CO5410187A1 - Formulacion oral de dosis unica de espinosad - Google Patents

Formulacion oral de dosis unica de espinosad

Info

Publication number
CO5410187A1
CO5410187A1 CO00059545A CO00059545A CO5410187A1 CO 5410187 A1 CO5410187 A1 CO 5410187A1 CO 00059545 A CO00059545 A CO 00059545A CO 00059545 A CO00059545 A CO 00059545A CO 5410187 A1 CO5410187 A1 CO 5410187A1
Authority
CO
Colombia
Prior art keywords
spinosyne
formulation
espinosad
oral formulation
weight
Prior art date
Application number
CO00059545A
Other languages
English (en)
Inventor
Snyder Daniel Earl
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22526570&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO5410187(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of CO5410187A1 publication Critical patent/CO5410187A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/02Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms
    • A01N43/04Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom
    • A01N43/22Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom rings with more than six members
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides

Abstract

Una formulación oral de dosis única que comprende de 0.1 a 75% por peso de una espinosina, o un derivado o sal del mismo fisiológicamente aceptable, y un portador fisiológicamente aceptable, en una forma de dosificación oral adecuada para su administración una vez cada siete días.Una formulación de la reivindicación 1 en donde la espinosina es espinosina A.Una formulación de la reivindicación 1 o 2 en donde la forma de dosificación es en una tableta y la cantidad de la espinosina es entre 1 y 75% en peso de la tableta.Una formulación de la reivindicación 1 o 2 en donde la forma de dosificación es un alimento animal y la cantidad de la espinosina comprende entre 0.1 y 10 % por peso del alimento.
CO00059545A 1999-08-12 2000-08-09 Formulacion oral de dosis unica de espinosad CO5410187A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US14861899P 1999-08-12 1999-08-12

Publications (1)

Publication Number Publication Date
CO5410187A1 true CO5410187A1 (es) 2004-06-30

Family

ID=22526570

Family Applications (1)

Application Number Title Priority Date Filing Date
CO00059545A CO5410187A1 (es) 1999-08-12 2000-08-09 Formulacion oral de dosis unica de espinosad

Country Status (25)

Country Link
US (1) US6664237B1 (es)
EP (1) EP1207756B1 (es)
JP (2) JP5046455B2 (es)
KR (1) KR100706146B1 (es)
AT (1) ATE324039T1 (es)
AU (1) AU775488B2 (es)
BE (1) BE2011C013I2 (es)
BR (1) BR0013116B1 (es)
CA (1) CA2379329C (es)
CO (1) CO5410187A1 (es)
CY (1) CY1105000T1 (es)
DE (2) DE122011100022I1 (es)
DK (1) DK1207756T3 (es)
ES (1) ES2261229T3 (es)
FR (1) FR11C0017I2 (es)
HU (1) HUP0202825A2 (es)
IL (2) IL147828A0 (es)
MX (1) MXPA02001505A (es)
MY (1) MY125485A (es)
NO (1) NO20020686L (es)
NZ (1) NZ516790A (es)
PT (1) PT1207756E (es)
TW (1) TWI244373B (es)
WO (1) WO2001011963A1 (es)
ZA (1) ZA200200565B (es)

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US6933318B1 (en) 1999-08-12 2005-08-23 Eli Lilly And Company Topical organic ectoparasiticidal formulations
AUPQ441699A0 (en) 1999-12-02 2000-01-06 Eli Lilly And Company Pour-on formulations
DE10135550A1 (de) * 2001-07-20 2003-01-30 Bayer Cropscience Ag Verfahren zum Herstellen von neuen Spinosyn-Derivaten
IL160619A0 (en) 2001-09-17 2004-07-25 Lilly Co Eli Pesticidal formulations pesticidal formulations
DE602004017347D1 (de) * 2003-11-04 2008-12-04 Intervet Int Bv Azol-pestiziden
JP4883296B2 (ja) 2004-03-05 2012-02-22 日産化学工業株式会社 イソキサゾリン置換ベンズアミド化合物及び有害生物防除剤
SG159395A1 (en) * 2004-04-29 2010-03-30 Lilly Co Eli Use of spinosyns for wound healing
PT1744763E (pt) * 2004-04-29 2010-03-31 Lilly Co Eli Espinosinas para cura de feridas
BRPI0609930A2 (pt) 2005-05-26 2011-10-11 Lilly Co Eli uso de uma quantidade eficaz de uma espinosina, método para melhorar a produção de peixe criado em aquacultura, e, formulação
KR100855417B1 (ko) * 2006-10-27 2008-08-29 일라이 릴리 앤드 캄파니 스피노신을 포함하는 상처 치유용 제약 조성물
DK2957284T3 (en) * 2007-06-27 2018-02-05 Du Pont PROCEDURE TO CHECK ANIMALS FOR ANIMALS
US9820977B2 (en) 2008-10-03 2017-11-21 Bayer Healthcare Llc Systemic treatment of blood-sucking and blood-consuming parasites by oral administration of a parasiticidal agent
UA108200C2 (uk) * 2009-05-08 2015-04-10 Лікарські форми та способи застосування ектопаразитоцидів
AU2013273709B2 (en) * 2009-05-08 2015-04-23 Eli Lilly And Company Ectoparasiticidal methods and formulations
TWI510189B (zh) * 2009-06-19 2015-12-01 Lilly Co Eli 殺外寄生蟲之方法及調配物
WO2010150100A1 (en) 2009-06-24 2010-12-29 Entarco Sa The use of spinosyns and spinosyn compositions against diseases caused by protozoans, viral infections and cancer
KR20120098930A (ko) 2010-01-25 2012-09-05 일라이 릴리 앤드 캄파니 말과 말파리 유충을 내부적으로 억제 또는 처리하기 위한 방법
CA2817001C (en) * 2010-11-05 2015-09-29 Eli Lilly And Company Methods for inhibiting insect infestations
ITMI20111945A1 (it) * 2011-10-26 2013-04-27 Zapi Ind Chimiche Spa Formulazione in forma idonea a veicolare un quantitativo dosato di una sostanza attiva
CN103125501A (zh) * 2011-11-30 2013-06-05 上海农乐生物制品股份有限公司 一种阿维菌素·多杀霉素水乳剂及其制备方法
TW201416077A (zh) * 2012-07-26 2014-05-01 Lilly Co Eli 單一劑量口服調配物及使用殺外寄生蟲劑賜諾殺(spinosad)以治療貓之方法
CA2885964C (en) 2012-11-14 2017-09-26 Eli Lilly And Company Ectoparasiticidal methods and formulations comprising spinetoram, benzyl alcohol and propylene carbonate
WO2020012406A1 (en) * 2018-07-11 2020-01-16 Jubilant Generics Limited Veterinary dosage forms
CN109221133A (zh) * 2018-09-28 2019-01-18 绩溪农华生物科技有限公司 一种多杀菌素增效水乳剂及其制备方法
CN117500498A (zh) * 2021-03-11 2024-02-02 碗中动物健康公司 用于控制哺乳动物中的蚤和蜱侵袭的方法
WO2022192618A1 (en) * 2021-03-11 2022-09-15 In The Bowl Animal Health, Inc. Feed and methods for controlling tick infestations in a mammal
AU2022296599A1 (en) * 2021-06-25 2023-12-14 In The Bowl Animal Health, Inc. Oral feline feed and methods for controlling flea infestations in a feline
WO2022271937A2 (en) * 2021-06-25 2022-12-29 In The Bowl Animal Health, Inc. Oral feline feed and methods for controlling flea infestations in a feline

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US576253A (en) * 1897-02-02 Manhole-cover
MA21697A1 (fr) * 1988-12-19 1990-07-01 Dow Agrosciences Llc Composes de macrolides.
US5362634A (en) 1989-10-30 1994-11-08 Dowelanco Process for producing A83543 compounds
JPH0375316A (ja) * 1989-08-18 1991-03-29 Tokyo Gas Denro Kk 熱処理炉
US5145684A (en) 1991-01-25 1992-09-08 Sterling Drug Inc. Surface modified drug nanoparticles
US5227295A (en) 1991-11-08 1993-07-13 Dowelanco Process for isolating A83543 and its components
US5202242A (en) 1991-11-08 1993-04-13 Dowelanco A83543 compounds and processes for production thereof
US5539089A (en) 1991-11-08 1996-07-23 Dowelanco A83543 aglycones and pseudoglycones
US5591606A (en) * 1992-11-06 1997-01-07 Dowelanco Process for the production of A83543 compounds with Saccharopolyspora spinosa
CA2156194C (en) 1993-03-12 2008-01-08 Jon S. Mynderse New a83543 compounds and process for production thereof
WO1997000265A1 (en) 1995-06-14 1997-01-03 Dowelanco Synthetic modification to spinosyn compounds
US5695776A (en) 1996-03-12 1997-12-09 Fmc Corporation Termite bait apparatus having grooves
US6001981A (en) * 1996-06-13 1999-12-14 Dow Agrosciences Llc Synthetic modification of Spinosyn compounds
GB9624501D0 (en) * 1996-11-26 1997-01-15 Zeneca Ltd Insecticial compositions and method
JPH11139912A (ja) * 1997-11-06 1999-05-25 Nissan Chem Ind Ltd 安定化される農薬組成物
CN100527958C (zh) * 1997-12-23 2009-08-19 辛根塔参与股份公司 大环内酯在害虫防治中的应用
BRPI9911795B8 (pt) 1998-07-02 2021-05-25 Elanco Us Inc formulação de xampu pediculicida para controle de pediculus humanus humanus, pediculus humanus capitas ou pthius pubis em um ser humano, formulação condicionadora pediculicida capilar, formulação de loção antipiolho e uso de uma espinosina ou sal da mesma”
WO2000060940A1 (en) 1999-04-12 2000-10-19 Dow Agrosciences Llc Aqueous dispersions of agricultural chemicals
AU6605300A (en) 1999-08-12 2001-03-13 Eli Lilly And Company Control of ectoparasites using spinosyns
WO2001012156A1 (en) 1999-08-12 2001-02-22 Eli Lilly And Company Topical organic ectoparasiticidal formulations
DE60015161T2 (de) 1999-09-13 2006-02-02 Dow Agrosciences Llc, Indianapolis Pestizide makrolide
AUPQ441699A0 (en) 1999-12-02 2000-01-06 Eli Lilly And Company Pour-on formulations

Also Published As

Publication number Publication date
HUP0202825A2 (en) 2003-03-28
MY125485A (en) 2006-08-30
IL147828A0 (en) 2002-08-14
FR11C0017I1 (es) 2011-08-07
DE60027575D1 (de) 2006-06-01
ATE324039T1 (de) 2006-05-15
BR0013116B1 (pt) 2013-01-22
BR0013116A (pt) 2002-04-30
KR100706146B1 (ko) 2007-04-11
ZA200200565B (en) 2003-11-26
NO20020686L (no) 2002-04-09
NO20020686D0 (no) 2002-02-11
NZ516790A (en) 2003-03-28
DK1207756T3 (da) 2006-08-14
WO2001011963A1 (en) 2001-02-22
CA2379329C (en) 2009-10-20
EP1207756B1 (en) 2006-04-26
JP5046455B2 (ja) 2012-10-10
EP1207756A1 (en) 2002-05-29
DE60027575T2 (de) 2007-02-15
CA2379329A1 (en) 2001-02-22
KR20020032550A (ko) 2002-05-03
ES2261229T3 (es) 2006-11-16
AU775488B2 (en) 2004-08-05
JP5427217B2 (ja) 2014-02-26
AU6747600A (en) 2001-03-13
BE2011C013I2 (es) 2019-10-16
JP2003506463A (ja) 2003-02-18
IL147828A (en) 2006-08-20
CY1105000T1 (el) 2010-03-03
PT1207756E (pt) 2006-07-31
TWI244373B (en) 2005-12-01
MXPA02001505A (es) 2002-07-02
JP2012001563A (ja) 2012-01-05
FR11C0017I2 (fr) 2012-06-15
DE122011100022I1 (de) 2011-10-20
US6664237B1 (en) 2003-12-16

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