CH612427A5 - Process for the preparation of heterocyclic compounds substituted by acylamino groups - Google Patents

Process for the preparation of heterocyclic compounds substituted by acylamino groups

Info

Publication number
CH612427A5
CH612427A5 CH685576A CH685576A CH612427A5 CH 612427 A5 CH612427 A5 CH 612427A5 CH 685576 A CH685576 A CH 685576A CH 685576 A CH685576 A CH 685576A CH 612427 A5 CH612427 A5 CH 612427A5
Authority
CH
Switzerland
Prior art keywords
preparation
heterocyclic compounds
compounds substituted
acylamino groups
groups
Prior art date
Application number
CH685576A
Inventor
William James Ross
John Pomfret Verge
William Robert Nige Williamson
Original Assignee
Lilly Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Industries Ltd filed Critical Lilly Industries Ltd
Publication of CH612427A5 publication Critical patent/CH612427A5/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • C07D271/07—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/10—1,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles
    • C07D271/113—1,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/08—1,2,4-Thiadiazoles; Hydrogenated 1,2,4-thiadiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/12—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
    • C07D285/125—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • C07D285/135—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Compounds of formula <IMAGE> in which Ar is a 1,2,4- or 1,3,4-oxadiazolyl or else a 1,2,4- or 1,3,4-thiadiazolyl group, which groups are substituted or unsubstituted, are prepared by acylation of a corresponding compound ArNHR'. The compounds obtained have an antiallergic activity.
CH685576A 1975-06-05 1976-06-01 Process for the preparation of heterocyclic compounds substituted by acylamino groups CH612427A5 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB24224/75A GB1551735A (en) 1975-06-05 1975-06-05 Acylated aminothiazoles and aminooxadiazoles

Publications (1)

Publication Number Publication Date
CH612427A5 true CH612427A5 (en) 1979-07-31

Family

ID=10208350

Family Applications (2)

Application Number Title Priority Date Filing Date
CH685576A CH612427A5 (en) 1975-06-05 1976-06-01 Process for the preparation of heterocyclic compounds substituted by acylamino groups
CH20579A CH616933A5 (en) 1975-06-05 1979-01-10 Heterocyclic compounds substituted by acylamino groups and process for their preparation

Family Applications After (1)

Application Number Title Priority Date Filing Date
CH20579A CH616933A5 (en) 1975-06-05 1979-01-10 Heterocyclic compounds substituted by acylamino groups and process for their preparation

Country Status (34)

Country Link
JP (1) JPS51146468A (en)
AR (1) AR217240A1 (en)
AT (1) AT346843B (en)
AU (1) AU503150B2 (en)
BE (1) BE842579A (en)
BG (1) BG27359A3 (en)
CA (1) CA1085860A (en)
CH (2) CH612427A5 (en)
CS (1) CS200494B2 (en)
DD (1) DD125075A5 (en)
DE (1) DE2625285A1 (en)
DK (1) DK243276A (en)
EG (1) EG12226A (en)
ES (1) ES448590A1 (en)
FI (1) FI63394C (en)
FR (1) FR2313049A1 (en)
GB (1) GB1551735A (en)
GR (1) GR60380B (en)
HU (1) HU174191B (en)
IE (1) IE43474B1 (en)
IL (1) IL49692A (en)
LU (1) LU75070A1 (en)
MX (1) MX3483E (en)
NL (1) NL7606178A (en)
NO (1) NO144346C (en)
NZ (1) NZ181011A (en)
OA (1) OA05346A (en)
PH (1) PH16077A (en)
PL (1) PL103004B1 (en)
PT (1) PT65182B (en)
SE (1) SE428561B (en)
SU (1) SU639451A3 (en)
YU (1) YU137176A (en)
ZA (1) ZA763209B (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2834945A1 (en) * 1977-08-15 1979-03-01 Lilly Co Eli THIADIAZOLYLBENZAMIDES, METHOD FOR THE PRODUCTION THEREOF AND INSECTICIDES CONTAINING THE SAME
DE2805757A1 (en) * 1978-02-10 1979-08-16 Bayer Ag N-AZOLYLALKYL HALOGEN ACETANILIDES, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS HERBICIDES
DE2805756A1 (en) * 1978-02-10 1979-08-16 Bayer Ag N-AZOLYLALKYL ANILINE AND THE METHOD FOR MANUFACTURING IT
US4285959A (en) * 1979-05-18 1981-08-25 Ciba-Geigy Corporation 3-(N-1,3,4-Thiadiazolyl-2)-aminoalkyl-alkyl-acrylates and use thereof as bactericides
US4264616A (en) * 1980-08-29 1981-04-28 Gulf Oil Corporation 2-Iodoacetylimino-3-methyl-5-trifluoromethyl-1,3,4-thiadiazol-4-ine and use as a fungicide
MA19269A1 (en) * 1980-09-16 1982-04-01 Lilly Co Eli IMPROVEMENT RELATING TO N-ARYLBENZAMIDE DERIVATIVES.
DE3120804A1 (en) 1981-05-25 1982-12-16 Basf Ag, 6700 Ludwigshafen N-SUBSTITUTED 2-METHYLNAPHTHYLAMID, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE FOR CONTROLLING FUNGI
US4874864A (en) * 1988-05-24 1989-10-17 Pfizer Inc. Benzamide protease inhibitors
AU2010601A (en) * 1999-12-16 2001-07-03 Novartis Ag Organic compounds
TW200503994A (en) * 2003-01-24 2005-02-01 Novartis Ag Organic compounds
RU2448961C1 (en) * 2011-02-03 2012-04-27 Открытое акционерное общество "Всероссийский научный центр по безопасности биологически активных веществ" (ОАО "ВНЦ БАВ") Pharmaceutical composition possessing antiinflammatory, broncholytic, anti-tuberculosis activity

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3720684A (en) * 1970-10-13 1973-03-13 Velsicol Chemical Corp 5-halo-1,2,4-thiadiazoles
IL35743A (en) * 1970-11-27 1974-10-22 Peretz B 3-isopropyl-5-amino-1,2,4-thiadiazole compounds

Also Published As

Publication number Publication date
SU639451A3 (en) 1978-12-25
FI761585A (en) 1976-12-06
BE842579A (en) 1976-12-03
AU1461976A (en) 1977-12-08
CS200494B2 (en) 1980-09-15
FI63394B (en) 1983-02-28
ES448590A1 (en) 1977-11-16
EG12226A (en) 1978-12-31
HU174191B (en) 1979-11-28
PL103004B1 (en) 1979-05-31
NL7606178A (en) 1976-12-07
IE43474B1 (en) 1981-03-11
PH16077A (en) 1983-06-20
AT346843B (en) 1978-11-27
BG27359A3 (en) 1979-10-12
CA1085860A (en) 1980-09-16
IL49692A0 (en) 1976-08-31
LU75070A1 (en) 1978-01-18
ZA763209B (en) 1978-01-25
IE43474L (en) 1976-12-05
PT65182A (en) 1976-07-01
GR60380B (en) 1978-05-23
JPS51146468A (en) 1976-12-16
NO144346B (en) 1981-05-04
NO144346C (en) 1981-08-12
FI63394C (en) 1983-06-10
AR217240A1 (en) 1980-03-14
CH616933A5 (en) 1980-04-30
OA05346A (en) 1981-02-28
FR2313049A1 (en) 1976-12-31
YU137176A (en) 1982-10-31
MX3483E (en) 1980-12-16
PT65182B (en) 1978-11-06
AU503150B2 (en) 1979-08-23
FR2313049B1 (en) 1978-12-15
NZ181011A (en) 1978-11-13
SE7606226L (en) 1976-12-06
DE2625285A1 (en) 1976-12-23
SE428561B (en) 1983-07-11
NO761913L (en) 1976-12-07
GB1551735A (en) 1979-09-12
DD125075A5 (en) 1977-03-30
IL49692A (en) 1980-07-31
DK243276A (en) 1976-12-06
ATA412276A (en) 1978-04-15

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Legal Events

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