CO2020001506A2 - Nuevos compuestos - Google Patents

Nuevos compuestos

Info

Publication number
CO2020001506A2
CO2020001506A2 CONC2020/0001506A CO2020001506A CO2020001506A2 CO 2020001506 A2 CO2020001506 A2 CO 2020001506A2 CO 2020001506 A CO2020001506 A CO 2020001506A CO 2020001506 A2 CO2020001506 A2 CO 2020001506A2
Authority
CO
Colombia
Prior art keywords
new compounds
treatment
compounds
mycobacteria
tuberculosis
Prior art date
Application number
CONC2020/0001506A
Other languages
English (en)
Inventor
De Francisco Esther Porras
Modesto Jesús Remuiñan-Blanco
Marilyne Bourotte
Benoit Deprez
Nicolas Willand
Original Assignee
Glaxosmithkline Ip Dev Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=59713957&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO2020001506(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Glaxosmithkline Ip Dev Ltd filed Critical Glaxosmithkline Ip Dev Ltd
Publication of CO2020001506A2 publication Critical patent/CO2020001506A2/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/10—Spiro-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/438—The ring being spiro-condensed with carbocyclic or heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/06—Antibacterial agents for tuberculosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

La invención se refiere a compuestos de fórmula (I) y su uso en terapia, por ejemplo en el tratamiento de infecciones micobacterianas o en el tratamiento de enfermedades causadas por micobacteria, tales como la tuberculosis. (I).
CONC2020/0001506A 2017-08-16 2020-02-11 Nuevos compuestos CO2020001506A2 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP17382569 2017-08-16
PCT/EP2018/072143 WO2019034700A1 (en) 2017-08-16 2018-08-15 NEW COMPOUNDS

Publications (1)

Publication Number Publication Date
CO2020001506A2 true CO2020001506A2 (es) 2020-05-29

Family

ID=59713957

Family Applications (1)

Application Number Title Priority Date Filing Date
CONC2020/0001506A CO2020001506A2 (es) 2017-08-16 2020-02-11 Nuevos compuestos

Country Status (25)

Country Link
US (1) US11254689B2 (es)
EP (1) EP3668879B1 (es)
JP (1) JP7171726B2 (es)
KR (1) KR102657360B1 (es)
CN (1) CN110997680B (es)
AU (1) AU2018317804B2 (es)
BR (1) BR112020003192A2 (es)
CA (1) CA3072838A1 (es)
CL (1) CL2020000362A1 (es)
CO (1) CO2020001506A2 (es)
CY (1) CY1124851T1 (es)
DK (1) DK3668879T3 (es)
ES (1) ES2899365T3 (es)
HR (1) HRP20211895T1 (es)
HU (1) HUE056928T2 (es)
IL (1) IL272562B2 (es)
LT (1) LT3668879T (es)
MX (1) MX2020001808A (es)
PL (1) PL3668879T3 (es)
PT (1) PT3668879T (es)
RS (1) RS62708B1 (es)
SG (1) SG11202000988RA (es)
SI (1) SI3668879T1 (es)
WO (1) WO2019034700A1 (es)
ZA (1) ZA202000585B (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111184718A (zh) * 2018-11-15 2020-05-22 鲁南制药集团股份有限公司 法罗培南在制备治疗初治病原学阳性肺结核药物中的用途

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR041198A1 (es) 2002-10-11 2005-05-04 Otsuka Pharma Co Ltd Compuesto 2,3-dihidro-6-nitroimidazo[2,1-b] oxaxol, y composiciones farmaceuticas que lo contienen
DE102005044813A1 (de) * 2005-05-19 2007-10-04 Grünenthal GmbH Substituierte Spiro-Verbindungen und deren Verwendung zur Herstellung von Arzneimitteln
FR3000065A1 (fr) * 2012-12-21 2014-06-27 Univ Lille Ii Droit & Sante Composes bicycliques ayant une activite potentialisatrice de l'activite d'un antibiotique actif contre les mycobacteries-composition et produit pharmaceutiques comprenant de tels composes
FR3000064A1 (fr) * 2012-12-21 2014-06-27 Univ Lille Ii Droit & Sante Composes de type spiroisoxazoline ayant une activite potentialisatrice de l'activite d'un antibiotique-composition et produit pharmaceutiques comprenant de tels composes

Also Published As

Publication number Publication date
SI3668879T1 (sl) 2022-04-29
CN110997680B (zh) 2022-10-21
IL272562B2 (en) 2023-08-01
RS62708B1 (sr) 2022-01-31
BR112020003192A2 (pt) 2020-09-15
AU2018317804A1 (en) 2020-02-20
RU2020109677A (ru) 2021-09-16
US11254689B2 (en) 2022-02-22
IL272562A (en) 2020-03-31
JP2020531575A (ja) 2020-11-05
MX2020001808A (es) 2022-07-19
PT3668879T (pt) 2021-12-02
DK3668879T3 (da) 2021-12-06
ES2899365T3 (es) 2022-03-11
LT3668879T (lt) 2022-03-25
ZA202000585B (en) 2021-07-28
AU2018317804B2 (en) 2021-04-22
JP7171726B2 (ja) 2022-11-15
CY1124851T1 (el) 2022-11-25
PL3668879T3 (pl) 2022-02-21
CL2020000362A1 (es) 2020-07-10
EP3668879A1 (en) 2020-06-24
HUE056928T2 (hu) 2022-03-28
RU2020109677A3 (es) 2021-09-28
SG11202000988RA (en) 2020-03-30
EP3668879B1 (en) 2021-09-29
HRP20211895T1 (hr) 2022-08-19
CN110997680A (zh) 2020-04-10
KR102657360B1 (ko) 2024-04-16
WO2019034700A1 (en) 2019-02-21
CA3072838A1 (en) 2019-02-21
US20210032268A1 (en) 2021-02-04
IL272562B1 (en) 2023-04-01
KR20200041344A (ko) 2020-04-21

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