CO5280081A1 - Antibacterianos de piperidiniloxi oxazolidinona, composicion farmaceutica que los comprende y proceso para su preparacion - Google Patents
Antibacterianos de piperidiniloxi oxazolidinona, composicion farmaceutica que los comprende y proceso para su preparacionInfo
- Publication number
- CO5280081A1 CO5280081A1 CO00097143A CO00097143A CO5280081A1 CO 5280081 A1 CO5280081 A1 CO 5280081A1 CO 00097143 A CO00097143 A CO 00097143A CO 00097143 A CO00097143 A CO 00097143A CO 5280081 A1 CO5280081 A1 CO 5280081A1
- Authority
- CO
- Colombia
- Prior art keywords
- alkyl
- theteroaryl
- taryl
- chr5r6
- jpeg
- Prior art date
Links
- OJDXCDWDJDRGFE-UHFFFAOYSA-N 3-piperidin-1-yloxy-1,3-oxazolidin-2-one Chemical compound O=C1OCCN1ON1CCCCC1 OJDXCDWDJDRGFE-UHFFFAOYSA-N 0.000 title 1
- 229940088710 antibiotic agent Drugs 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 7
- 125000002877 alkyl aryl group Chemical group 0.000 abstract 3
- 125000002252 acyl group Chemical group 0.000 abstract 2
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- -1 cyclic amino derivative Chemical class 0.000 abstract 1
- 125000003106 haloaryl group Chemical group 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 230000003287 optical effect Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Physical Education & Sports Medicine (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Rheumatology (AREA)
- Communicable Diseases (AREA)
- Immunology (AREA)
- Oncology (AREA)
- Dermatology (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US17292399P | 1999-12-21 | 1999-12-21 | |
| US09/729,342 US6518285B2 (en) | 1999-12-21 | 2000-12-05 | Piperidinyloxy and pyrrolidinyloxy oxazolidinone antibacterials |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CO5280081A1 true CO5280081A1 (es) | 2003-05-30 |
Family
ID=22629768
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CO00097143A CO5280081A1 (es) | 1999-12-21 | 2000-12-21 | Antibacterianos de piperidiniloxi oxazolidinona, composicion farmaceutica que los comprende y proceso para su preparacion |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US6518285B2 (https=) |
| EP (1) | EP1246810B1 (https=) |
| JP (1) | JP2003518106A (https=) |
| CN (1) | CN1227238C (https=) |
| AR (1) | AR029420A1 (https=) |
| AT (1) | ATE326452T1 (https=) |
| AU (1) | AU784314B2 (https=) |
| CA (1) | CA2395204C (https=) |
| CO (1) | CO5280081A1 (https=) |
| CY (1) | CY1106124T1 (https=) |
| DE (1) | DE60028085T2 (https=) |
| DK (1) | DK1246810T3 (https=) |
| ES (1) | ES2265365T3 (https=) |
| MX (1) | MXPA02006323A (https=) |
| MY (1) | MY127677A (https=) |
| PT (1) | PT1246810E (https=) |
| WO (1) | WO2001046164A1 (https=) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9928568D0 (en) | 1999-12-03 | 2000-02-02 | Zeneca Ltd | Chemical compounds |
| GB0009803D0 (en) | 2000-04-25 | 2000-06-07 | Astrazeneca Ab | Chemical compounds |
| WO2003031443A1 (en) | 2001-10-04 | 2003-04-17 | Morphochem Aktiengesellschaft für kombinatorische Chemie | Dual actions antibiotics comprising a oxazoldinone and a quinolone or naphthyridinone moiety |
| US6940748B2 (en) | 2002-05-16 | 2005-09-06 | Micron Technology, Inc. | Stacked 1T-nMTJ MRAM structure |
| EP1594852A1 (en) * | 2003-02-07 | 2005-11-16 | Ranbaxy Laboratories, Ltd. | Oxazolidinone derivatives as antimicrobials |
| JP4805139B2 (ja) | 2003-04-30 | 2011-11-02 | モルホケム アクツィエンゲゼルシャフト フューア コンビナートリッシュ ヒェミー | 炭疽および他の感染を治療するためのオキサゾリジノン‐キノリンハイブリッド抗生物質の使用 |
| DE10340485B4 (de) | 2003-09-03 | 2015-05-13 | Morphochem AG Aktiengesellschaft für kombinatorische Chemie | Verfahren zur Herstellung von Oxazolidinon-Chinolon Hybriden |
| US8158797B2 (en) | 2003-12-18 | 2012-04-17 | Morphochem Aktiengesellschaft Fur Kombinatorische Chemie | Oxazolidinone-quinolone hybrid antibiotics |
| BRPI0417193B8 (pt) | 2003-12-18 | 2021-05-25 | Morphochem Ag Fuer Komb Chemie | antibióticos híbridos de oxazolidinona-quinolona, seus sais monossódicos, dissódicos ou trissódicos e seus pró-fármacos, composições farmacêuticas, e seu uso |
| MX2007003318A (es) | 2004-09-20 | 2007-05-18 | Xenon Pharmaceuticals Inc | Derivados heterociclicos y su uso como agentes terapeuticos. |
| BRPI0515482A (pt) | 2004-09-20 | 2008-07-22 | Xenon Pharmaceuticals Inc | derivados heterocìclicos e seus usos como agentes terapêuticos |
| MX2007003332A (es) | 2004-09-20 | 2007-06-05 | Xenon Pharmaceuticals Inc | Derivados heterociclicos y su uso como inhibidores de estearoil-coa-desaturasa. |
| BRPI0515500A (pt) * | 2004-09-20 | 2008-07-29 | Xenon Pharmaceuticals Inc | derivados piridazina para inibição de estearoil-coa-desaturase |
| AU2005286728A1 (en) | 2004-09-20 | 2006-03-30 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as mediators of stearoyl-CoA desaturase |
| CA2618646A1 (en) | 2005-06-03 | 2007-11-15 | Xenon Pharmaceuticals Inc. | Aminothiazole derivatives as human stearoyl-coa desaturase inhibitors |
| EP2407459A1 (en) | 2005-09-27 | 2012-01-18 | Shionogi & Co., Ltd. | Synthetic intermediate in the production of a sulfonamide derivative having PGD2 receptor antagonistic activity |
| JP5209254B2 (ja) * | 2007-08-30 | 2013-06-12 | 日本曹達株式会社 | 置換フェノキシアザビシクロオクタン誘導体の製造方法 |
| CN108785728A (zh) * | 2017-05-05 | 2018-11-13 | 国家纳米科学中心 | 含药物中间体修饰的纳米金的抗菌敷料、其制备方法及应用 |
| CN109503569B (zh) * | 2019-01-03 | 2021-01-15 | 山东大学 | 噻唑类衍生物及其制备方法和应用 |
| JP2024538778A (ja) * | 2021-10-12 | 2024-10-23 | エフ． ホフマン－ラ ロシュ アーゲー | 細菌感染症の処置のためのスルホニルピペラジニル化合物 |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES533097A0 (es) | 1983-06-07 | 1985-08-01 | Du Pont | Un procedimiento para la preparacion de nuevos derivados del amino-metil-oxooxazolidinil-benzeno. |
| US4705799A (en) | 1983-06-07 | 1987-11-10 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl benzenes useful as antibacterial agents |
| JPS608277A (ja) * | 1983-06-07 | 1985-01-17 | ザ・デュポン・メルク・ファーマシュウティカル・カンパニー | アミノメチルオキソオキサゾリジニルベンゼン誘導体 |
| CA1260948A (en) * | 1984-12-05 | 1989-09-26 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl benzene derivatives useful as antibacterial agents |
| EP0610265B1 (en) | 1991-11-01 | 1996-12-27 | PHARMACIA & UPJOHN COMPANY | Substituted aryl- and heteroarylphenyloxazolidinones useful as antibacterial agents |
| MY115155A (en) * | 1993-09-09 | 2003-04-30 | Upjohn Co | Substituted oxazine and thiazine oxazolidinone antimicrobials. |
| PT792273E (pt) | 1994-11-15 | 2003-06-30 | Upjohn Co | Produtos antibacterianos de oxazolidinona substituida com oxazina e tiazina biciclicas |
| ATE205205T1 (de) | 1995-02-03 | 2001-09-15 | Upjohn Co | Durch hetero-aromatische ring substituierte phenyloxazolidinone als antimikrobielles mittel |
| US6124334A (en) | 1995-02-03 | 2000-09-26 | Pharmacia & Upjohn Company | Hetero-aromatic ring substituted phenyloxazolidinone antimicrobials |
| HRP960159A2 (en) * | 1995-04-21 | 1997-08-31 | Bayer Ag | Benzocyclopentane oxazolidinones containing heteroatoms |
| DE69614847T2 (de) | 1995-05-11 | 2002-04-04 | Pharmacia & Upjohn Co., Kalamazoo | Spirocyclische und bicyclische diazinyl- und carbazinyloxazolidinone |
| US5883093A (en) | 1995-09-12 | 1999-03-16 | Pharmacia & Upjohn Company | Phenyloxazolidinone antimicrobials |
| DE19601264A1 (de) | 1996-01-16 | 1997-07-17 | Bayer Ag | Pyrido-annellierte Thienyl- und Furanyl-Oxazolidinone |
| DE19604223A1 (de) | 1996-02-06 | 1997-08-07 | Bayer Ag | Neue substituierte Oxazolidinone |
| DK1114819T3 (da) | 1996-04-11 | 2008-04-14 | Pharmacia & Upjohn Co Llc | Fremgangsmåde til fremstilling af oxazolidinoner |
| SK156499A3 (en) | 1997-05-30 | 2000-06-12 | Upjohn Co | Oxazolidinone antibacterial agents having a thiocarbonyl functionality |
| GB9717807D0 (en) | 1997-08-22 | 1997-10-29 | Zeneca Ltd | Chemical compounds |
| AU9001598A (en) | 1997-09-11 | 1999-03-29 | Hokuriku Seiyaku Co. Ltd | Thiourea derivatives |
| JPH11322729A (ja) | 1998-03-09 | 1999-11-24 | Hokuriku Seiyaku Co Ltd | ジチオカルバミド酸誘導体 |
| JP2000204084A (ja) * | 1998-11-11 | 2000-07-25 | Hokuriku Seiyaku Co Ltd | チオカルバミド酸誘導体 |
-
2000
- 2000-12-05 US US09/729,342 patent/US6518285B2/en not_active Expired - Lifetime
- 2000-12-14 MX MXPA02006323A patent/MXPA02006323A/es active IP Right Grant
- 2000-12-14 DE DE60028085T patent/DE60028085T2/de not_active Expired - Fee Related
- 2000-12-14 EP EP00986365A patent/EP1246810B1/en not_active Expired - Lifetime
- 2000-12-14 PT PT00986365T patent/PT1246810E/pt unknown
- 2000-12-14 WO PCT/US2000/033835 patent/WO2001046164A1/en not_active Ceased
- 2000-12-14 CA CA002395204A patent/CA2395204C/en not_active Expired - Fee Related
- 2000-12-14 DK DK00986365T patent/DK1246810T3/da active
- 2000-12-14 AT AT00986365T patent/ATE326452T1/de not_active IP Right Cessation
- 2000-12-14 CN CNB008189803A patent/CN1227238C/zh not_active Expired - Fee Related
- 2000-12-14 ES ES00986365T patent/ES2265365T3/es not_active Expired - Lifetime
- 2000-12-14 JP JP2001547075A patent/JP2003518106A/ja active Pending
- 2000-12-14 AU AU22617/01A patent/AU784314B2/en not_active Ceased
- 2000-12-20 MY MYPI20006020A patent/MY127677A/en unknown
- 2000-12-20 AR ARP000106796A patent/AR029420A1/es unknown
- 2000-12-21 CO CO00097143A patent/CO5280081A1/es not_active Application Discontinuation
-
2006
- 2006-07-21 CY CY20061101016T patent/CY1106124T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US20020103377A1 (en) | 2002-08-01 |
| MXPA02006323A (es) | 2003-09-22 |
| CA2395204A1 (en) | 2001-06-28 |
| EP1246810A1 (en) | 2002-10-09 |
| DE60028085D1 (de) | 2006-06-22 |
| PT1246810E (pt) | 2006-08-31 |
| AU784314B2 (en) | 2006-03-09 |
| CN1434810A (zh) | 2003-08-06 |
| DE60028085T2 (de) | 2006-12-07 |
| CN1227238C (zh) | 2005-11-16 |
| AR029420A1 (es) | 2003-06-25 |
| CA2395204C (en) | 2008-02-05 |
| ATE326452T1 (de) | 2006-06-15 |
| DK1246810T3 (da) | 2006-09-18 |
| CY1106124T1 (el) | 2011-06-08 |
| EP1246810B1 (en) | 2006-05-17 |
| ES2265365T3 (es) | 2007-02-16 |
| WO2001046164A1 (en) | 2001-06-28 |
| AU2261701A (en) | 2001-07-03 |
| US6518285B2 (en) | 2003-02-11 |
| MY127677A (en) | 2006-12-29 |
| JP2003518106A (ja) | 2003-06-03 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Application granted | ||
| FD | Application lapsed |