CS200494B2 - Process for preparing therapeutical acylaminosubstituted five-memberd heterocyclic compounds - Google Patents

Process for preparing therapeutical acylaminosubstituted five-memberd heterocyclic compounds Download PDF

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Publication number
CS200494B2
CS200494B2 CS763692A CS369276A CS200494B2 CS 200494 B2 CS200494 B2 CS 200494B2 CS 763692 A CS763692 A CS 763692A CS 369276 A CS369276 A CS 369276A CS 200494 B2 CS200494 B2 CS 200494B2
Authority
CS
Czechoslovakia
Prior art keywords
methyl
group
substituted
compound
formula
Prior art date
Application number
CS763692A
Other languages
Czech (cs)
English (en)
Inventor
William J Ross
John P Verge
William R Williamson
Original Assignee
Lilly Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Industries Ltd filed Critical Lilly Industries Ltd
Publication of CS200494B2 publication Critical patent/CS200494B2/cs

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/061,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/061,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • C07D271/071,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/101,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles
    • C07D271/1131,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01Five-membered rings
    • C07D285/02Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/081,2,4-Thiadiazoles; Hydrogenated 1,2,4-thiadiazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01Five-membered rings
    • C07D285/02Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/121,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
    • C07D285/1251,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • C07D285/135Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
CS763692A 1975-06-05 1976-06-03 Process for preparing therapeutical acylaminosubstituted five-memberd heterocyclic compounds CS200494B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB24224/75A GB1551735A (en) 1975-06-05 1975-06-05 Acylated aminothiazoles and aminooxadiazoles

Publications (1)

Publication Number Publication Date
CS200494B2 true CS200494B2 (en) 1980-09-15

Family

ID=10208350

Family Applications (1)

Application Number Title Priority Date Filing Date
CS763692A CS200494B2 (en) 1975-06-05 1976-06-03 Process for preparing therapeutical acylaminosubstituted five-memberd heterocyclic compounds

Country Status (34)

Country Link
JP (1) JPS51146468A (sv)
AR (1) AR217240A1 (sv)
AT (1) AT346843B (sv)
AU (1) AU503150B2 (sv)
BE (1) BE842579A (sv)
BG (1) BG27359A3 (sv)
CA (1) CA1085860A (sv)
CH (2) CH612427A5 (sv)
CS (1) CS200494B2 (sv)
DD (1) DD125075A5 (sv)
DE (1) DE2625285A1 (sv)
DK (1) DK243276A (sv)
EG (1) EG12226A (sv)
ES (1) ES448590A1 (sv)
FI (1) FI63394C (sv)
FR (1) FR2313049A1 (sv)
GB (1) GB1551735A (sv)
GR (1) GR60380B (sv)
HU (1) HU174191B (sv)
IE (1) IE43474B1 (sv)
IL (1) IL49692A (sv)
LU (1) LU75070A1 (sv)
MX (1) MX3483E (sv)
NL (1) NL7606178A (sv)
NO (1) NO144346C (sv)
NZ (1) NZ181011A (sv)
OA (1) OA05346A (sv)
PH (1) PH16077A (sv)
PL (1) PL103004B1 (sv)
PT (1) PT65182B (sv)
SE (1) SE428561B (sv)
SU (1) SU639451A3 (sv)
YU (1) YU137176A (sv)
ZA (1) ZA763209B (sv)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH636866A5 (de) * 1977-08-15 1983-06-30 Lilly Co Eli Thiadiazolylbenzamide und sie enthaltende insektizide mittel.
DE2805756A1 (de) 1978-02-10 1979-08-16 Bayer Ag N-azolylalkyl-aniline sowie verfahren zu ihrer herstellung
DE2805757A1 (de) * 1978-02-10 1979-08-16 Bayer Ag N-azolylalkyl-halogenacetanilide, verfahren zu ihrer herstellung sowie ihre verwendung als herbizide
US4285959A (en) * 1979-05-18 1981-08-25 Ciba-Geigy Corporation 3-(N-1,3,4-Thiadiazolyl-2)-aminoalkyl-alkyl-acrylates and use thereof as bactericides
US4264616A (en) * 1980-08-29 1981-04-28 Gulf Oil Corporation 2-Iodoacetylimino-3-methyl-5-trifluoromethyl-1,3,4-thiadiazol-4-ine and use as a fungicide
MA19269A1 (fr) * 1980-09-16 1982-04-01 Lilly Co Eli Perfectionnement relatif a des derives de n-arylbenzamides .
DE3120804A1 (de) 1981-05-25 1982-12-16 Basf Ag, 6700 Ludwigshafen N-substituierte 2-methylnaphthylamide, verfahren zu ihrer herstellung und ihre verwendung zur bekaempfung von pilzen
US4874864A (en) * 1988-05-24 1989-10-17 Pfizer Inc. Benzamide protease inhibitors
WO2001046165A2 (en) * 1999-12-16 2001-06-28 Novartis Ag N-heteroaryl-amides and their use as parasiticides
TW200503994A (en) * 2003-01-24 2005-02-01 Novartis Ag Organic compounds
RU2448961C1 (ru) * 2011-02-03 2012-04-27 Открытое акционерное общество "Всероссийский научный центр по безопасности биологически активных веществ" (ОАО "ВНЦ БАВ") Фармацевтическая композиция, обладающая противовоспалительной, бронхолитической, противотуберкулезной активностями

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3720684A (en) * 1970-10-13 1973-03-13 Velsicol Chemical Corp 5-halo-1,2,4-thiadiazoles
IL35743A (en) * 1970-11-27 1974-10-22 Peretz B 3-isopropyl-5-amino-1,2,4-thiadiazole compounds

Also Published As

Publication number Publication date
DE2625285A1 (de) 1976-12-23
AT346843B (de) 1978-11-27
AR217240A1 (es) 1980-03-14
DK243276A (da) 1976-12-06
PT65182A (en) 1976-07-01
ZA763209B (en) 1978-01-25
IL49692A0 (en) 1976-08-31
ES448590A1 (es) 1977-11-16
AU1461976A (en) 1977-12-08
NO144346B (no) 1981-05-04
CH612427A5 (en) 1979-07-31
NL7606178A (nl) 1976-12-07
DD125075A5 (sv) 1977-03-30
ATA412276A (de) 1978-04-15
SE428561B (sv) 1983-07-11
HU174191B (hu) 1979-11-28
NO144346C (no) 1981-08-12
FI761585A (sv) 1976-12-06
SE7606226L (sv) 1976-12-06
IL49692A (en) 1980-07-31
FI63394C (fi) 1983-06-10
GB1551735A (en) 1979-09-12
IE43474L (en) 1976-12-05
OA05346A (fr) 1981-02-28
BG27359A3 (en) 1979-10-12
BE842579A (fr) 1976-12-03
MX3483E (es) 1980-12-16
NZ181011A (en) 1978-11-13
NO761913L (sv) 1976-12-07
PH16077A (en) 1983-06-20
FI63394B (fi) 1983-02-28
FR2313049B1 (sv) 1978-12-15
CH616933A5 (en) 1980-04-30
PL103004B1 (pl) 1979-05-31
AU503150B2 (en) 1979-08-23
YU137176A (en) 1982-10-31
SU639451A3 (ru) 1978-12-25
CA1085860A (en) 1980-09-16
FR2313049A1 (fr) 1976-12-31
EG12226A (en) 1978-12-31
LU75070A1 (sv) 1978-01-18
IE43474B1 (en) 1981-03-11
PT65182B (en) 1978-11-06
JPS51146468A (en) 1976-12-16
GR60380B (en) 1978-05-23

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