CS161892A3 - Heterocyclic derivatives, process of their preparation and pharmaceuticalcompositions in which said derivatives are comprised - Google Patents
Heterocyclic derivatives, process of their preparation and pharmaceuticalcompositions in which said derivatives are comprisedInfo
- Publication number
- CS161892A3 CS161892A3 CS921618A CS161892A CS161892A3 CS 161892 A3 CS161892 A3 CS 161892A3 CS 921618 A CS921618 A CS 921618A CS 161892 A CS161892 A CS 161892A CS 161892 A3 CS161892 A3 CS 161892A3
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- derivatives
- pharmaceuticalcompositions
- comprised
- preparation
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Psychiatry (AREA)
- Endocrinology (AREA)
- Urology & Nephrology (AREA)
- Hospice & Palliative Care (AREA)
- Vascular Medicine (AREA)
- Diabetes (AREA)
- Anesthesiology (AREA)
- Ophthalmology & Optometry (AREA)
- Pain & Pain Management (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB919111759A GB9111759D0 (en) | 1991-05-31 | 1991-05-31 | Heterocyclic compounds |
GB919116309A GB9116309D0 (en) | 1991-07-29 | 1991-07-29 | Bicyclic derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
CS161892A3 true CS161892A3 (en) | 1992-12-16 |
Family
ID=26298984
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CS921618A CS161892A3 (en) | 1991-05-31 | 1992-05-26 | Heterocyclic derivatives, process of their preparation and pharmaceuticalcompositions in which said derivatives are comprised |
Country Status (21)
Country | Link |
---|---|
US (2) | US5217976A (sl) |
EP (1) | EP0516392B1 (sl) |
JP (1) | JPH05163271A (sl) |
KR (1) | KR920021545A (sl) |
CN (1) | CN1073174A (sl) |
AT (1) | ATE204873T1 (sl) |
AU (1) | AU1625192A (sl) |
CA (1) | CA2068946A1 (sl) |
CS (1) | CS161892A3 (sl) |
DE (1) | DE69232022D1 (sl) |
FI (1) | FI922481A (sl) |
GB (1) | GB2256196B (sl) |
HU (1) | HUT61303A (sl) |
IE (1) | IE921506A1 (sl) |
IL (1) | IL101860A0 (sl) |
NO (1) | NO922147L (sl) |
OA (1) | OA09982A (sl) |
PL (1) | PL294736A1 (sl) |
SI (1) | SI9200095A (sl) |
TW (1) | TW213914B (sl) |
YU (1) | YU56192A (sl) |
Families Citing this family (71)
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EP0872235A1 (en) * | 1992-04-13 | 1998-10-21 | Zeneca Limited | Therapeutic agents |
GB9208116D0 (en) | 1992-04-13 | 1992-05-27 | Ici Plc | Therapeutic agents |
GB9211270D0 (en) * | 1992-05-28 | 1992-07-15 | Ici Plc | Nitrogen compounds |
US5466692A (en) * | 1993-03-24 | 1995-11-14 | American Home Products Corporation | Substituted pyridopyrimidines and antihypertensives |
EP0863143A1 (en) * | 1993-03-24 | 1998-09-09 | American Home Products Corporation | Intermediates useful in the production of pyridopyrimidone angiotensin AII antagonists |
US5468867A (en) * | 1994-05-27 | 1995-11-21 | Syntex (U.S.A.) Inc. | Process for preparing1-butyl-2-[2'-(2H-tetrazol-5-yl)biphenyl-4-ylmethyl1-1H-indole-3-carboxylic acid |
US5412102A (en) * | 1994-05-27 | 1995-05-02 | Syntex (U.S.A.) Inc. | Processes for preparing 1-butyl-2-[2'-(2H-tetrazol-5-yl) biphenyl-4-ylmethyl]-1H-indole-3-carboxylic acid |
US5801183A (en) * | 1995-01-27 | 1998-09-01 | State Of Oregon, Acting By And Through The Oregon State Board Of Higher Education, Acting For And On Behalf Of The Oregon Health Sciences University And The University Of Oregon | Aza and aza (N-oxy) analogs of glycine/NMDA receptor antagonists |
TW486479B (en) * | 1997-07-15 | 2002-05-11 | Dainippon Pharmaceutical Co | 5-substituted-3-oxadiazolyl-1,6-naphthyridin-2(1H)-one derivatives |
SE9903028D0 (sv) | 1999-08-27 | 1999-08-27 | Astra Ab | New use |
IL155089A0 (en) | 2000-10-12 | 2003-10-31 | Merck & Co Inc | Aza and polyaza-naphthalenyl carboxamides useful as hiv integrase inhibitors |
ATE364385T1 (de) * | 2000-10-12 | 2007-07-15 | Merck & Co Inc | Aza- und polyaza-naphthalenylcarbonsäureamide als hiv-integrase-hemmer |
EP1326610B1 (en) * | 2000-10-12 | 2006-11-15 | Merck & Co., Inc. | Aza-and polyaza-naphthalenyl carboxamides useful as hiv integrase inhibitors |
AR036256A1 (es) * | 2001-08-17 | 2004-08-25 | Merck & Co Inc | Sal sodica de un inhibidor de integrasa del vih, procesos para su preparacion, composiciones farmaceuticas que lo contienen y su uso para la manufactura de un medicamento |
JP2005504807A (ja) | 2001-09-26 | 2005-02-17 | バイエル・フアーマシユーチカルズ・コーポレーシヨン | 抗糖尿病薬としての1,8−ナフチリジン誘導体 |
ES2291642T3 (es) * | 2002-01-17 | 2008-03-01 | MERCK & CO., INC. | Hidroxinaftiridinoncarboxamidas utiles como inhibidores de la integrasa de vih. |
JP4494020B2 (ja) * | 2002-03-15 | 2010-06-30 | メルク・シャープ・エンド・ドーム・コーポレイション | Hivインテグラーゼ阻害剤として有用なn−(置換ベンジル)−8−ヒドロキシ−1,6−ナフチリジン−7−カルボキサミド |
AU2003248549B2 (en) | 2002-05-24 | 2010-04-08 | Millennium Pharmaceuticals, Inc. | CCR9 inhibitors and methods of use thereof |
AU2003252259A1 (en) * | 2002-07-26 | 2004-02-16 | Nihon Nohyaku Co., Ltd. | Novel haloalkylsulfonanilide derivatives, herbicides and usage thereof |
JP2004107323A (ja) * | 2002-07-26 | 2004-04-08 | Nippon Nohyaku Co Ltd | 新規なハロアルキルスルホンアニリド誘導体及び除草剤並びにその使用方法 |
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US8563579B2 (en) * | 2009-01-15 | 2013-10-22 | Anvyl Llc | α-7 nicotinic acetylcholine receptor allosteric modulators, their derivatives and uses thereof |
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CN113388007A (zh) | 2013-06-05 | 2021-09-14 | 博士医疗爱尔兰有限公司 | 鸟苷酸环化酶c的超纯激动剂、制备和使用所述激动剂的方法 |
CN104418853B (zh) * | 2013-08-28 | 2016-09-07 | 北大方正集团有限公司 | 取代的萘啶-2-酮化合物、制备方法、用途及药物组合物 |
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CN109071426A (zh) | 2016-03-30 | 2018-12-21 | 基因泰克公司 | 取代的苯甲酰胺及其使用方法 |
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TW202000651A (zh) | 2018-02-26 | 2020-01-01 | 美商建南德克公司 | 治療性組成物及其使用方法 |
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TW202334089A (zh) | 2021-11-02 | 2023-09-01 | 美商夫雷爾醫療公司 | Pparg反向激動劑及其用途 |
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-
1992
- 1992-05-14 AU AU16251/92A patent/AU1625192A/en not_active Abandoned
- 1992-05-14 IL IL101860A patent/IL101860A0/xx unknown
- 1992-05-15 HU HU9201608A patent/HUT61303A/hu unknown
- 1992-05-19 CA CA002068946A patent/CA2068946A1/en not_active Abandoned
- 1992-05-26 CS CS921618A patent/CS161892A3/cs unknown
- 1992-05-27 GB GB9211211A patent/GB2256196B/en not_active Revoked
- 1992-05-27 DE DE69232022T patent/DE69232022D1/de not_active Expired - Lifetime
- 1992-05-27 AT AT92304791T patent/ATE204873T1/de active
- 1992-05-27 EP EP92304791A patent/EP0516392B1/en not_active Expired - Lifetime
- 1992-05-29 PL PL29473692A patent/PL294736A1/xx unknown
- 1992-05-29 KR KR1019920009442A patent/KR920021545A/ko not_active Application Discontinuation
- 1992-05-29 OA OA60222A patent/OA09982A/fr unknown
- 1992-05-29 US US07/890,453 patent/US5217976A/en not_active Expired - Fee Related
- 1992-05-29 CN CN92104257A patent/CN1073174A/zh active Pending
- 1992-05-29 YU YU56192A patent/YU56192A/sh unknown
- 1992-05-29 FI FI922481A patent/FI922481A/fi not_active Application Discontinuation
- 1992-05-29 NO NO92922147A patent/NO922147L/no unknown
- 1992-05-29 SI SI19929200095A patent/SI9200095A/sl unknown
- 1992-06-01 JP JP4140731A patent/JPH05163271A/ja active Pending
- 1992-06-12 TW TW081104601A patent/TW213914B/zh active
- 1992-07-01 IE IE150692A patent/IE921506A1/en not_active Application Discontinuation
-
1993
- 1993-04-02 US US08/042,321 patent/US5294620A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
AU1625192A (en) | 1992-12-03 |
PL294736A1 (en) | 1993-05-31 |
ATE204873T1 (de) | 2001-09-15 |
IE921506A1 (en) | 1992-12-02 |
CA2068946A1 (en) | 1992-12-01 |
YU56192A (sh) | 1994-11-15 |
HUT61303A (en) | 1992-12-28 |
NO922147D0 (no) | 1992-05-29 |
NO922147L (no) | 1992-12-01 |
EP0516392A3 (en) | 1993-01-27 |
GB2256196B (en) | 1995-05-10 |
US5294620A (en) | 1994-03-15 |
EP0516392B1 (en) | 2001-08-29 |
HU9201608D0 (en) | 1992-08-28 |
GB2256196A (en) | 1992-12-02 |
TW213914B (sl) | 1993-10-01 |
DE69232022D1 (de) | 2001-10-04 |
EP0516392A2 (en) | 1992-12-02 |
JPH05163271A (ja) | 1993-06-29 |
OA09982A (fr) | 1996-03-29 |
IL101860A0 (en) | 1992-12-30 |
US5217976A (en) | 1993-06-08 |
FI922481A (fi) | 1992-12-01 |
KR920021545A (ko) | 1992-12-18 |
CN1073174A (zh) | 1993-06-16 |
SI9200095A (en) | 1992-12-31 |
FI922481A0 (fi) | 1992-05-29 |
GB9211211D0 (en) | 1992-07-08 |
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