CN1921858A - 哌啶基烷基氨基甲酸酯衍生物、其制备方法及其作为faah酶抑制剂的应用 - Google Patents

哌啶基烷基氨基甲酸酯衍生物、其制备方法及其作为faah酶抑制剂的应用 Download PDF

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CN1921858A
CN1921858A CNA2005800058637A CN200580005863A CN1921858A CN 1921858 A CN1921858 A CN 1921858A CN A2005800058637 A CNA2005800058637 A CN A2005800058637A CN 200580005863 A CN200580005863 A CN 200580005863A CN 1921858 A CN1921858 A CN 1921858A
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group
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phenyl
groups
compound
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A·阿布亚布德拉
A·阿尔马里奥加西亚
C·霍奈尔特
J·热纳斯
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Sanofi Aventis France
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CN102369200B (zh) * 2009-02-05 2015-05-20 赛诺菲 5元杂环化合物的氮杂螺烷基-烷基氨基甲酸酯衍生物、其制备方法和其治疗用途

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FR2866886B1 (fr) * 2004-02-26 2007-08-31 Sanofi Synthelabo Derives d'aryl-et d'heteroaryl-akylcarbamates, leur preparation et leur application en therapeutique
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WO2007061862A2 (en) * 2005-11-18 2007-05-31 Janssen Pharmaceutica N.V. 2-keto-oxazoles as modulators of fatty acid amide hydrolase
EP1966132A2 (en) 2005-12-15 2008-09-10 Boehringer Ingelheim International Gmbh Compounds which modulate the cb2 receptor
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WO2010005782A1 (en) 2008-07-10 2010-01-14 Boehringer Ingelheim International Gmbh Sulfone compounds which modulate the cb2 receptor
PE20110397A1 (es) 2008-09-25 2011-07-01 Boehringer Ingelheim Int Compuestos que modulan selectivamente el receptor cb2
US8299103B2 (en) 2009-06-15 2012-10-30 Boehringer Ingelheim International Gmbh Compounds which selectively modulate the CB2 receptor
WO2010147791A1 (en) 2009-06-16 2010-12-23 Boehringer Ingelheim International Gmbh Azetidine 2 -carboxamide derivatives which modulate the cb2 receptor
JP2013505295A (ja) 2009-09-22 2013-02-14 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｃｂ２受容体を選択的に調節する化合物
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EP2542539B1 (en) 2010-03-05 2014-02-26 Boehringer Ingelheim International GmbH Tetrazole compounds which selectively modulate the cb2 receptor
WO2012012307A1 (en) 2010-07-22 2012-01-26 Boehringer Ingelheim International Gmbh Sulfonyl compounds which modulate the cb2 rece
EP2803668A1 (en) 2013-05-17 2014-11-19 Boehringer Ingelheim International Gmbh Novel (cyano-dimethyl-methyl)-isoxazoles and -[1,3,4]thiadiazoles

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RU2216540C2 (ru) * 1997-11-18 2003-11-20 Тейджин Лимитед Производные циклических аминов, способ ингибирования
JP2001523695A (ja) * 1997-11-24 2001-11-27 ザ スクリップス リサーチ インスティテュート ギャップ結合連絡の阻害剤
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FR2850377B1 (fr) * 2003-01-23 2009-02-20 Sanofi Synthelabo Derives d'arylalkylcarbamates, leur preparation et leur application en therapeutique
FR2854633B1 (fr) * 2003-05-07 2005-06-24 Sanofi Synthelabo Derives de piperidinyl-et piperazinyl-alkylcarbamates, leur preparation et leur application en therapeutique
FR2860514A1 (fr) * 2003-10-03 2005-04-08 Sanofi Synthelabo Derives d'arylalkylcarbamates, leur preparation et leur application en therapeutique
FR2866886B1 (fr) * 2004-02-26 2007-08-31 Sanofi Synthelabo Derives d'aryl-et d'heteroaryl-akylcarbamates, leur preparation et leur application en therapeutique

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CN102369200B (zh) * 2009-02-05 2015-05-20 赛诺菲 5元杂环化合物的氮杂螺烷基-烷基氨基甲酸酯衍生物、其制备方法和其治疗用途
CN102459232A (zh) * 2009-05-12 2012-05-16 赛诺菲 7-氮杂-螺[3.5]壬烷-7-甲酸酯衍生物、其制备及其治疗用途
CN102459232B (zh) * 2009-05-12 2014-05-07 赛诺菲 7-氮杂-螺[3.5]壬烷-7-甲酸酯衍生物、其制备及其治疗用途

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IL177534A0 (en) 2006-12-10
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DK1720550T3 (da) 2009-08-10
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JP4796046B2 (ja) 2011-10-19
RU2384569C2 (ru) 2010-03-20
PL1720550T3 (pl) 2009-09-30
RU2006134025A (ru) 2008-04-10
DE602005013923D1 (de) 2009-05-28
CY1109231T1 (el) 2014-07-02
US7781590B2 (en) 2010-08-24
US20070021403A1 (en) 2007-01-25
FR2866885B1 (fr) 2007-08-31
ZA200606964B (en) 2008-01-30
EP1720550B1 (fr) 2009-04-15
PT1720550E (pt) 2009-06-04

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