ATE203992T1 - Pyrroloimidazolyl und imidazopyridinyl substituierte 1h-benzimidazolderivate als aromatase inhibitoren - Google Patents

Pyrroloimidazolyl und imidazopyridinyl substituierte 1h-benzimidazolderivate als aromatase inhibitoren

Info

Publication number
ATE203992T1
ATE203992T1 AT93903211T AT93903211T ATE203992T1 AT E203992 T1 ATE203992 T1 AT E203992T1 AT 93903211 T AT93903211 T AT 93903211T AT 93903211 T AT93903211 T AT 93903211T AT E203992 T1 ATE203992 T1 AT E203992T1
Authority
AT
Austria
Prior art keywords
phenyl
substituted
amino
6alkyl
pyrroloimidazolyl
Prior art date
Application number
AT93903211T
Other languages
English (en)
Inventor
Marcel August Constant Janssen
Alfons Herman Marg Raeymaekers
Eddy Jean Edgard Freyne
Michael Nicholas Greco
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Application granted granted Critical
Publication of ATE203992T1 publication Critical patent/ATE203992T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02E—REDUCTION OF GREENHOUSE GAS [GHG] EMISSIONS, RELATED TO ENERGY GENERATION, TRANSMISSION OR DISTRIBUTION
    • Y02E50/00—Technologies for the production of fuel of non-fossil origin
    • Y02E50/10—Biofuels, e.g. bio-diesel

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
AT93903211T 1992-01-27 1993-01-20 Pyrroloimidazolyl und imidazopyridinyl substituierte 1h-benzimidazolderivate als aromatase inhibitoren ATE203992T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US82656492A 1992-01-27 1992-01-27
PCT/EP1993/000129 WO1993015079A1 (en) 1992-01-27 1993-01-20 Pyrroloimidazolyl and imidazopyridinyl substituted 1h-benzimidazole derivatives as aromatase inhibitors

Publications (1)

Publication Number Publication Date
ATE203992T1 true ATE203992T1 (de) 2001-08-15

Family

ID=25246906

Family Applications (1)

Application Number Title Priority Date Filing Date
AT93903211T ATE203992T1 (de) 1992-01-27 1993-01-20 Pyrroloimidazolyl und imidazopyridinyl substituierte 1h-benzimidazolderivate als aromatase inhibitoren

Country Status (20)

Country Link
EP (1) EP0625155B1 (de)
JP (1) JPH07503242A (de)
KR (1) KR100263412B1 (de)
CN (2) CN1036007C (de)
AT (1) ATE203992T1 (de)
AU (1) AU668708B2 (de)
CA (1) CA2127689A1 (de)
DE (1) DE69330557T2 (de)
DK (1) DK0625155T3 (de)
ES (1) ES2161714T3 (de)
FI (1) FI106462B (de)
GR (1) GR3036545T3 (de)
HU (1) HU222117B1 (de)
IL (1) IL104498A (de)
MX (1) MX9300412A (de)
NO (1) NO301118B1 (de)
PT (1) PT625155E (de)
TW (1) TW221690B (de)
WO (1) WO1993015079A1 (de)
ZA (1) ZA93561B (de)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU6015796A (en) * 1995-06-14 1997-01-15 Yamanouchi Pharmaceutical Co., Ltd. Fused imidazole derivatives and medicinal composition thereof
MY134929A (en) * 2000-11-17 2008-01-31 Takeda Pharmaceutical Novel imidazole derivatives, production method thereof and use thereof
WO2005000795A2 (en) * 2003-06-10 2005-01-06 Smithkline Beecham Corporation Aniline derivatived androgen-, glucocorticoid-, mineralcorticoid- and progesterone- receptor modulators
CN100496525C (zh) * 2004-04-02 2009-06-10 李嫦梅 从洋蓟根、茎、叶中提取活性成份的方法及其应用
BRPI0511621A (pt) * 2004-05-28 2008-01-02 Speedel Experimenta Ag compostos orgánicos
ATE490241T1 (de) * 2004-05-28 2010-12-15 Novartis Ag Heterocyclische verbindungen und deren verwendung als aldosteronsynthaseinhibitoren
CA2568165A1 (en) 2004-05-28 2005-12-15 Speedel Experimenta Ag Heterocyclic compounds and their use as aldosterone synthase inhibitors
AR049667A1 (es) * 2004-07-09 2006-08-23 Speedel Experimenta Ag Heterociclos condensados conteniendo n como inhibidores de aromatasa y procedimiento para prepararlos
EP1854463A4 (de) * 2005-03-03 2011-03-23 Takeda Pharmaceutical Zusammensetzung mit kontrollierter freisetzung
GT200600381A (es) 2005-08-25 2007-03-28 Compuestos organicos
CN101250559B (zh) * 2008-03-14 2010-12-29 厦门大学 一种利用天然抗菌剂防治酒精发酵染菌的方法
SI2804863T1 (sl) 2012-01-17 2016-05-31 Novartis Ag Nove oblike in soli zaviralca sinteze ali aromataze dihidropropirolo(1,2-c)imidazolil aldosterona
CN106665636A (zh) * 2015-11-07 2017-05-17 郑州明德生物科技有限公司 采用月桂酰精氨酸乙酯抑制酒精发酵污染微生物的方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4426450A (en) * 1981-08-24 1984-01-17 Fermentec Corporation Fermentation process and apparatus
GB8820730D0 (en) * 1988-09-02 1988-10-05 Erba Carlo Spa Substituted 5 6 7 8-tetrahydroimidazo/1.5-a/pyridines & process for their preparation
CA2026792A1 (en) * 1989-11-01 1991-05-02 Michael N. Greco (6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-5-yl)- and (5,6,7,8-tetrahydroimidazo[1,5-a]pyridin-5-yl) substituted 1h-benzotriazole derivatives
US5059431A (en) * 1990-12-07 1991-10-22 State Of Oregon Acting By And Through The State Board Of Higher Education On Behalf Of Oregon State University Process for deacidifying wine

Also Published As

Publication number Publication date
ES2161714T3 (es) 2001-12-16
JPH07503242A (ja) 1995-04-06
AU3450593A (en) 1993-09-01
TW221690B (de) 1994-03-11
WO1993015079A1 (en) 1993-08-05
EP0625155B1 (de) 2001-08-08
EP0625155A1 (de) 1994-11-23
FI943511A0 (fi) 1994-07-26
GR3036545T3 (en) 2001-12-31
KR100263412B1 (ko) 2000-08-01
HUT70853A (en) 1995-11-28
IL104498A0 (en) 1993-05-13
CN1036007C (zh) 1997-10-01
CA2127689A1 (en) 1993-08-05
DE69330557T2 (de) 2002-06-20
MX9300412A (es) 1993-07-01
NO301118B1 (no) 1997-09-15
ZA93561B (en) 1994-07-26
PT625155E (pt) 2002-01-30
DE69330557D1 (de) 2001-09-13
NO942748D0 (no) 1994-07-22
AU668708B2 (en) 1996-05-16
IL104498A (en) 1996-07-23
NO942748L (no) 1994-09-26
DK0625155T3 (da) 2001-11-12
HU9402208D0 (en) 1994-09-28
FI943511A (fi) 1994-07-26
HU222117B1 (hu) 2003-04-28
CN1095415A (zh) 1994-11-23
CN1074907A (zh) 1993-08-04
CN1049687C (zh) 2000-02-23
FI106462B (fi) 2001-02-15

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