NL7606178A - PROCESS FOR THE PREPARATION OF PHARMACOLOGICALLY ACTIVE HETEROARYL DERIVATIVES. - Google Patents

PROCESS FOR THE PREPARATION OF PHARMACOLOGICALLY ACTIVE HETEROARYL DERIVATIVES.

Info

Publication number
NL7606178A
NL7606178A NL7606178A NL7606178A NL7606178A NL 7606178 A NL7606178 A NL 7606178A NL 7606178 A NL7606178 A NL 7606178A NL 7606178 A NL7606178 A NL 7606178A NL 7606178 A NL7606178 A NL 7606178A
Authority
NL
Netherlands
Prior art keywords
preparation
pharmacologically active
heteroaryl derivatives
active heteroaryl
derivatives
Prior art date
Application number
NL7606178A
Other languages
Dutch (nl)
Original Assignee
Lilly Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Industries Ltd filed Critical Lilly Industries Ltd
Publication of NL7606178A publication Critical patent/NL7606178A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/061,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/061,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • C07D271/071,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/101,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles
    • C07D271/1131,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01Five-membered rings
    • C07D285/02Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/081,2,4-Thiadiazoles; Hydrogenated 1,2,4-thiadiazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01Five-membered rings
    • C07D285/02Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/121,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
    • C07D285/1251,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • C07D285/135Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
NL7606178A 1975-06-05 1976-06-08 PROCESS FOR THE PREPARATION OF PHARMACOLOGICALLY ACTIVE HETEROARYL DERIVATIVES. NL7606178A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB24224/75A GB1551735A (en) 1975-06-05 1975-06-05 Acylated aminothiazoles and aminooxadiazoles

Publications (1)

Publication Number Publication Date
NL7606178A true NL7606178A (en) 1976-12-07

Family

ID=10208350

Family Applications (1)

Application Number Title Priority Date Filing Date
NL7606178A NL7606178A (en) 1975-06-05 1976-06-08 PROCESS FOR THE PREPARATION OF PHARMACOLOGICALLY ACTIVE HETEROARYL DERIVATIVES.

Country Status (34)

Country Link
JP (1) JPS51146468A (en)
AR (1) AR217240A1 (en)
AT (1) AT346843B (en)
AU (1) AU503150B2 (en)
BE (1) BE842579A (en)
BG (1) BG27359A3 (en)
CA (1) CA1085860A (en)
CH (2) CH612427A5 (en)
CS (1) CS200494B2 (en)
DD (1) DD125075A5 (en)
DE (1) DE2625285A1 (en)
DK (1) DK243276A (en)
EG (1) EG12226A (en)
ES (1) ES448590A1 (en)
FI (1) FI63394C (en)
FR (1) FR2313049A1 (en)
GB (1) GB1551735A (en)
GR (1) GR60380B (en)
HU (1) HU174191B (en)
IE (1) IE43474B1 (en)
IL (1) IL49692A (en)
LU (1) LU75070A1 (en)
MX (1) MX3483E (en)
NL (1) NL7606178A (en)
NO (1) NO144346C (en)
NZ (1) NZ181011A (en)
OA (1) OA05346A (en)
PH (1) PH16077A (en)
PL (1) PL103004B1 (en)
PT (1) PT65182B (en)
SE (1) SE428561B (en)
SU (1) SU639451A3 (en)
YU (1) YU137176A (en)
ZA (1) ZA763209B (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH636866A5 (en) * 1977-08-15 1983-06-30 Lilly Co Eli THIADIAZOLYLBENZAMIDES AND INSECTICIDES CONTAINING THEM.
DE2805757A1 (en) * 1978-02-10 1979-08-16 Bayer Ag N-AZOLYLALKYL HALOGEN ACETANILIDES, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS HERBICIDES
DE2805756A1 (en) * 1978-02-10 1979-08-16 Bayer Ag N-AZOLYLALKYL ANILINE AND THE METHOD FOR MANUFACTURING IT
US4285959A (en) * 1979-05-18 1981-08-25 Ciba-Geigy Corporation 3-(N-1,3,4-Thiadiazolyl-2)-aminoalkyl-alkyl-acrylates and use thereof as bactericides
US4264616A (en) * 1980-08-29 1981-04-28 Gulf Oil Corporation 2-Iodoacetylimino-3-methyl-5-trifluoromethyl-1,3,4-thiadiazol-4-ine and use as a fungicide
MA19269A1 (en) * 1980-09-16 1982-04-01 Lilly Co Eli IMPROVEMENT RELATING TO N-ARYLBENZAMIDE DERIVATIVES.
DE3120804A1 (en) 1981-05-25 1982-12-16 Basf Ag, 6700 Ludwigshafen N-SUBSTITUTED 2-METHYLNAPHTHYLAMID, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE FOR CONTROLLING FUNGI
US4874864A (en) * 1988-05-24 1989-10-17 Pfizer Inc. Benzamide protease inhibitors
WO2001046165A2 (en) * 1999-12-16 2001-06-28 Novartis Ag N-heteroaryl-amides and their use as parasiticides
TW200503994A (en) * 2003-01-24 2005-02-01 Novartis Ag Organic compounds
RU2448961C1 (en) * 2011-02-03 2012-04-27 Открытое акционерное общество "Всероссийский научный центр по безопасности биологически активных веществ" (ОАО "ВНЦ БАВ") Pharmaceutical composition possessing antiinflammatory, broncholytic, anti-tuberculosis activity

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3720684A (en) * 1970-10-13 1973-03-13 Velsicol Chemical Corp 5-halo-1,2,4-thiadiazoles
IL35743A (en) * 1970-11-27 1974-10-22 Peretz B 3-isopropyl-5-amino-1,2,4-thiadiazole compounds

Also Published As

Publication number Publication date
NO144346C (en) 1981-08-12
MX3483E (en) 1980-12-16
EG12226A (en) 1978-12-31
GB1551735A (en) 1979-09-12
IL49692A0 (en) 1976-08-31
IL49692A (en) 1980-07-31
AU503150B2 (en) 1979-08-23
DK243276A (en) 1976-12-06
CH616933A5 (en) 1980-04-30
PL103004B1 (en) 1979-05-31
PH16077A (en) 1983-06-20
SU639451A3 (en) 1978-12-25
AR217240A1 (en) 1980-03-14
IE43474L (en) 1976-12-05
OA05346A (en) 1981-02-28
YU137176A (en) 1982-10-31
GR60380B (en) 1978-05-23
ATA412276A (en) 1978-04-15
IE43474B1 (en) 1981-03-11
JPS51146468A (en) 1976-12-16
CH612427A5 (en) 1979-07-31
NZ181011A (en) 1978-11-13
CS200494B2 (en) 1980-09-15
BG27359A3 (en) 1979-10-12
AU1461976A (en) 1977-12-08
FR2313049A1 (en) 1976-12-31
NO761913L (en) 1976-12-07
LU75070A1 (en) 1978-01-18
BE842579A (en) 1976-12-03
SE7606226L (en) 1976-12-06
FI63394C (en) 1983-06-10
ES448590A1 (en) 1977-11-16
NO144346B (en) 1981-05-04
CA1085860A (en) 1980-09-16
DD125075A5 (en) 1977-03-30
PT65182B (en) 1978-11-06
ZA763209B (en) 1978-01-25
SE428561B (en) 1983-07-11
FR2313049B1 (en) 1978-12-15
DE2625285A1 (en) 1976-12-23
AT346843B (en) 1978-11-27
FI63394B (en) 1983-02-28
PT65182A (en) 1976-07-01
HU174191B (en) 1979-11-28
FI761585A (en) 1976-12-06

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Legal Events

Date Code Title Description
BA A request for search or an international-type search has been filed
BB A search report has been drawn up
BC A request for examination has been filed
A85 Still pending on 85-01-01
BV The patent application has lapsed