FI943511A0 - Pyrroloimidatsolyyli- ja imidatsopyridinyylisubstituoidut 1H-bentsimidatsolijohdannaiset aromataasi-inhibiittoreina - Google Patents

Pyrroloimidatsolyyli- ja imidatsopyridinyylisubstituoidut 1H-bentsimidatsolijohdannaiset aromataasi-inhibiittoreina

Info

Publication number
FI943511A0
FI943511A0 FI943511A FI943511A FI943511A0 FI 943511 A0 FI943511 A0 FI 943511A0 FI 943511 A FI943511 A FI 943511A FI 943511 A FI943511 A FI 943511A FI 943511 A0 FI943511 A0 FI 943511A0
Authority
FI
Finland
Prior art keywords
phenyl
substituted
amino
6alkyl
pyrroloimidazolyl
Prior art date
Application number
FI943511A
Other languages
English (en)
Swedish (sv)
Other versions
FI943511A (fi
FI106462B (fi
Inventor
Marcel August Constant Janssen
Alfons Herman Marg Raeymaekers
Eddy Jean Edgard Freyne
Michael Nicholas Greco
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of FI943511A publication Critical patent/FI943511A/fi
Publication of FI943511A0 publication Critical patent/FI943511A0/fi
Application granted granted Critical
Publication of FI106462B publication Critical patent/FI106462B/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02EREDUCTION OF GREENHOUSE GAS [GHG] EMISSIONS, RELATED TO ENERGY GENERATION, TRANSMISSION OR DISTRIBUTION
    • Y02E50/00Technologies for the production of fuel of non-fossil origin
    • Y02E50/10Biofuels, e.g. bio-diesel

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
FI943511A 1992-01-27 1994-07-26 Menetelmä uusien terapeuttisesti käyttökelpoisten pyrroloimidatsolyyli- ja imidatsopyridinyylisubstituoitujen 1H-bentsimidatsolijohdannaisten valmistamiseksi FI106462B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US82656492A 1992-01-27 1992-01-27
US82656492 1992-01-27
EP9300129 1993-01-20
PCT/EP1993/000129 WO1993015079A1 (en) 1992-01-27 1993-01-20 Pyrroloimidazolyl and imidazopyridinyl substituted 1h-benzimidazole derivatives as aromatase inhibitors

Publications (3)

Publication Number Publication Date
FI943511A FI943511A (fi) 1994-07-26
FI943511A0 true FI943511A0 (fi) 1994-07-26
FI106462B FI106462B (fi) 2001-02-15

Family

ID=25246906

Family Applications (1)

Application Number Title Priority Date Filing Date
FI943511A FI106462B (fi) 1992-01-27 1994-07-26 Menetelmä uusien terapeuttisesti käyttökelpoisten pyrroloimidatsolyyli- ja imidatsopyridinyylisubstituoitujen 1H-bentsimidatsolijohdannaisten valmistamiseksi

Country Status (20)

Country Link
EP (1) EP0625155B1 (fi)
JP (1) JPH07503242A (fi)
KR (1) KR100263412B1 (fi)
CN (2) CN1036007C (fi)
AT (1) ATE203992T1 (fi)
AU (1) AU668708B2 (fi)
CA (1) CA2127689A1 (fi)
DE (1) DE69330557T2 (fi)
DK (1) DK0625155T3 (fi)
ES (1) ES2161714T3 (fi)
FI (1) FI106462B (fi)
GR (1) GR3036545T3 (fi)
HU (1) HU222117B1 (fi)
IL (1) IL104498A (fi)
MX (1) MX9300412A (fi)
NO (1) NO301118B1 (fi)
PT (1) PT625155E (fi)
TW (1) TW221690B (fi)
WO (1) WO1993015079A1 (fi)
ZA (1) ZA93561B (fi)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU6015796A (en) * 1995-06-14 1997-01-15 Yamanouchi Pharmaceutical Co., Ltd. Fused imidazole derivatives and medicinal composition thereof
SI1334106T1 (sl) * 2000-11-17 2006-10-31 Takeda Pharmaceutical Imidazolni derivati, njihov proizvodni postopek in njihova uporaba
JP2007500245A (ja) * 2003-06-10 2007-01-11 スミスクライン ビーチャム コーポレーション 化合物
CN100496525C (zh) * 2004-04-02 2009-06-10 李嫦梅 从洋蓟根、茎、叶中提取活性成份的方法及其应用
CA2568164A1 (en) * 2004-05-28 2005-12-15 Speedel Experimenta Ag Heterocyclic compounds and their use as aldosterone synthase inhibitors
EP2261225A1 (en) 2004-05-28 2010-12-15 Novartis AG Heterocyclic compounds and their use as aldosterone synthase inhibitors
CA2568163A1 (en) * 2004-05-28 2005-12-15 Speedel Experimenta Ag Bicyclic, nitrogen-containing heterocycles as aromatase inhibitors
TW200617010A (en) * 2004-07-09 2006-06-01 Speedel Experimenta Ag Organic compounds
JP5159303B2 (ja) * 2005-03-03 2013-03-06 武田薬品工業株式会社 放出制御組成物
GT200600381A (es) * 2005-08-25 2007-03-28 Compuestos organicos
CN101250559B (zh) * 2008-03-14 2010-12-29 厦门大学 一种利用天然抗菌剂防治酒精发酵染菌的方法
JP5749410B2 (ja) 2012-01-17 2015-07-15 ノバルティス アーゲー ジヒドロピロロ[1,2−c]イミダゾリルアルドステロンシンターゼまたはアロマターゼ阻害薬の新たな形態および塩
CN106665636A (zh) * 2015-11-07 2017-05-17 郑州明德生物科技有限公司 采用月桂酰精氨酸乙酯抑制酒精发酵污染微生物的方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4426450A (en) * 1981-08-24 1984-01-17 Fermentec Corporation Fermentation process and apparatus
GB8820730D0 (en) * 1988-09-02 1988-10-05 Erba Carlo Spa Substituted 5 6 7 8-tetrahydroimidazo/1.5-a/pyridines & process for their preparation
CA2026792A1 (en) * 1989-11-01 1991-05-02 Michael N. Greco (6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-5-yl)- and (5,6,7,8-tetrahydroimidazo[1,5-a]pyridin-5-yl) substituted 1h-benzotriazole derivatives
US5059431A (en) * 1990-12-07 1991-10-22 State Of Oregon Acting By And Through The State Board Of Higher Education On Behalf Of Oregon State University Process for deacidifying wine

Also Published As

Publication number Publication date
NO942748L (no) 1994-09-26
HUT70853A (en) 1995-11-28
FI943511A (fi) 1994-07-26
CN1095415A (zh) 1994-11-23
ZA93561B (en) 1994-07-26
AU3450593A (en) 1993-09-01
CN1036007C (zh) 1997-10-01
JPH07503242A (ja) 1995-04-06
DE69330557T2 (de) 2002-06-20
GR3036545T3 (en) 2001-12-31
AU668708B2 (en) 1996-05-16
PT625155E (pt) 2002-01-30
WO1993015079A1 (en) 1993-08-05
DK0625155T3 (da) 2001-11-12
IL104498A0 (en) 1993-05-13
CN1049687C (zh) 2000-02-23
EP0625155B1 (en) 2001-08-08
NO301118B1 (no) 1997-09-15
NO942748D0 (no) 1994-07-22
DE69330557D1 (de) 2001-09-13
CA2127689A1 (en) 1993-08-05
EP0625155A1 (en) 1994-11-23
HU222117B1 (hu) 2003-04-28
KR100263412B1 (ko) 2000-08-01
TW221690B (fi) 1994-03-11
HU9402208D0 (en) 1994-09-28
CN1074907A (zh) 1993-08-04
ATE203992T1 (de) 2001-08-15
FI106462B (fi) 2001-02-15
IL104498A (en) 1996-07-23
ES2161714T3 (es) 2001-12-16
MX9300412A (es) 1993-07-01

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