CR11621A - Antagonistas n,n-disustituidos de aminoalquilbifenilo de receptores d2 de prostaglandina - Google Patents

Antagonistas n,n-disustituidos de aminoalquilbifenilo de receptores d2 de prostaglandina

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Publication number
CR11621A
CR11621A CR11621A CR11621A CR11621A CR 11621 A CR11621 A CR 11621A CR 11621 A CR11621 A CR 11621A CR 11621 A CR11621 A CR 11621A CR 11621 A CR11621 A CR 11621A
Authority
CR
Costa Rica
Prior art keywords
antagonists
receptors
bifenyl
prostaglandine
disabled
Prior art date
Application number
CR11621A
Other languages
English (en)
Inventor
Howard Hutchinson John
Andrew Stearns Brian
Melissa Scott Jill
Pham Truong Yen
Roger Roppe Jeffrey
Simon Stock Nicholas
M Aruda Jeannie
Jon Seiders Thomas
Wang Bowei
Volkots Deborah
Original Assignee
Amira Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Amira Pharmaceuticals Inc filed Critical Amira Pharmaceuticals Inc
Publication of CR11621A publication Critical patent/CR11621A/es

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    • C07C233/46—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/47—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of an acyclic saturated carbon skeleton
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Abstract

Se describen aqui compuestos que son antagonistas de receptores PGD2. Tambien se describe composiciones farmaceuticas y medicamentos que incluyen los compuestos aqui descritos que son antagonistas de receptores PGD2. Tambien se describen aqui metodos para utilizar tales antagonistas de receptores PGD2, solos y en combinaciones con otros compuestos, para tratar condiciones o enfermedades respiratorias, cardiovasculares y otras dependientes de PGD2 o mediadas por PGD2.
CR11621A 2008-02-01 2010-08-06 Antagonistas n,n-disustituidos de aminoalquilbifenilo de receptores d2 de prostaglandina CR11621A (es)

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AU2009210446B2 (en) 2012-07-26
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WO2009099902A1 (en) 2009-08-13
EP2257524A1 (en) 2010-12-08
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US8362044B2 (en) 2013-01-29
US20110039852A1 (en) 2011-02-17
US8338484B2 (en) 2012-12-25
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ES2566739T3 (es) 2016-04-15
DOP2010000234A (es) 2010-10-15
US20120058123A1 (en) 2012-03-08
US8168678B2 (en) 2012-05-01
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AU2009210446A1 (en) 2009-08-13
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MX2010008260A (es) 2010-12-20
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US20090197959A1 (en) 2009-08-06
CA2713139C (en) 2013-04-23
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US20130158036A1 (en) 2013-06-20
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HK1149928A1 (en) 2011-10-21
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