CO5410187A1 - Formulacion oral de dosis unica de espinosad - Google Patents
Formulacion oral de dosis unica de espinosadInfo
- Publication number
- CO5410187A1 CO5410187A1 CO00059545A CO00059545A CO5410187A1 CO 5410187 A1 CO5410187 A1 CO 5410187A1 CO 00059545 A CO00059545 A CO 00059545A CO 00059545 A CO00059545 A CO 00059545A CO 5410187 A1 CO5410187 A1 CO 5410187A1
- Authority
- CO
- Colombia
- Prior art keywords
- spinosyne
- formulation
- espinosad
- oral formulation
- weight
- Prior art date
Links
- 238000009472 formulation Methods 0.000 title abstract 5
- 239000000203 mixture Substances 0.000 title abstract 5
- 239000002552 dosage form Substances 0.000 abstract 2
- 239000006186 oral dosage form Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/02—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms
- A01N43/04—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom
- A01N43/22—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom rings with more than six members
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
Abstract
Una formulación oral de dosis única que comprende de 0.1 a 75% por peso de una espinosina, o un derivado o sal del mismo fisiológicamente aceptable, y un portador fisiológicamente aceptable, en una forma de dosificación oral adecuada para su administración una vez cada siete días.Una formulación de la reivindicación 1 en donde la espinosina es espinosina A.Una formulación de la reivindicación 1 o 2 en donde la forma de dosificación es en una tableta y la cantidad de la espinosina es entre 1 y 75% en peso de la tableta.Una formulación de la reivindicación 1 o 2 en donde la forma de dosificación es un alimento animal y la cantidad de la espinosina comprende entre 0.1 y 10 % por peso del alimento.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US14861899P | 1999-08-12 | 1999-08-12 |
Publications (1)
Publication Number | Publication Date |
---|---|
CO5410187A1 true CO5410187A1 (es) | 2004-06-30 |
Family
ID=22526570
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CO00059545A CO5410187A1 (es) | 1999-08-12 | 2000-08-09 | Formulacion oral de dosis unica de espinosad |
Country Status (25)
Country | Link |
---|---|
US (1) | US6664237B1 (es) |
EP (1) | EP1207756B1 (es) |
JP (2) | JP5046455B2 (es) |
KR (1) | KR100706146B1 (es) |
AT (1) | ATE324039T1 (es) |
AU (1) | AU775488B2 (es) |
BE (1) | BE2011C013I2 (es) |
BR (1) | BR0013116B1 (es) |
CA (1) | CA2379329C (es) |
CO (1) | CO5410187A1 (es) |
CY (1) | CY1105000T1 (es) |
DE (2) | DE122011100022I1 (es) |
DK (1) | DK1207756T3 (es) |
ES (1) | ES2261229T3 (es) |
FR (1) | FR11C0017I2 (es) |
HU (1) | HUP0202825A2 (es) |
IL (2) | IL147828A0 (es) |
MX (1) | MXPA02001505A (es) |
MY (1) | MY125485A (es) |
NO (1) | NO20020686L (es) |
NZ (1) | NZ516790A (es) |
PT (1) | PT1207756E (es) |
TW (1) | TWI244373B (es) |
WO (1) | WO2001011963A1 (es) |
ZA (1) | ZA200200565B (es) |
Families Citing this family (28)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6933318B1 (en) | 1999-08-12 | 2005-08-23 | Eli Lilly And Company | Topical organic ectoparasiticidal formulations |
AUPQ441699A0 (en) | 1999-12-02 | 2000-01-06 | Eli Lilly And Company | Pour-on formulations |
DE10135550A1 (de) * | 2001-07-20 | 2003-01-30 | Bayer Cropscience Ag | Verfahren zum Herstellen von neuen Spinosyn-Derivaten |
IL160619A0 (en) | 2001-09-17 | 2004-07-25 | Lilly Co Eli | Pesticidal formulations pesticidal formulations |
DE602004017347D1 (de) * | 2003-11-04 | 2008-12-04 | Intervet Int Bv | Azol-pestiziden |
JP4883296B2 (ja) | 2004-03-05 | 2012-02-22 | 日産化学工業株式会社 | イソキサゾリン置換ベンズアミド化合物及び有害生物防除剤 |
SG159395A1 (en) * | 2004-04-29 | 2010-03-30 | Lilly Co Eli | Use of spinosyns for wound healing |
PT1744763E (pt) * | 2004-04-29 | 2010-03-31 | Lilly Co Eli | Espinosinas para cura de feridas |
BRPI0609930A2 (pt) | 2005-05-26 | 2011-10-11 | Lilly Co Eli | uso de uma quantidade eficaz de uma espinosina, método para melhorar a produção de peixe criado em aquacultura, e, formulação |
KR100855417B1 (ko) * | 2006-10-27 | 2008-08-29 | 일라이 릴리 앤드 캄파니 | 스피노신을 포함하는 상처 치유용 제약 조성물 |
DK2957284T3 (en) * | 2007-06-27 | 2018-02-05 | Du Pont | PROCEDURE TO CHECK ANIMALS FOR ANIMALS |
US9820977B2 (en) | 2008-10-03 | 2017-11-21 | Bayer Healthcare Llc | Systemic treatment of blood-sucking and blood-consuming parasites by oral administration of a parasiticidal agent |
UA108200C2 (uk) * | 2009-05-08 | 2015-04-10 | Лікарські форми та способи застосування ектопаразитоцидів | |
AU2013273709B2 (en) * | 2009-05-08 | 2015-04-23 | Eli Lilly And Company | Ectoparasiticidal methods and formulations |
TWI510189B (zh) * | 2009-06-19 | 2015-12-01 | Lilly Co Eli | 殺外寄生蟲之方法及調配物 |
WO2010150100A1 (en) | 2009-06-24 | 2010-12-29 | Entarco Sa | The use of spinosyns and spinosyn compositions against diseases caused by protozoans, viral infections and cancer |
KR20120098930A (ko) | 2010-01-25 | 2012-09-05 | 일라이 릴리 앤드 캄파니 | 말과 말파리 유충을 내부적으로 억제 또는 처리하기 위한 방법 |
CA2817001C (en) * | 2010-11-05 | 2015-09-29 | Eli Lilly And Company | Methods for inhibiting insect infestations |
ITMI20111945A1 (it) * | 2011-10-26 | 2013-04-27 | Zapi Ind Chimiche Spa | Formulazione in forma idonea a veicolare un quantitativo dosato di una sostanza attiva |
CN103125501A (zh) * | 2011-11-30 | 2013-06-05 | 上海农乐生物制品股份有限公司 | 一种阿维菌素·多杀霉素水乳剂及其制备方法 |
TW201416077A (zh) * | 2012-07-26 | 2014-05-01 | Lilly Co Eli | 單一劑量口服調配物及使用殺外寄生蟲劑賜諾殺(spinosad)以治療貓之方法 |
CA2885964C (en) | 2012-11-14 | 2017-09-26 | Eli Lilly And Company | Ectoparasiticidal methods and formulations comprising spinetoram, benzyl alcohol and propylene carbonate |
WO2020012406A1 (en) * | 2018-07-11 | 2020-01-16 | Jubilant Generics Limited | Veterinary dosage forms |
CN109221133A (zh) * | 2018-09-28 | 2019-01-18 | 绩溪农华生物科技有限公司 | 一种多杀菌素增效水乳剂及其制备方法 |
CN117500498A (zh) * | 2021-03-11 | 2024-02-02 | 碗中动物健康公司 | 用于控制哺乳动物中的蚤和蜱侵袭的方法 |
WO2022192618A1 (en) * | 2021-03-11 | 2022-09-15 | In The Bowl Animal Health, Inc. | Feed and methods for controlling tick infestations in a mammal |
AU2022296599A1 (en) * | 2021-06-25 | 2023-12-14 | In The Bowl Animal Health, Inc. | Oral feline feed and methods for controlling flea infestations in a feline |
WO2022271937A2 (en) * | 2021-06-25 | 2022-12-29 | In The Bowl Animal Health, Inc. | Oral feline feed and methods for controlling flea infestations in a feline |
Family Cites Families (22)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US576253A (en) * | 1897-02-02 | Manhole-cover | ||
MA21697A1 (fr) * | 1988-12-19 | 1990-07-01 | Dow Agrosciences Llc | Composes de macrolides. |
US5362634A (en) | 1989-10-30 | 1994-11-08 | Dowelanco | Process for producing A83543 compounds |
JPH0375316A (ja) * | 1989-08-18 | 1991-03-29 | Tokyo Gas Denro Kk | 熱処理炉 |
US5145684A (en) | 1991-01-25 | 1992-09-08 | Sterling Drug Inc. | Surface modified drug nanoparticles |
US5227295A (en) | 1991-11-08 | 1993-07-13 | Dowelanco | Process for isolating A83543 and its components |
US5202242A (en) | 1991-11-08 | 1993-04-13 | Dowelanco | A83543 compounds and processes for production thereof |
US5539089A (en) | 1991-11-08 | 1996-07-23 | Dowelanco | A83543 aglycones and pseudoglycones |
US5591606A (en) * | 1992-11-06 | 1997-01-07 | Dowelanco | Process for the production of A83543 compounds with Saccharopolyspora spinosa |
CA2156194C (en) | 1993-03-12 | 2008-01-08 | Jon S. Mynderse | New a83543 compounds and process for production thereof |
WO1997000265A1 (en) | 1995-06-14 | 1997-01-03 | Dowelanco | Synthetic modification to spinosyn compounds |
US5695776A (en) | 1996-03-12 | 1997-12-09 | Fmc Corporation | Termite bait apparatus having grooves |
US6001981A (en) * | 1996-06-13 | 1999-12-14 | Dow Agrosciences Llc | Synthetic modification of Spinosyn compounds |
GB9624501D0 (en) * | 1996-11-26 | 1997-01-15 | Zeneca Ltd | Insecticial compositions and method |
JPH11139912A (ja) * | 1997-11-06 | 1999-05-25 | Nissan Chem Ind Ltd | 安定化される農薬組成物 |
CN100527958C (zh) * | 1997-12-23 | 2009-08-19 | 辛根塔参与股份公司 | 大环内酯在害虫防治中的应用 |
BRPI9911795B8 (pt) | 1998-07-02 | 2021-05-25 | Elanco Us Inc | formulação de xampu pediculicida para controle de pediculus humanus humanus, pediculus humanus capitas ou pthius pubis em um ser humano, formulação condicionadora pediculicida capilar, formulação de loção antipiolho e uso de uma espinosina ou sal da mesma |
WO2000060940A1 (en) | 1999-04-12 | 2000-10-19 | Dow Agrosciences Llc | Aqueous dispersions of agricultural chemicals |
AU6605300A (en) | 1999-08-12 | 2001-03-13 | Eli Lilly And Company | Control of ectoparasites using spinosyns |
WO2001012156A1 (en) | 1999-08-12 | 2001-02-22 | Eli Lilly And Company | Topical organic ectoparasiticidal formulations |
DE60015161T2 (de) | 1999-09-13 | 2006-02-02 | Dow Agrosciences Llc, Indianapolis | Pestizide makrolide |
AUPQ441699A0 (en) | 1999-12-02 | 2000-01-06 | Eli Lilly And Company | Pour-on formulations |
-
2000
- 2000-08-02 ES ES00955247T patent/ES2261229T3/es not_active Expired - Lifetime
- 2000-08-02 JP JP2001516326A patent/JP5046455B2/ja not_active Expired - Lifetime
- 2000-08-02 AU AU67476/00A patent/AU775488B2/en not_active Expired
- 2000-08-02 EP EP00955247A patent/EP1207756B1/en not_active Expired - Lifetime
- 2000-08-02 DE DE201112100022 patent/DE122011100022I1/de active Pending
- 2000-08-02 CA CA002379329A patent/CA2379329C/en not_active Expired - Lifetime
- 2000-08-02 PT PT00955247T patent/PT1207756E/pt unknown
- 2000-08-02 WO PCT/US2000/019557 patent/WO2001011963A1/en active IP Right Grant
- 2000-08-02 BR BRPI0013116-4A patent/BR0013116B1/pt not_active IP Right Cessation
- 2000-08-02 DK DK00955247T patent/DK1207756T3/da active
- 2000-08-02 AT AT00955247T patent/ATE324039T1/de active
- 2000-08-02 MX MXPA02001505A patent/MXPA02001505A/es active IP Right Grant
- 2000-08-02 IL IL14782800A patent/IL147828A0/xx active IP Right Grant
- 2000-08-02 DE DE60027575T patent/DE60027575T2/de not_active Expired - Lifetime
- 2000-08-02 HU HU0202825A patent/HUP0202825A2/hu unknown
- 2000-08-02 KR KR1020027001773A patent/KR100706146B1/ko not_active IP Right Cessation
- 2000-08-02 US US10/049,345 patent/US6664237B1/en not_active Expired - Lifetime
- 2000-08-02 NZ NZ516790A patent/NZ516790A/xx not_active IP Right Cessation
- 2000-08-09 CO CO00059545A patent/CO5410187A1/es not_active Application Discontinuation
- 2000-08-11 MY MYPI20003662A patent/MY125485A/en unknown
- 2000-08-11 TW TW089116161A patent/TWI244373B/zh not_active IP Right Cessation
-
2002
- 2002-01-22 ZA ZA200200565A patent/ZA200200565B/en unknown
- 2002-01-24 IL IL147828A patent/IL147828A/en unknown
- 2002-02-11 NO NO20020686A patent/NO20020686L/no not_active Application Discontinuation
-
2006
- 2006-06-29 CY CY20061100888T patent/CY1105000T1/el unknown
-
2011
- 2011-05-24 FR FR11C0017C patent/FR11C0017I2/fr active Active
- 2011-05-24 BE BE2011C013C patent/BE2011C013I2/fr unknown
- 2011-09-29 JP JP2011214050A patent/JP5427217B2/ja not_active Expired - Lifetime
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD | Application lapsed |