CO2017001603A2 - Compuestos aminopirimidinilo inhibidores de jak - Google Patents

Compuestos aminopirimidinilo inhibidores de jak

Info

Publication number
CO2017001603A2
CO2017001603A2 CONC2017/0001603A CO2017001603A CO2017001603A2 CO 2017001603 A2 CO2017001603 A2 CO 2017001603A2 CO 2017001603 A CO2017001603 A CO 2017001603A CO 2017001603 A2 CO2017001603 A2 CO 2017001603A2
Authority
CO
Colombia
Prior art keywords
alkyl
aryl
heteroaryl
cycloalkyl
group
Prior art date
Application number
CONC2017/0001603A
Other languages
English (en)
Spanish (es)
Inventor
Ivan Viktorovich Efremov
Jean-Baptiste Telliez
John I Trujillo
Eddine Saiah
Andrew Fensome
Ariamala Gopalsamy
Brian S Gerstenberger
Zhao-Kui Wan
Betsy PIERCE
Liying Zhang
Li Xing
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=54148580&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO2017001603(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of CO2017001603A2 publication Critical patent/CO2017001603A2/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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CONC2017/0001603A 2014-08-21 2017-02-17 Compuestos aminopirimidinilo inhibidores de jak CO2017001603A2 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201462039969P 2014-08-21 2014-08-21
PCT/IB2015/056021 WO2016027195A1 (en) 2014-08-21 2015-08-07 Aminopyrimidinyl compounds as jak inhibitors

Publications (1)

Publication Number Publication Date
CO2017001603A2 true CO2017001603A2 (es) 2017-05-10

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CONC2017/0001603A CO2017001603A2 (es) 2014-08-21 2017-02-17 Compuestos aminopirimidinilo inhibidores de jak

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US (5) US9663526B2 (cg-RX-API-DMAC7.html)
EP (1) EP3183247B9 (cg-RX-API-DMAC7.html)
JP (1) JP6218260B2 (cg-RX-API-DMAC7.html)
KR (1) KR101877189B1 (cg-RX-API-DMAC7.html)
CN (1) CN107074867B (cg-RX-API-DMAC7.html)
AP (1) AP2017009748A0 (cg-RX-API-DMAC7.html)
AR (1) AR101599A1 (cg-RX-API-DMAC7.html)
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US10463675B2 (en) 2019-11-05
IL250709B (en) 2019-05-30
NO2721710T3 (cg-RX-API-DMAC7.html) 2018-03-31
JP2017524022A (ja) 2017-08-24
CL2017000406A1 (es) 2017-10-06

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