CO7000775A2 - Nuevas formas y sales de un dihidropirrolo [1,2-c] imidazolilo, inhibidor de la aldosterona sintasa o aromatasa - Google Patents

Nuevas formas y sales de un dihidropirrolo [1,2-c] imidazolilo, inhibidor de la aldosterona sintasa o aromatasa

Info

Publication number
CO7000775A2
CO7000775A2 CO14146898A CO14146898A CO7000775A2 CO 7000775 A2 CO7000775 A2 CO 7000775A2 CO 14146898 A CO14146898 A CO 14146898A CO 14146898 A CO14146898 A CO 14146898A CO 7000775 A2 CO7000775 A2 CO 7000775A2
Authority
CO
Colombia
Prior art keywords
dihydropyrrolo
imidazolyl
salts
new forms
aromatase inhibitor
Prior art date
Application number
CO14146898A
Other languages
English (en)
Inventor
Paul Sutton
Eric Loeser
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47604250&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO7000775(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of CO7000775A2 publication Critical patent/CO7000775A2/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/38Drugs for disorders of the endocrine system of the suprarenal hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/38Drugs for disorders of the endocrine system of the suprarenal hormones
    • A61P5/46Drugs for disorders of the endocrine system of the suprarenal hormones for decreasing, blocking or antagonising the activity of glucocorticosteroids

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CO14146898A 2012-01-17 2014-07-08 Nuevas formas y sales de un dihidropirrolo [1,2-c] imidazolilo, inhibidor de la aldosterona sintasa o aromatasa CO7000775A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261587280P 2012-01-17 2012-01-17

Publications (1)

Publication Number Publication Date
CO7000775A2 true CO7000775A2 (es) 2014-07-21

Family

ID=47604250

Family Applications (1)

Application Number Title Priority Date Filing Date
CO14146898A CO7000775A2 (es) 2012-01-17 2014-07-08 Nuevas formas y sales de un dihidropirrolo [1,2-c] imidazolilo, inhibidor de la aldosterona sintasa o aromatasa

Country Status (41)

Country Link
US (2) US9334276B2 (es)
EP (1) EP2804863B1 (es)
JP (1) JP5749410B2 (es)
KR (2) KR20140141687A (es)
CN (1) CN104039793B (es)
AP (1) AP2014007762A0 (es)
AR (1) AR089728A1 (es)
AU (1) AU2013209952B2 (es)
BR (1) BR112014017260A8 (es)
CA (1) CA2863339C (es)
CL (1) CL2014001863A1 (es)
CO (1) CO7000775A2 (es)
CR (1) CR20140345A (es)
CU (1) CU20140086A7 (es)
CY (1) CY1117914T1 (es)
DK (1) DK2804863T3 (es)
EA (1) EA026232B1 (es)
ES (1) ES2564143T3 (es)
GT (1) GT201400155A (es)
HK (1) HK1198536A1 (es)
HR (1) HRP20160178T1 (es)
HU (1) HUE026984T2 (es)
IL (1) IL233541B (es)
IN (1) IN2014DN06781A (es)
JO (1) JO3137B1 (es)
MA (1) MA35858B1 (es)
MX (1) MX2014008686A (es)
NZ (1) NZ626277A (es)
PE (1) PE20142358A1 (es)
PH (1) PH12014501638A1 (es)
PL (1) PL2804863T3 (es)
RS (1) RS54589B1 (es)
SG (1) SG11201404061YA (es)
SI (1) SI2804863T1 (es)
SM (1) SMT201600083B (es)
TN (1) TN2014000256A1 (es)
TW (1) TWI609869B (es)
UA (1) UA114803C2 (es)
UY (1) UY34576A (es)
WO (1) WO2013109514A1 (es)
ZA (1) ZA201404314B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2012008212A (es) * 2010-01-14 2012-08-03 Novartis Ag Uso de un agente modificador de hormonas suprarrenales.
EP2815749A1 (en) 2013-06-20 2014-12-24 IP Gesellschaft für Management mbH Solid form of 4-amino-2-(2,6-dioxopiperidine-3-yl)isoindoline-1,3-dione having specified X-ray diffraction pattern
JP6731136B2 (ja) * 2014-07-07 2020-07-29 レコルダティ アーゲー 医薬製剤
CA2973539A1 (en) * 2015-01-29 2016-08-04 Novartis Ag Process for the production of condensed imidazolo derivatives
WO2016164476A2 (en) * 2015-04-06 2016-10-13 Millendo Therapeutics, Inc. Combination therapy for treating disorders associated with excess cortisol production
WO2018078049A1 (en) * 2016-10-27 2018-05-03 Damian Pharma Ag Aldosterone synthase inhibitor
EP3532056A1 (en) * 2016-10-27 2019-09-04 Damian Pharma AG Aldosterone synthase inhibitor
US11992479B2 (en) 2018-05-03 2024-05-28 Damian Pharma Ag R-fadrozole for use in the treatment of aldostonerism

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US1315449A (en) * 1918-11-15 1919-09-09 Frank B Yingling Shaper-feed.
US4617307A (en) * 1984-06-20 1986-10-14 Ciba-Geigy Corporation Substituted imidazo[1,5-A]pyridine derivatives as aromatase inhibitors
US5066656A (en) 1989-11-01 1991-11-19 Janssen Pharmaceutica N.V. Pharmacologically active (6,7-dihydro-5H-pyrrolo[1,2-c]imidazol-5-yl)- and (5,6,7,8-tetrahydroimidazo[1,5-a]pyridin-5-yl) substituted 1H-benzotriazole derivatives
MTP1076B (en) * 1990-01-12 1991-09-30 Ciba Geigy Ag Hemihydrate
ATE203992T1 (de) 1992-01-27 2001-08-15 Janssen Pharmaceutica Nv Pyrroloimidazolyl und imidazopyridinyl substituierte 1h-benzimidazolderivate als aromatase inhibitoren
BR0316306A (pt) * 2002-11-18 2005-09-27 Novartis Ag Compostos orgânicos
GT200600381A (es) * 2005-08-25 2007-03-28 Compuestos organicos
MX2009006481A (es) 2006-12-18 2009-06-26 Novartis Ag Derivados de imidazol 1-sustituidos, y su uso como inhibidores de la sintasa de aldosterona.
US8575160B2 (en) 2009-11-30 2013-11-05 Novartis Ag Imidazole derivatives as aldosterone synthase inhibitors
MX2012008212A (es) * 2010-01-14 2012-08-03 Novartis Ag Uso de un agente modificador de hormonas suprarrenales.

Also Published As

Publication number Publication date
CY1117914T1 (el) 2017-05-17
CA2863339A1 (en) 2013-07-25
BR112014017260A8 (pt) 2017-07-04
EA201491374A1 (ru) 2014-12-30
EP2804863A1 (en) 2014-11-26
CN104039793A (zh) 2014-09-10
KR20140093726A (ko) 2014-07-28
EA026232B1 (ru) 2017-03-31
HUE026984T2 (en) 2016-08-29
PH12014501638B1 (en) 2014-10-13
MA35858B1 (fr) 2014-12-01
HK1198536A1 (en) 2015-05-15
JO3137B1 (ar) 2017-09-20
AR089728A1 (es) 2014-09-10
PH12014501638A1 (en) 2014-10-13
US9334276B2 (en) 2016-05-10
CN104039793B (zh) 2017-05-10
IN2014DN06781A (es) 2015-05-22
DK2804863T3 (en) 2016-03-07
PL2804863T3 (pl) 2016-06-30
UY34576A (es) 2013-09-02
NZ626277A (en) 2015-10-30
SG11201404061YA (en) 2014-08-28
CA2863339C (en) 2021-03-23
SMT201600083B (it) 2016-04-29
ES2564143T8 (es) 2020-11-18
AU2013209952A1 (en) 2014-07-24
CU20140086A7 (es) 2014-12-26
WO2013109514A1 (en) 2013-07-25
CL2014001863A1 (es) 2014-11-07
HRP20160178T1 (hr) 2016-03-25
RS54589B1 (en) 2016-08-31
US20160176883A1 (en) 2016-06-23
JP5749410B2 (ja) 2015-07-15
KR20140141687A (ko) 2014-12-10
EP2804863B1 (en) 2015-12-02
AP2014007762A0 (en) 2014-07-31
TW201335161A (zh) 2013-09-01
ES2564143T3 (es) 2016-03-18
JP2015503627A (ja) 2015-02-02
IL233541B (en) 2018-12-31
BR112014017260A2 (pt) 2017-06-13
UA114803C2 (uk) 2017-08-10
ZA201404314B (en) 2015-08-26
US20140364470A1 (en) 2014-12-11
IL233541A0 (en) 2014-08-31
GT201400155A (es) 2017-09-28
TWI609869B (zh) 2018-01-01
SI2804863T1 (sl) 2016-05-31
TN2014000256A1 (en) 2015-09-30
AU2013209952B2 (en) 2016-09-01
PE20142358A1 (es) 2015-01-30
CR20140345A (es) 2014-09-09
MX2014008686A (es) 2014-08-27

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