FI66023C/fi not_active IP Right Cessation
- 1979-01-25 CS CS79568A patent/CS207753B2/cs unknown
- 1979-01-25 US US06/006,693 patent/US4207316A/en not_active Expired - Lifetime
- 1979-01-25 ES ES477162A patent/ES477162A1/es not_active Expired
- 1979-01-25 GB GB7902611A patent/GB2014150B/en not_active Expired
- 1979-01-30 IE IE134/79A patent/IE47729B1/en unknown
- 1979-12-11 SU SU792851801A patent/SU1103797A3/ru active
- 1979-12-11 SU SU792853126A patent/SU927123A3/ru active
- 1979-12-11 SU SU792851803A patent/SU880253A3/ru active
- 1979-12-11 SU SU792851807A patent/SU890979A3/ru active
- 1979-12-11 SU SU792853125A patent/SU876060A3/ru active
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